TWI370121B - Process for the preparation of a 2-pyridylethylcarboxamide derivative - Google Patents

Process for the preparation of a 2-pyridylethylcarboxamide derivative

Info

Publication number
TWI370121B
TWI370121B TW094145400A TW94145400A TWI370121B TW I370121 B TWI370121 B TW I370121B TW 094145400 A TW094145400 A TW 094145400A TW 94145400 A TW94145400 A TW 94145400A TW I370121 B TWI370121 B TW I370121B
Authority
TW
Taiwan
Prior art keywords
preparation
derivative
pyridylethylcarboxamide derivative
general formula
pyridylethylcarboxamide
Prior art date
Application number
TW094145400A
Other languages
English (en)
Other versions
TW200637822A (en
Inventor
Frederic Lhermitte
Pierre-Yves Coqueron
Philippe Desbordes
Thomas Himmler
Original Assignee
Bayer Cropscience Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Sa filed Critical Bayer Cropscience Sa
Publication of TW200637822A publication Critical patent/TW200637822A/zh
Application granted granted Critical
Publication of TWI370121B publication Critical patent/TWI370121B/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/56—Amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/68—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/69—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
TW094145400A 2004-12-21 2005-12-20 Process for the preparation of a 2-pyridylethylcarboxamide derivative TWI370121B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04356203 2004-12-21

Publications (2)

Publication Number Publication Date
TW200637822A TW200637822A (en) 2006-11-01
TWI370121B true TWI370121B (en) 2012-08-11

Family

ID=34931762

Family Applications (2)

Application Number Title Priority Date Filing Date
TW100146039A TWI379826B (en) 2004-12-21 2005-12-20 Intermediate compound for the preparation of a 2-pyridylethylcarboxamide derivative
TW094145400A TWI370121B (en) 2004-12-21 2005-12-20 Process for the preparation of a 2-pyridylethylcarboxamide derivative

Family Applications Before (1)

Application Number Title Priority Date Filing Date
TW100146039A TWI379826B (en) 2004-12-21 2005-12-20 Intermediate compound for the preparation of a 2-pyridylethylcarboxamide derivative

Country Status (13)

Country Link
US (2) US7790901B2 (zh)
EP (1) EP1831169B1 (zh)
JP (2) JP4869251B2 (zh)
KR (1) KR101312816B1 (zh)
CN (1) CN101080391B (zh)
AT (1) ATE553083T1 (zh)
BR (1) BRPI0516905B1 (zh)
DK (1) DK1831169T3 (zh)
ES (1) ES2383903T3 (zh)
IL (2) IL183662A (zh)
MX (1) MX2007007105A (zh)
TW (2) TWI379826B (zh)
WO (1) WO2006067103A2 (zh)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2606728A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
AU2012331284B2 (en) * 2011-11-02 2016-06-30 Bayer Animal Health Gmbh Compounds with nematicidal activity
KR20140088532A (ko) 2011-11-02 2014-07-10 바이엘 인텔렉쳐 프로퍼티 게엠베하 살선충 활성을 갖는 화합물
EP2589292A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
EP2606727A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
EP2589294A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
CA2878247C (en) 2012-07-12 2021-01-19 Nissan Chemical Industries, Ltd. Oxime-substituted amide compound and pest control agent
CN103535354A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535362A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535353A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535355A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
UY35772A (es) 2013-10-14 2015-05-29 Bayer Cropscience Ag Nuevos compuestos plaguicidas
US10167250B2 (en) * 2014-06-16 2019-01-01 Srf Limited Process for the preparation of 2-(trihalomethyl) benzamide
KR101719565B1 (ko) * 2014-10-02 2017-03-24 한국화학연구원 광산화환원 촉매와 CF3SO2Cl을 사용한 알켄 화합물의 클로로트리플루오로메틸레이션 방법
EP3558945B1 (en) * 2016-12-21 2021-05-05 Bayer CropScience Aktiengesellschaft Process for the preparation of a n-[2-(2-pyridinyl)ethyl]carboxamide derivative
BR112021001395A2 (pt) * 2018-07-26 2021-04-27 Bayer Aktiengesellschaft forma cristalina de fluopiram
CN108822024B (zh) * 2018-08-28 2021-03-09 陕西恒润化学工业有限公司 一种氟吡菌酰胺及其合成方法
CN108752268A (zh) * 2018-08-28 2018-11-06 陕西恒润化学工业有限公司 一种2-（3-氯-5-三氟甲基吡啶）-丙二酸二甲酯及其合成方法
CN110437138B (zh) * 2019-08-12 2021-03-02 大连九信精细化工有限公司 一种氟吡菌酰胺的改进合成工艺
CN112979539B (zh) * 2021-05-17 2021-07-20 湖南速博生物技术有限公司 一种氟吡菌酰胺中间体的合成方法
CN113429338B (zh) * 2021-05-20 2023-05-02 陕西泰合利华工业有限公司 一种合成氟吡菌酰胺的方法
CN113620867B (zh) * 2021-09-03 2023-06-16 内蒙古蓝科生物科技有限公司 一种氟吡菌酰胺的合成方法
CN114195667A (zh) * 2021-11-30 2022-03-18 江西永通科技股份有限公司 一种邻三氟甲基苯甲酰胺的合成方法

