UY35370A - Moduladores benzoimidazol-2-il pirimidina del receptor de histamina h4 - Google Patents

Moduladores benzoimidazol-2-il pirimidina del receptor de histamina h4

Info

Publication number
UY35370A
UY35370A UY0001035370A UY35370A UY35370A UY 35370 A UY35370 A UY 35370A UY 0001035370 A UY0001035370 A UY 0001035370A UY 35370 A UY35370 A UY 35370A UY 35370 A UY35370 A UY 35370A
Authority
UY
Uruguay
Prior art keywords
benzoimidazol
receptor
histamine
modulators
pyrimidine
Prior art date
Application number
UY0001035370A
Other languages
English (en)
Inventor
Conza Matteo
Magali B Hickey
Horns Stefan
Lochner Susanne
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of UY35370A publication Critical patent/UY35370A/es

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    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C30B7/00Single-crystal growth from solutions using solvents which are liquid at normal temperature, e.g. aqueous solutions
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Abstract

Benzoimidazol-2-il pirimidinas, métodos de purifi cación de estas, y composiciones farmacéuticas y métodos para el tratamiento de estados patológicos , trastornos y afecciones mediados por la activid ad del receptor H4 que incluyen alergia, asma, en fermedades autoinmunes y prurito.
UY0001035370A 2013-03-06 2014-03-06 Moduladores benzoimidazol-2-il pirimidina del receptor de histamina h4 UY35370A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361773706P 2013-03-06 2013-03-06
US201361776260P 2013-03-11 2013-03-11
US201361784909P 2013-03-14 2013-03-14

Publications (1)

Publication Number Publication Date
UY35370A true UY35370A (es) 2014-09-30

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UY0001035370A UY35370A (es) 2013-03-06 2014-03-06 Moduladores benzoimidazol-2-il pirimidina del receptor de histamina h4

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US (4) US8859575B2 (es)
EP (2) EP3660011A1 (es)
JP (1) JP6471103B2 (es)
KR (1) KR102230383B1 (es)
CN (1) CN105025898B (es)
AU (1) AU2014225675B2 (es)
BR (1) BR112015021463A8 (es)
CA (1) CA2903737C (es)
CL (1) CL2015002434A1 (es)
CR (1) CR20150435A (es)
CY (1) CY1122545T1 (es)
DK (1) DK2964229T3 (es)
DO (1) DOP2016000027A (es)
EA (1) EA201591648A1 (es)
ES (1) ES2773543T3 (es)
GT (1) GT201500243A (es)
HK (1) HK1218513A1 (es)
HR (1) HRP20200253T1 (es)
HU (1) HUE047681T2 (es)
IL (1) IL240247B (es)
JO (1) JO3516B1 (es)
LT (1) LT2964229T (es)
MX (1) MX2015011688A (es)
MY (1) MY180726A (es)
NZ (1) NZ710640A (es)
PE (1) PE20151536A1 (es)
PH (1) PH12015501731A1 (es)
PL (1) PL2964229T3 (es)
PT (1) PT2964229T (es)
RS (1) RS59909B1 (es)
SA (1) SA515360981B1 (es)
SG (1) SG11201507117XA (es)
SI (1) SI2964229T1 (es)
TW (1) TWI617554B (es)
UA (1) UA118754C2 (es)
UY (1) UY35370A (es)
WO (1) WO2014138368A1 (es)
ZA (1) ZA201507351B (es)

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EA016264B1 (ru) 2006-03-31 2012-03-30 Янссен Фармацевтика Н.В. Бензоимидазол-2-илпиримидины и пиразины в качестве модуляторов рецептора гистамина н
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JO3509B1 (ar) 2013-03-14 2020-07-05 Janssen Pharmaceutica Nv معدلات p2x7
JO3773B1 (ar) 2013-03-14 2021-01-31 Janssen Pharmaceutica Nv معدلات p2x7
US9040534B2 (en) 2013-03-14 2015-05-26 Janssen Pharmaceutica Nv [1,2,4]triazolo[4,3-a]pyrazines as P2X7 modulators
US9096596B2 (en) 2013-03-14 2015-08-04 Janssen Pharmaceutica Nv P2X7 modulators
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