UY24938A1 - Derivados de pirimidina y procedimientos para la preparación de los mismos - Google Patents

Derivados de pirimidina y procedimientos para la preparación de los mismos

Info

Publication number
UY24938A1
UY24938A1 UY24938A UY24938A UY24938A1 UY 24938 A1 UY24938 A1 UY 24938A1 UY 24938 A UY24938 A UY 24938A UY 24938 A UY24938 A UY 24938A UY 24938 A1 UY24938 A1 UY 24938A1
Authority
UY
Uruguay
Prior art keywords
pyrimidine
methyl
procedures
preparation
same
Prior art date
Application number
UY24938A
Other languages
English (en)
Spanish (es)
Inventor
Man Soon Hwang
Woo Jeon Shim
Song Jin Lee
Keun Seog Song
Seung Kyu Lee
Wook Lee Jong
Original Assignee
Yuhan Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yuhan Corp filed Critical Yuhan Corp
Publication of UY24938A1 publication Critical patent/UY24938A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
UY24938A 1997-03-27 1998-03-26 Derivados de pirimidina y procedimientos para la preparación de los mismos UY24938A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR19970010863 1997-03-27
KR19970010862 1997-03-27

Publications (1)

Publication Number Publication Date
UY24938A1 true UY24938A1 (es) 2001-01-31

Family

ID=26632616

Family Applications (1)

Application Number Title Priority Date Filing Date
UY24938A UY24938A1 (es) 1997-03-27 1998-03-26 Derivados de pirimidina y procedimientos para la preparación de los mismos

Country Status (21)

Country Link
US (1) US6352993B1 (en:Method)
EP (1) EP1015444B1 (en:Method)
JP (1) JP3176379B2 (en:Method)
KR (1) KR100278857B1 (en:Method)
CN (1) CN1118464C (en:Method)
AR (1) AR012181A1 (en:Method)
AT (1) ATE241613T1 (en:Method)
AU (1) AU720385B2 (en:Method)
BR (1) BR9808070A (en:Method)
CA (1) CA2284795C (en:Method)
DE (1) DE69815126T2 (en:Method)
DK (1) DK1015444T3 (en:Method)
ES (1) ES2200324T3 (en:Method)
HU (1) HUP0000851A3 (en:Method)
IN (1) IN188411B (en:Method)
PT (1) PT1015444E (en:Method)
RU (1) RU2203894C2 (en:Method)
TR (1) TR199902383T2 (en:Method)
TW (1) TW542831B (en:Method)
UY (1) UY24938A1 (en:Method)
WO (1) WO1998043968A1 (en:Method)

