EE200100613A - 13-metüülerütromütsiini derivaadid - Google Patents

13-metüülerütromütsiini derivaadid

Info

Publication number
EE200100613A
EE200100613A EEP200100613A EEP200100613A EE200100613A EE 200100613 A EE200100613 A EE 200100613A EE P200100613 A EEP200100613 A EE P200100613A EE P200100613 A EEP200100613 A EE P200100613A EE 200100613 A EE200100613 A EE 200100613A
Authority
EE
Estonia
Prior art keywords
methylerythromycin
derivatives
methylerythromycin derivatives
Prior art date
Application number
EEP200100613A
Other languages
English (en)
Inventor
Philip Dirlam John
Kaneko Takushi
Alastair Irvine Mcarthur Hamish
Su Wei-Guo
Wu Yong-Jin
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200100613A publication Critical patent/EE200100613A/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
EEP200100613A 1999-05-24 2000-04-25 13-metüülerütromütsiini derivaadid EE200100613A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13546899P 1999-05-24 1999-05-24
PCT/IB2000/000502 WO2000071557A1 (en) 1999-05-24 2000-04-25 13-methyl-erythromycin derivatives

Publications (1)

Publication Number Publication Date
EE200100613A true EE200100613A (et) 2003-02-17

Family

ID=22468240

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100613A EE200100613A (et) 1999-05-24 2000-04-25 13-metüülerütromütsiini derivaadid

Country Status (32)

Country Link
US (2) US20030100518A1 (et)
EP (1) EP1180110A1 (et)
JP (1) JP2003500414A (et)
KR (1) KR20020016799A (et)
CN (1) CN1351608A (et)
AP (1) AP2001002302A0 (et)
AR (1) AR020032A1 (et)
AU (1) AU3832100A (et)
BG (1) BG106127A (et)
BR (1) BR0010938A (et)
CA (1) CA2373117C (et)
CZ (1) CZ20013733A3 (et)
DZ (1) DZ3045A1 (et)
EA (1) EA200100983A1 (et)
EE (1) EE200100613A (et)
HK (1) HK1045523A1 (et)
HR (1) HRP20010866A2 (et)
HU (1) HUP0201516A3 (et)
IL (1) IL145739A0 (et)
IS (1) IS6128A (et)
MA (1) MA26740A1 (et)
NO (1) NO20015172L (et)
OA (1) OA11945A (et)
PA (1) PA8495101A1 (et)
PE (1) PE20010171A1 (et)
PL (1) PL352720A1 (et)
SK (1) SK15162001A3 (et)
TN (1) TNSN00108A1 (et)
TR (1) TR200103395T2 (et)
UY (1) UY26161A1 (et)
WO (1) WO2000071557A1 (et)
ZA (1) ZA200109595B (et)

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Publication number Priority date Publication date Assignee Title
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AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
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US6514944B2 (en) 1999-04-16 2003-02-04 Kosan Biosciences, Inc. Macrolide antiinfective agents
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US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6399582B1 (en) 1999-04-16 2002-06-04 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
IL145739A0 (en) 1999-05-24 2002-07-25 Pfizer Prod Inc 13-methyl-erythromycin derivatives
DE60104240T2 (de) 2000-06-30 2005-08-04 Pfizer Products Inc., Groton Makrolid-Antibiotika
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CN101568343A (zh) 2006-06-12 2009-10-28 雷蒙特亚特特拉维夫大学有限公司 用于治疗癌症的方法
CN101175322B (zh) * 2007-11-16 2010-12-15 华为技术有限公司 一种小区选择的方法
KR101043637B1 (ko) * 2009-07-13 2011-06-24 태석정공 주식회사 휴대용 듀얼 모니터의 카메라 모듈 결합구조
AR085286A1 (es) 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd Derivado de macrolido sustituido en la posicion c-4
BR112015015075A2 (pt) 2012-12-24 2019-01-15 Univ Ramot agentes para tratar doenças genéticas resultantes de mutações sem sentido e métodos para identificar as mesmas.
MX377459B (es) 2013-04-04 2025-03-10 Harvard College Macrolidos y metodos para su preparacion y uso.
WO2016057798A1 (en) 2014-10-08 2016-04-14 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
CN107530365A (zh) 2015-03-25 2018-01-02 哈佛大学的校长及成员们 具有修饰的脱氧糖胺糖的大环内酯及其用途

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Also Published As

Publication number Publication date
EP1180110A1 (en) 2002-02-20
CA2373117A1 (en) 2000-11-30
US6777543B2 (en) 2004-08-17
KR20020016799A (ko) 2002-03-06
CZ20013733A3 (cs) 2002-11-13
NO20015172D0 (no) 2001-10-23
CA2373117C (en) 2006-02-28
WO2000071557A1 (en) 2000-11-30
HUP0201516A2 (en) 2002-08-28
ZA200109595B (en) 2003-05-28
AR020032A1 (es) 2002-03-27
TNSN00108A1 (fr) 2002-05-30
PE20010171A1 (es) 2001-02-10
HRP20010866A2 (en) 2003-06-30
HK1045523A1 (zh) 2002-11-29
HUP0201516A3 (en) 2003-03-28
EA200100983A1 (ru) 2002-10-31
BG106127A (bg) 2002-05-31
DZ3045A1 (fr) 2004-03-27
SK15162001A3 (sk) 2003-02-04
IS6128A (is) 2001-10-26
US20030229031A1 (en) 2003-12-11
BR0010938A (pt) 2002-03-19
AU3832100A (en) 2000-12-12
PL352720A1 (en) 2003-09-08
MA26740A1 (fr) 2004-12-20
PA8495101A1 (es) 2002-08-26
UY26161A1 (es) 2000-12-29
US20030100518A1 (en) 2003-05-29
AP2001002302A0 (en) 2001-10-25
NO20015172L (no) 2002-01-23
CN1351608A (zh) 2002-05-29
OA11945A (en) 2006-04-13
JP2003500414A (ja) 2003-01-07
IL145739A0 (en) 2002-07-25
TR200103395T2 (tr) 2002-04-22

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