ZA200209520B - Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. - Google Patents
Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. Download PDFInfo
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- ZA200209520B ZA200209520B ZA200209520A ZA200209520A ZA200209520B ZA 200209520 B ZA200209520 B ZA 200209520B ZA 200209520 A ZA200209520 A ZA 200209520A ZA 200209520 A ZA200209520 A ZA 200209520A ZA 200209520 B ZA200209520 B ZA 200209520B
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- South Africa
- Prior art keywords
- microemulsion
- surfactant
- biologically active
- preparation
- days
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- 238000013268 sustained release Methods 0.000 title claims description 19
- 239000012730 sustained-release form Substances 0.000 title claims description 19
- 238000007911 parenteral administration Methods 0.000 title claims description 9
- 150000002433 hydrophilic molecules Chemical class 0.000 title claims description 3
- 239000008194 pharmaceutical composition Substances 0.000 title description 5
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Dispersion Chemistry (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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IT2000MI001173A IT1318539B1 (it) | 2000-05-26 | 2000-05-26 | Composizioni farmaceutiche a rilascio prolungato per lasomministrazione parenterale di sostanze idrofile biologicamente |
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ZA200209520B true ZA200209520B (en) | 2003-11-24 |
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ZA200209520A ZA200209520B (en) | 2000-05-26 | 2002-11-22 | Sustained release pharmaceutical compositions for parenteral administration of hydrophilic compounds. |
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US (1) | US7157099B2 (pt) |
EP (1) | EP1283700B1 (pt) |
JP (1) | JP4954423B2 (pt) |
KR (1) | KR100802625B1 (pt) |
CN (1) | CN100479856C (pt) |
AT (1) | ATE321533T1 (pt) |
AU (2) | AU8178601A (pt) |
BR (1) | BRPI0111016B8 (pt) |
CA (1) | CA2409854C (pt) |
CY (1) | CY1105262T1 (pt) |
CZ (1) | CZ302059B6 (pt) |
DE (1) | DE60118395T2 (pt) |
DK (1) | DK1283700T3 (pt) |
ES (1) | ES2257428T3 (pt) |
HR (1) | HRP20020929A2 (pt) |
HU (1) | HU228926B1 (pt) |
IL (1) | IL153011A0 (pt) |
IT (1) | IT1318539B1 (pt) |
MX (1) | MXPA02011539A (pt) |
NO (1) | NO334880B1 (pt) |
PL (1) | PL203354B1 (pt) |
PT (1) | PT1283700E (pt) |
RU (1) | RU2272615C2 (pt) |
SI (1) | SI1283700T1 (pt) |
SK (1) | SK16552002A3 (pt) |
WO (1) | WO2001089479A2 (pt) |
YU (1) | YU88202A (pt) |
ZA (1) | ZA200209520B (pt) |
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EP0671937A4 (en) * | 1992-10-16 | 1996-09-18 | Smithkline Beecham Corp | COMPOSITIONS FOR PHARMACEUTICAL EMULSIONS. |
SE512663C2 (sv) * | 1997-10-23 | 2000-04-17 | Biogram Ab | Inkapslingsförfarande för aktiv substans i en bionedbrytbar polymer |
WO1999021533A2 (en) * | 1997-10-24 | 1999-05-06 | Neorx Corporation | Delivery vehicles for bioactive agents and uses thereof |
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