TNSN00108A1 - Derives d'erythromycine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant - Google Patents

Derives d'erythromycine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Info

Publication number
TNSN00108A1
TNSN00108A1 TNTNSN00108A TNSN00108A TNSN00108A1 TN SN00108 A1 TNSN00108 A1 TN SN00108A1 TN TNSN00108 A TNTNSN00108 A TN TNSN00108A TN SN00108 A TNSN00108 A TN SN00108A TN SN00108 A1 TNSN00108 A1 TN SN00108A1
Authority
TN
Tunisia
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
erythromycin derivatives
novel erythromycin
Prior art date
Application number
TNTNSN00108A
Other languages
English (en)
Inventor
Su Wei-Guo
Philip Dirlam John
Alastair Irvine Mcarthur Hamish
Wu Yong-Jin
Kaneko Takushi
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN00108A1 publication Critical patent/TNSN00108A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

L’INVENTION CONCERNE DES COMPOSES DE FORMULE 1 : DANS LAQUELLE R1, R2, R3, R4, R5, R17, Rf, A , X ET Y REPRESENTENT DIVERS RADICAUX. ELLE CONCERNE EGALEMENT UN PROCEDE POUR LEUR PREPARATION ET DES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT. APPLICATION : UTILISATION DE CES COMPOSES ET COMPOSITIONS DANS LE TRAITEMENT D’INFECTIONS.
TNTNSN00108A 1999-05-24 2000-05-23 Derives d'erythromycine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant TNSN00108A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13546899P 1999-05-24 1999-05-24

Publications (1)

Publication Number Publication Date
TNSN00108A1 true TNSN00108A1 (fr) 2002-05-30

Family

ID=22468240

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN00108A TNSN00108A1 (fr) 1999-05-24 2000-05-23 Derives d'erythromycine nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant

Country Status (32)

Country Link
US (2) US20030100518A1 (fr)
EP (1) EP1180110A1 (fr)
JP (1) JP2003500414A (fr)
KR (1) KR20020016799A (fr)
CN (1) CN1351608A (fr)
AP (1) AP2001002302A0 (fr)
AR (1) AR020032A1 (fr)
AU (1) AU3832100A (fr)
BG (1) BG106127A (fr)
BR (1) BR0010938A (fr)
CA (1) CA2373117C (fr)
CZ (1) CZ20013733A3 (fr)
DZ (1) DZ3045A1 (fr)
EA (1) EA200100983A1 (fr)
EE (1) EE200100613A (fr)
HK (1) HK1045523A1 (fr)
HR (1) HRP20010866A2 (fr)
HU (1) HUP0201516A3 (fr)
IL (1) IL145739A0 (fr)
IS (1) IS6128A (fr)
MA (1) MA26740A1 (fr)
NO (1) NO20015172L (fr)
OA (1) OA11945A (fr)
PA (1) PA8495101A1 (fr)
PE (1) PE20010171A1 (fr)
PL (1) PL352720A1 (fr)
SK (1) SK15162001A3 (fr)
TN (1) TNSN00108A1 (fr)
TR (1) TR200103395T2 (fr)
UY (1) UY26161A1 (fr)
WO (1) WO2000071557A1 (fr)
ZA (1) ZA200109595B (fr)

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AP2007004026A0 (en) 2004-12-21 2007-06-30 Pfizer Prod Inc Macrolides
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CN101175322B (zh) * 2007-11-16 2010-12-15 华为技术有限公司 一种小区选择的方法
KR101043637B1 (ko) * 2009-07-13 2011-06-24 태석정공 주식회사 휴대용 듀얼 모니터의 카메라 모듈 결합구조
AR085286A1 (es) 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd Derivado de macrolido sustituido en la posicion c-4
EP2934548A2 (fr) 2012-12-24 2015-10-28 Ramot at Tel-Aviv University Ltd Agents permettant de traiter des maladies génétiques résultant de mutations non-sens et leurs procédés d'identification
EP2988597B1 (fr) 2013-04-04 2022-06-08 President and Fellows of Harvard College Macrolides et leurs procédés de préparation et d'utilisation
JP2017531663A (ja) 2014-10-08 2017-10-26 プレジデント アンド フェローズ オブ ハーバード カレッジ １４員ケトライドならびにそれらの調製および使用の方法
EP3273969A4 (fr) 2015-03-25 2018-11-21 President and Fellows of Harvard College Macrolides à sucres modifiés de type désosamine et utilisations de ceux-ci

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Also Published As

Publication number Publication date
HUP0201516A2 (en) 2002-08-28
AP2001002302A0 (en) 2001-10-25
PL352720A1 (en) 2003-09-08
DZ3045A1 (fr) 2004-03-27
AR020032A1 (es) 2002-03-27
HK1045523A1 (zh) 2002-11-29
WO2000071557A1 (fr) 2000-11-30
US20030100518A1 (en) 2003-05-29
BG106127A (bg) 2002-05-31
JP2003500414A (ja) 2003-01-07
HUP0201516A3 (en) 2003-03-28
SK15162001A3 (sk) 2003-02-04
KR20020016799A (ko) 2002-03-06
NO20015172D0 (no) 2001-10-23
NO20015172L (no) 2002-01-23
EA200100983A1 (ru) 2002-10-31
EP1180110A1 (fr) 2002-02-20
IL145739A0 (en) 2002-07-25
MA26740A1 (fr) 2004-12-20
US6777543B2 (en) 2004-08-17
ZA200109595B (en) 2003-05-28
TR200103395T2 (tr) 2002-04-22
CN1351608A (zh) 2002-05-29
EE200100613A (et) 2003-02-17
UY26161A1 (es) 2000-12-29
PA8495101A1 (es) 2002-08-26
HRP20010866A2 (en) 2003-06-30
IS6128A (is) 2001-10-26
CA2373117C (fr) 2006-02-28
CA2373117A1 (fr) 2000-11-30
CZ20013733A3 (cs) 2002-11-13
AU3832100A (en) 2000-12-12
PE20010171A1 (es) 2001-02-10
US20030229031A1 (en) 2003-12-11
OA11945A (en) 2006-04-13
BR0010938A (pt) 2002-03-19

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