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WO2004012659A2 (en) 2002-08-01 2004-02-12 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
US20070161637A1 (en) * 2003-07-22 2007-07-12 Neurogen Corporation Substituted pyridin-2-ylamine analogues
JP4800216B2 (ja) * 2003-10-24 2011-10-26 エグゼリクシス， インコーポレイテッド ｐ７０Ｓ６キナーゼモジュレーターおよび使用方法
CN1874772A (zh) 2003-11-03 2006-12-06 阿斯利康(瑞典)有限公司 治疗隐匿性胃食管反流的咪唑并[1,2－a]吡啶衍生物
KR101122376B1 (ko) * 2005-03-09 2012-03-26 주식회사유한양행 신규의 5,6-다이메틸피리미딘 유도체 및 그의 제조방법
JP2009511548A (ja) * 2005-10-14 2009-03-19 ノイロサーチ アクティーゼルスカブ 新規ピリミジン−２，４−ジアミン誘導体及び小コンダクタンスのカルシウム依存性カリウムチャネルのモジュレーターとしてのこれらの使用
JP4946482B2 (ja) 2007-02-08 2012-06-06 船井電機株式会社 緩衝用梱包材及びｔｖ受像機の緩衝用梱包材
US8367684B2 (en) * 2007-06-13 2013-02-05 Valeant Pharmaceuticals International Derivatives of 4-(N-azacycloalkyl) anilides as potassium channel modulators
CA2732950C (en) 2008-08-05 2013-10-01 Daiichi Sankyo Company, Limited Imidazopyridin-2-one derivatives
GB0908394D0 (en) 2009-05-15 2009-06-24 Univ Leuven Kath Novel viral replication inhibitors
GB0913636D0 (en) 2009-08-05 2009-09-16 Univ Leuven Kath Novel viral replication inhibitors
WO2012065963A2 (en) 2010-11-15 2012-05-24 Katholieke Universiteit Leuven Novel antiviral compounds
CN103402997B (zh) 2011-02-25 2015-08-26 柳韩洋行 二氨基嘧啶衍生物及其制备方法
CA2864825C (en) * 2012-02-17 2021-01-26 Abbvie Inc. Diaminopyrimidines useful as inhibitors of the human respiratory syncytial virus (rsv)
US9309271B2 (en) 2012-05-29 2016-04-12 Momentive Performance Materials Gmbh Preparation of isocyanato silanes
DK2922828T3 (da) 2012-11-21 2020-08-31 Ptc Therapeutics Inc 4,6-diamino-pyrimidin-derivater som bmi-1-inhibitorer til at behandle cancer
US10035801B2 (en) 2013-03-13 2018-07-31 Genentech, Inc. Pyrazolo compounds and uses thereof
EA034866B1 (ru) 2013-08-30 2020-03-31 ПиТиСи ТЕРАПЬЮТИКС, ИНК. Замещенные пиримидиновые ингибиторы bmi-1
CN104903312B (zh) * 2013-10-07 2019-01-29 卡德门企业有限公司 Rho激酶抑制剂
EP3071553A4 (en) 2013-11-21 2017-08-02 PTC Therapeutics, Inc. Substituted pyridine and pyrazine bmi-1 inhibitors
US10370360B2 (en) 2014-10-22 2019-08-06 The Board Of Regents Of The University Of Texas System Small-molecule inhibitors targeting discoidin domain receptor 1 and uses thereof
CN105669642B (zh) * 2014-11-19 2020-06-09 江苏天士力帝益药业有限公司 一种盐酸洛氟普啶的制备方法
DK3397622T3 (en) * 2016-01-04 2022-06-07 ObsEva SA Co-administration af alpha-aminoester af hydroxypropylthiazolidincarboxamid-derivat og et tokolytisk middel
EP3606915A1 (de) * 2017-04-05 2020-02-12 Bayer CropScience Aktiengesellschaft 2-amino-5-oxyalkyl-pyrimidinderivate und deren verwendung zur bekämpfung unerwünschten pflanzenwachstums
BR112021002630A2 (pt) 2018-08-17 2021-05-11 Ptc Therapeutics, Inc. método para tratar câncer pancreático
CN114685369B (zh) * 2022-05-17 2024-02-02 河南省科学院高新技术研究中心 一种利用离子液体制备1-甲基-1,2,3,4-四氢异喹啉的方法

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GB1182584A (en) 1966-03-31 1970-02-25 Ici Ltd Pyrimidine derivates and the use thereof as fungicides
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JPH09501918A (ja) * 1993-08-12 1997-02-25 アストラ・アクチエボラーグ 酸化窒素合成酵素活性を有するアミジン誘導体
DK0640599T3 (da) 1993-08-26 1998-09-28 Ono Pharmaceutical Co 4-Aminopyrimidin-derivater
RU2153494C2 (ru) 1993-10-12 2000-07-27 Дзе Дюпон Мерк Фармасьютикал Компани 1-n-алкил-n-арилпиримидинамины, способ лечения заболеваний, фармацевтическая композиция
EP0775120B1 (en) * 1994-08-13 2003-06-04 Yuhan Corporation Novel pyrimidine derivatives and processes for the preparation thereof
PT900214E (pt) * 1996-05-04 2002-03-28 Yuhan Corp Processo para a preparacao de derivados da pirimidina

Also Published As

Publication number Publication date
BR9808070A (pt) 2000-03-08
EP1015444B1 (en) 2003-05-28
CA2284795A1 (en) 1998-10-08
CA2284795C (en) 2004-01-20
US6352993B1 (en) 2002-03-05
ES2200324T3 (es) 2004-03-01
CN1251586A (zh) 2000-04-26
DE69815126T2 (de) 2004-04-08
KR19980080789A (ko) 1998-11-25
WO1998043968A1 (en) 1998-10-08
KR100278857B1 (ko) 2001-01-15
RU2203894C2 (ru) 2003-05-10
TW542831B (en) 2003-07-21
JP3176379B2 (ja) 2001-06-18
HK1026418A1 (en) 2000-12-15
HUP0000851A3 (en) 2002-04-29
HUP0000851A1 (hu) 2001-04-28
DK1015444T3 (da) 2003-08-18
IN188411B (en:Method) 2002-09-21
DE69815126D1 (de) 2003-07-03
PT1015444E (pt) 2003-10-31
AU6523998A (en) 1998-10-22
EP1015444A1 (en) 2000-07-05
TR199902383T2 (xx) 2000-06-21
JP2000513014A (ja) 2000-10-03
ATE241613T1 (de) 2003-06-15
AU720385B2 (en) 2000-06-01
AR012181A1 (es) 2000-09-27
CN1118464C (zh) 2003-08-20

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Legal Events

Date Code Title Description
VENC Patent expired

Effective date: 20180326