ZA200403684B - Macrolides. - Google Patents

Macrolides.

Info

Publication number
ZA200403684B
ZA200403684B ZA200403684A ZA200403684A ZA200403684B ZA 200403684 B ZA200403684 B ZA 200403684B ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 B ZA200403684 B ZA 200403684B
Authority
ZA
South Africa
Prior art keywords
macrolides
Prior art date
Application number
ZA200403684A
Other languages
English (en)
Inventor
Sulejman Alihodzic
Andrea Berdik
Stefano Biondi
Federica Damiani
Miljenko Dumic
Antun Hutinec
Sergio Luciuro
Zorica Marusic-Istuk
Alfredo Paio
Anna Quaglia
Vlado Stimac
Daniele Andreotti
Ilaria Bientinesi
Manuela Ciraco
Marko Djerek
Vesna Erakovic
Gorjana Lazarevski
Natasa Marsic
Stjepan Mutak
Drazen Pavlovic
Wolfgang Schoenfeld
Jessica Tibasco
Original Assignee
Glaxo Group Ltd
Pliva Istrazivacki Inst D O O
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Pliva Istrazivacki Inst D O O filed Critical Glaxo Group Ltd
Publication of ZA200403684B publication Critical patent/ZA200403684B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
ZA200403684A 2001-11-14 2004-05-13 Macrolides. ZA200403684B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0127349.9A GB0127349D0 (en) 2001-11-14 2001-11-14 Macrolides

Publications (1)

Publication Number Publication Date
ZA200403684B true ZA200403684B (en) 2005-09-13

Family

ID=9925777

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200403684A ZA200403684B (en) 2001-11-14 2004-05-13 Macrolides.

Country Status (20)

Country Link
US (1) US7202221B2 (cg-RX-API-DMAC7.html)
EP (1) EP1453846B1 (cg-RX-API-DMAC7.html)
JP (1) JP2005515978A (cg-RX-API-DMAC7.html)
CN (1) CN1307194C (cg-RX-API-DMAC7.html)
AR (1) AR037371A1 (cg-RX-API-DMAC7.html)
AT (1) ATE362479T1 (cg-RX-API-DMAC7.html)
BR (1) BR0214132A (cg-RX-API-DMAC7.html)
CA (1) CA2466975A1 (cg-RX-API-DMAC7.html)
DE (1) DE60220180T2 (cg-RX-API-DMAC7.html)
EA (1) EA007433B1 (cg-RX-API-DMAC7.html)
ES (1) ES2287332T3 (cg-RX-API-DMAC7.html)
GB (1) GB0127349D0 (cg-RX-API-DMAC7.html)
HR (1) HRP20040433A2 (cg-RX-API-DMAC7.html)
HU (1) HUP0402225A3 (cg-RX-API-DMAC7.html)
IL (1) IL161710A0 (cg-RX-API-DMAC7.html)
PL (1) PL371472A1 (cg-RX-API-DMAC7.html)
RS (1) RS41904A (cg-RX-API-DMAC7.html)
UA (1) UA77210C2 (cg-RX-API-DMAC7.html)
WO (1) WO2003042228A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200403684B (cg-RX-API-DMAC7.html)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US7135573B2 (en) 2002-05-13 2006-11-14 Enanta Pharmaceuticals, Inc. Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US7910558B2 (en) 2002-05-13 2011-03-22 Enanta Pharmaceuticals, Inc. Bridged macrocyclic compounds and processes for the preparation thereof
US7022679B2 (en) 2002-05-13 2006-04-04 Enanta Pharmaceuticals, Inc. Processes for the preparation of 6-11 bicyclic erythromycin derivatives
US6764998B1 (en) 2003-06-18 2004-07-20 Enanta Pharmaceuticals, Inc. 6,11-4C-bicyclic 9a-azalide derivatives
KR20040107525A (ko) * 2002-05-14 2004-12-20 더 리전트 오브 더 유니버시티 오브 캘리포니아 치환된 퀴놀론 카르복실산, 이들의 유도체, 그의 작용부위 및 용도
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
GB0225384D0 (en) 2002-10-31 2002-12-11 Glaxo Group Ltd Novel compounds
US6645941B1 (en) 2003-03-26 2003-11-11 Enanta Pharmaceuticals, Inc. 6,11-3C-bicyclic 9a-azalide derivatives
ATE348837T1 (de) * 2003-05-13 2007-01-15 Glaxo Group Ltd Neue 14- und 15-gliedrige ringverbindungen
GB0310980D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310984D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310979D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310986D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
WO2005030227A1 (en) 2003-09-23 2005-04-07 Enanta Pharmaceuticals, Inc. 9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
WO2005070113A2 (en) 2004-01-09 2005-08-04 Enanta Pharmaceuticals, Inc. 9n-substituted 6-11 bicyclic erythromycin derivatives
US8202843B2 (en) 2004-02-27 2012-06-19 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
EP1756134A1 (en) * 2004-05-06 2007-02-28 GlaxoSmithKline istrazivacki centar Zagreb d.o.o. Carbamate linked macrolides useful for the treatment of microbial infections
JP2007536371A (ja) * 2004-05-06 2007-12-13 グラクソスミスクライン・イストラジヴァッキ・センタル・ザグレブ・ドルズバ・ゼー・オメイェノ・オドゴヴォルノスティオ 微生物感染症の治療に有用なエステル結合マクロライド
WO2006047167A2 (en) * 2004-10-21 2006-05-04 Janssen Pharmaceutica, N.V. 9 alkyl and 9 alkylidenyl 6-0 alkyl-11, 12 carbamate ketolide antimicrobials
GB0424959D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424951D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424958D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424961D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
WO2008017696A1 (en) * 2006-08-09 2008-02-14 Basilea Pharmaceutica Ag New macrolides useful against inflammatory and allergic disseases
CN101541331A (zh) 2006-08-24 2009-09-23 沃克哈特研究中心 具有抗微生物活性的新颖大环内酯和酮内酯
KR101617897B1 (ko) 2008-02-08 2016-05-03 바실리어 파마슈티카 아게 신규 마크로라이드 및 그의 용도
EP2435460B1 (en) 2009-05-27 2015-01-07 Wockhardt Limited Ketolide compounds having antimicrobial activity
CN103384676B (zh) 2010-12-09 2016-02-03 沃克哈特有限公司 酮内酯化合物
CA2826174A1 (en) * 2011-01-31 2012-08-09 Meiji Seika Pharma Co., Ltd. Novel macrolide derivative
CN103619849B (zh) 2011-03-01 2016-05-25 沃克哈特有限公司 酮内酯中间体的制备方法
CN119060110A (zh) * 2023-05-30 2024-12-03 北京理工大学 一种红霉素衍生物及其制备方法和应用

