UA72039C2 - A method for the preparation of citalopram - Google Patents

A method for the preparation of citalopram Download PDF

Info

Publication number
UA72039C2
UA72039C2 UA2002118821A UA2002118821A UA72039C2 UA 72039 C2 UA72039 C2 UA 72039C2 UA 2002118821 A UA2002118821 A UA 2002118821A UA 2002118821 A UA2002118821 A UA 2002118821A UA 72039 C2 UA72039 C2 UA 72039C2
Authority
UA
Ukraine
Prior art keywords
formula
compound
differs
intermediate compound
interaction
Prior art date
Application number
UA2002118821A
Other languages
English (en)
Ukrainian (uk)
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of UA72039C2 publication Critical patent/UA72039C2/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
UA2002118821A 2000-05-12 2001-10-05 A method for the preparation of citalopram UA72039C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200000783 2000-05-12
PCT/DK2001/000333 WO2001085712A1 (en) 2000-05-12 2001-05-10 Method for the preparation of citalopram

Publications (1)

Publication Number Publication Date
UA72039C2 true UA72039C2 (en) 2005-01-17

Family

ID=8159493

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2002118821A UA72039C2 (en) 2000-05-12 2001-10-05 A method for the preparation of citalopram

Country Status (29)

Country Link
US (1) US6660873B2 (pl)
EP (1) EP1296970B1 (pl)
JP (1) JP2003532721A (pl)
CN (1) CN100422166C (pl)
AR (1) AR032455A1 (pl)
AT (1) ATE389645T1 (pl)
AU (2) AU5823901A (pl)
BG (1) BG65820B1 (pl)
BR (1) BR0110996A (pl)
CA (1) CA2408292C (pl)
CZ (1) CZ20024065A3 (pl)
DE (1) DE60133280T2 (pl)
DK (1) DK1296970T3 (pl)
EA (1) EA005674B1 (pl)
ES (1) ES2301541T3 (pl)
HR (1) HRP20020881A2 (pl)
HU (1) HUP0301942A2 (pl)
IL (2) IL152645A0 (pl)
IS (1) IS2586B (pl)
MX (1) MXPA02011125A (pl)
NO (1) NO327963B1 (pl)
NZ (1) NZ522475A (pl)
PL (1) PL358144A1 (pl)
PT (1) PT1296970E (pl)
SI (1) SI1296970T1 (pl)
SK (1) SK287035B6 (pl)
UA (1) UA72039C2 (pl)
WO (1) WO2001085712A1 (pl)
ZA (1) ZA200208973B (pl)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1173431T4 (da) 1999-04-14 2010-01-04 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IN192057B (pl) * 2001-07-19 2004-02-14 Ranbaxy Lab Ltd
WO2004085416A1 (en) * 2003-03-24 2004-10-07 Hetero Drugs Limited Novel crystalline forms of (s)-citalopram oxalate
AU2003278409A1 (en) * 2003-10-28 2005-05-19 Krishnaji Upadhye Bhargav Improved process for the manufacture of citalopram hydrobromide
US20050143350A1 (en) * 2003-11-19 2005-06-30 Seed John C. Combination drug therapy to treat obesity
ES2285972T1 (es) 2004-08-23 2007-12-01 Sun Pharmaceutical Industries Limited Procedimiento de fabricacion de citalopram y enantiomeros.