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Publication number Priority date Publication date Assignee Title
DE1034644B (de) * 1956-09-26 1958-07-24 Bayer Ag Verfahren zur Herstellung von Acylaminomethyl-Verbindungen
JPS5363337A (en) * 1976-11-12 1978-06-06 Nippon Kayaku Co Ltd Benzamide derivs, process for their preparation and herbicides contg.the same as active constituents
ATE24504T1 (de) * 1981-03-19 1987-01-15 Ici Plc Amidderivate, verfahren zu ihrer herstellung, ihre verwendung als fungizide und pestizide, die sie enthalten.
DE4138026A1 (de) * 1991-11-19 1993-06-03 Bayer Ag Substituierte pyridin-4-carbonsaeureamide
PT1204323E (pt) * 1999-08-18 2004-11-30 Aventis Cropscience Gmbh Fungicidas
JP2001213869A (ja) * 2000-01-28 2001-08-07 Nippon Bayer Agrochem Co Ltd イソチアゾールカルボン酸誘導体および病害防除剤
US20060009461A1 (en) 2002-05-23 2006-01-12 Bhatia Pramila A Acetamides and benzamides that are useful in treating sexual dysfunction
US20040029887A1 (en) 2002-05-23 2004-02-12 Bhatia Pramila A. Acetamides and benzamides that are useful in treating sexual dysfunction
WO2003099266A2 (en) 2002-05-23 2003-12-04 Abbott Laboratories Acetamides and benzamides that are useful in treating sexual dysfunction
US20030232836A1 (en) 2002-05-23 2003-12-18 Stewart Andrew O. Acetamides and benzamides that are useful in treating sexual dysfunction
MXPA05001580A (es) * 2002-08-12 2005-04-25 Bayer Cropscience Sa Nuevos derivados de 2-piridiletilbenzamida.
EP1500651A1 (en) * 2003-07-25 2005-01-26 Bayer CropScience S.A. N-[2-(2-Pyridinyl)ethyl]benzamide compounds and their use as fungicides
EP1548007A1 (en) * 2003-12-19 2005-06-29 Bayer CropScience S.A. 2-Pyridinylethylcarboxamide derivatives and their use as fungicides
TWI368482B (en) * 2003-12-19 2012-07-21 Bayer Sas New 2-pyridinylethylbenzamide derivatives
EP1574511A1 (en) * 2004-03-03 2005-09-14 Bayer CropScience S.A. 2-Pyridinylethylcarboxamide derivatives and their use as fungicides

Also Published As

Publication number Publication date
US20100292485A1 (en) 2010-11-18
KR20070087668A (ko) 2007-08-28
JP5559745B2 (ja) 2014-07-23
ES2383903T3 (es) 2012-06-27
US20080086008A1 (en) 2008-04-10
WO2006067103A3 (en) 2006-11-16
KR101312816B1 (ko) 2013-09-27
IL183662A (en) 2012-06-28
EP1831169B1 (en) 2012-04-11
CN101080391B (zh) 2010-09-22
IL217962A0 (en) 2012-03-29
CN101080391A (zh) 2007-11-28
US8865908B2 (en) 2014-10-21
TWI379826B (en) 2012-12-21
DK1831169T3 (da) 2012-07-09
US7790901B2 (en) 2010-09-07
WO2006067103A2 (en) 2006-06-29
BRPI0516905A (pt) 2008-09-23
ATE553083T1 (de) 2012-04-15
JP4869251B2 (ja) 2012-02-08
IL183662A0 (en) 2007-09-20
JP2011236216A (ja) 2011-11-24
JP2008524307A (ja) 2008-07-10
MX2007007105A (es) 2007-08-08
IL217962A (en) 2015-02-26
TW201215594A (en) 2012-04-16
TW200637822A (en) 2006-11-01
EP1831169A2 (en) 2007-09-12
BRPI0516905B1 (pt) 2016-09-20

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