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0126344A2 (en) 1983-05-20 1984-11-28 Abbott Laboratories Tripeptide esters of therapeutic agents
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
AU623764B2 (en) * 1989-03-28 1992-05-21 Abbott Laboratories Erythromycin derivatives
CA2064634C (en) * 1991-04-04 1998-08-04 James V. Heck 9-deoxo-8a-aza-8a-homoerythromycin a derivatives modified at the 4"- and8a-positions
BR9708929A (pt) 1996-05-07 1999-08-03 Abbott Lab Composto composição farmacêutica e processos para controlar uma infecção bacteriana em um mamífero e para preparar compostos de macrólidos
EP0895999A1 (en) * 1997-08-06 1999-02-10 Pfizer Products Inc. C-4" substituted macrolide antibiotics
US6262030B1 (en) * 1998-11-03 2001-07-17 Pfizer Inc. Erythromycin derivatives
EP1180110A1 (en) 1999-05-24 2002-02-20 Pfizer Products Inc. 13-methyl-erythromycin derivatives
WO2001014397A1 (en) 1999-08-24 2001-03-01 Abbott Laboratories 9a-azalides with antibacterial activity
US6946446B2 (en) * 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
WO2001063539A2 (en) 2000-02-24 2001-08-30 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
JP2002173498A (ja) 2000-09-27 2002-06-21 Hokuriku Seiyaku Co Ltd エリスロマイシン誘導体
GB0025688D0 (en) * 2000-10-19 2000-12-06 Glaxo Group Ltd Macrolides

Also Published As

Publication number Publication date
IL161710A0 (en) 2004-09-27
UA77210C2 (en) 2006-11-15
RS41904A (sr) 2006-10-27
GB0127349D0 (en) 2002-01-02
CA2466975A1 (en) 2003-05-22
AR037371A1 (es) 2004-11-03
ES2287332T3 (es) 2007-12-16
EP1453846A1 (en) 2004-09-08
DE60220180D1 (de) 2007-06-28
HUP0402225A3 (en) 2006-01-30
HUP0402225A2 (hu) 2005-02-28
EA007433B1 (ru) 2006-10-27
EA200400536A1 (ru) 2004-12-30
JP2005515978A (ja) 2005-06-02
CN1612888A (zh) 2005-05-04
CN1307194C (zh) 2007-03-28
PL371472A1 (en) 2005-06-13
HRP20040433A2 (en) 2005-04-30
DE60220180T2 (de) 2008-01-17
BR0214132A (pt) 2004-09-14
ATE362479T1 (de) 2007-06-15
US7202221B2 (en) 2007-04-10
US20050080025A1 (en) 2005-04-14
EP1453846B1 (en) 2007-05-16
WO2003042228A1 (en) 2003-05-22

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