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143703A (pl) 1965-03-18
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
US5296507A (en) 1990-09-06 1994-03-22 H.Lundbeck A/S Treatment of cerbrovascular disorders
DE19626659A1 (de) 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
ES2148120T3 (es) 1997-07-08 2002-01-16 Lundbeck & Co As H Metodo para la preparacion de citalopram.
UA62985C2 (en) 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
EA002770B1 (ru) 1997-11-11 2002-08-29 Х.Лундбекк А/С Способ получения циталопрама
PL199423B1 (pl) 1998-10-20 2008-09-30 Lundbeck & Co As H Sposób wytwarzania citalopramu
IL143422A0 (en) 1998-12-23 2002-04-21 Lundbeck & Co As H Method for the preparation of 5-cyanophthalide
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
DK1173431T4 (da) 1999-04-14 2010-01-04 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991581A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991486A1 (it) 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
GB2360281B (en) 1999-10-25 2002-01-16 Lundbeck & Co As H Method for the preparation of citalopram
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
HUP0203635A3 (en) 1999-12-28 2005-02-28 Lundbeck & Co As H Method for the preparation of citalopram
PT1246813E (pt) 1999-12-30 2004-02-27 Lundbeck & Co As H Metodo para a preparacao de citalopram
CN1195749C (zh) 2000-01-14 2005-04-06 H.隆德贝克有限公司 制备5－氰基2－苯并[c]呋喃酮的方法
IT1317729B1 (it) 2000-01-18 2003-07-15 Norpharma S P A Procedimento per la preparazione della 5-carbossiftalide.
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010143A2 (en) 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
NL1017415C1 (nl) 2000-02-24 2001-05-18 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en) 2000-03-07 2000-04-26 Resolution Chemicals Limited Process for the preparation of citalopram
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
KR20020080481A (ko) 2000-03-13 2002-10-23 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
GB2357762B (en) 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
TR200202155T2 (tr) 2000-03-14 2002-12-23 H. Lundbeck A/S Sitalopramin preparasyon metodu
DE10190485T1 (de) 2000-03-16 2002-03-21 Lundbeck & Co As H Verfahren zur Herstellung von 5-Cyano-1-(4-fluorphenyl)-1,3-dihydroisobenzofuranen
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
CA2383963A1 (en) 2000-07-06 2002-01-17 Eva Bolzonella Method for the preparation of citalopram
CA2354877C (en) 2000-08-18 2006-05-02 H. Lundbeck A/S Method for the preparation of citalopram
WO2001045483A2 (en) 2000-12-22 2001-06-28 H. Lundbeck A/S Method for the preparation of pure citalopram
JP2003519121A (ja) 2000-12-28 2003-06-17 ハー・ルンドベック・アクチエゼルスカベット 純粋なシタロプラムの製造方法

Also Published As

Publication number Publication date
DE60133280T2 (de) 2009-04-16
US6660873B2 (en) 2003-12-09
BR0110996A (pt) 2003-03-18
CA2408292C (en) 2009-11-10
IL152645A (en) 2009-12-24
HK1056171A1 (zh) 2004-02-06
CN100422166C (zh) 2008-10-01
EA200201211A1 (ru) 2003-04-24
CA2408292A1 (en) 2001-11-15
NZ522475A (en) 2004-09-24
JP2003532721A (ja) 2003-11-05
CN1441795A (zh) 2003-09-10
ATE389645T1 (de) 2008-04-15
NO20025423L (no) 2002-11-12
WO2001085712A1 (en) 2001-11-15
DK1296970T3 (da) 2008-07-14
HUP0301942A2 (hu) 2003-09-29
EP1296970B1 (en) 2008-03-19
AU2001258239B2 (en) 2005-12-08
MXPA02011125A (es) 2003-03-10
AU5823901A (en) 2001-11-20
ES2301541T3 (es) 2008-07-01
NO20025423D0 (no) 2002-11-12
AR032455A1 (es) 2003-11-12
DE60133280D1 (de) 2008-04-30
CZ20024065A3 (cs) 2003-03-12
SI1296970T1 (sl) 2008-08-31
BG107349A (bg) 2003-09-30
EP1296970A1 (en) 2003-04-02
SK17542002A3 (sk) 2003-04-01
ZA200208973B (en) 2003-11-05
BG65820B1 (bg) 2010-01-29
SK287035B6 (sk) 2009-10-07
US20030134895A1 (en) 2003-07-17
IS2586B (is) 2010-02-15
NO327963B1 (no) 2009-10-26
IL152645A0 (en) 2003-06-24
HRP20020881A2 (en) 2004-12-31
IS6605A (is) 2002-10-31
PL358144A1 (pl) 2004-08-09
PT1296970E (pt) 2008-06-11
EA005674B1 (ru) 2005-04-28

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