TR200100177T2 - Antifungal Aktiviteye sahip bir bileşimin oral farmasötik kompozisyonu ve bu kompozisyonun hazırlanış metodu. - Google Patents

Antifungal Aktiviteye sahip bir bileşimin oral farmasötik kompozisyonu ve bu kompozisyonun hazırlanış metodu.

Info

Publication number
TR200100177T2
TR200100177T2 TR2001/00177T TR200100177T TR200100177T2 TR 200100177 T2 TR200100177 T2 TR 200100177T2 TR 2001/00177 T TR2001/00177 T TR 2001/00177T TR 200100177 T TR200100177 T TR 200100177T TR 200100177 T2 TR200100177 T2 TR 200100177T2
Authority
TR
Turkey
Prior art keywords
composition
antifungal activity
oral pharmaceutical
preparation
coating
Prior art date
Application number
TR2001/00177T
Other languages
English (en)
Inventor
Carlos Picornell Darder
Original Assignee
Liconsa Liberacion Controlada De Sustancias Activas, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8304581&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR200100177(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Liconsa Liberacion Controlada De Sustancias Activas, S.A. filed Critical Liconsa Liberacion Controlada De Sustancias Activas, S.A.
Publication of TR200100177T2 publication Critical patent/TR200100177T2/tr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Abstract

Aktif madde olarak antifungal aktiviteye sahip bir bilesimden, 50 ila 600 um partikül büyüklügüne sahip hareketsiz bir çekirdek ve püskürtme islemi ile elde edilen tek bir tabakadan ve antifungal aktiviteye sahip bir bilesimden, hidrofili polimer ve iyonik olmayan yüzey aktif maddesinden olusan bir solüsyondan meydana gelen ve anilan aktif parçayi kapsayan bir kaplamadan olusan tablet seklinde bir oral farmasötik kompozisyon. Tüm süreç boyunca sabit bir kaplama hizinda antifungal madde, hidrofilik polimer ve iyonik olmayan yüzey aktif maddesinden olusan bir solüsyonun püskürütülmesi yolu ile 50 ila 600 um arasinda bir büyüklüge sahip hareketsiz çekirdeklerle tek kat olarak kaplama islemini ve ayni aparatta anilan kaplamanin tek adimli bir kurutma islemini kapsayan metot.
TR2001/00177T 1998-07-21 1999-07-20 Antifungal Aktiviteye sahip bir bileşimin oral farmasötik kompozisyonu ve bu kompozisyonun hazırlanış metodu. TR200100177T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES009801539A ES2157731B1 (es) 1998-07-21 1998-07-21 Preparacion farmaceutica oral de un compuesto de actividad antifungica y procedimiento para su preparacion.

Publications (1)

Publication Number Publication Date
TR200100177T2 true TR200100177T2 (tr) 2001-07-23

Family

ID=8304581

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/00177T TR200100177T2 (tr) 1998-07-21 1999-07-20 Antifungal Aktiviteye sahip bir bileşimin oral farmasötik kompozisyonu ve bu kompozisyonun hazırlanış metodu.

Country Status (31)

Country Link
US (1) US6737082B1 (tr)
EP (1) EP1103252B1 (tr)
JP (1) JP4190732B2 (tr)
KR (1) KR100572135B1 (tr)
AT (1) ATE234077T1 (tr)
AU (1) AU750730B2 (tr)
BG (1) BG65187B1 (tr)
BR (1) BR9912300A (tr)
CA (1) CA2337509C (tr)
CZ (1) CZ291938B6 (tr)
DE (1) DE69905905T2 (tr)
DK (1) DK1103252T3 (tr)
EE (1) EE04415B1 (tr)
ES (2) ES2157731B1 (tr)
HK (1) HK1037531A1 (tr)
HR (1) HRP20010128B1 (tr)
HU (1) HU228895B1 (tr)
IL (1) IL140910A (tr)
ME (1) MEP26708A (tr)
MX (1) MXPA01000681A (tr)
NO (1) NO320054B1 (tr)
NZ (1) NZ509886A (tr)
PL (1) PL194740B1 (tr)
PT (1) PT1103252E (tr)
RS (1) RS50063B (tr)
RU (1) RU2209628C2 (tr)
SK (1) SK283279B6 (tr)
TR (1) TR200100177T2 (tr)
UA (1) UA64009C2 (tr)
WO (1) WO2000004881A1 (tr)
ZA (1) ZA200101293B (tr)

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FR2842736B1 (fr) * 2002-07-26 2005-07-22 Flamel Tech Sa Formulation pharmaceutique orale sous forme d'une pluralite de microcapsules permettant la liberation prolongee de principe(s) actif(s) peu soluble(s)
US20040115287A1 (en) * 2002-12-17 2004-06-17 Lipocine, Inc. Hydrophobic active agent compositions and methods
DK1438960T4 (da) * 2003-01-14 2013-03-25 Cimex Pharma Ag Sammensætning af itraconazol dispergeret i en hydrofil polymer med forhøjet biotilgængelighed
SI1438961T2 (sl) * 2003-01-14 2014-12-31 Cimex Pharma Ag Bioekvivalenten sestavek itrakonazola, dispergiranega v hidrofilnem polimeru
FR2852607B1 (fr) * 2003-03-20 2006-07-14 Procede de fabrication de microspheres de sucre de petite taille, les microspheres susceptibles d'etre obtenues par ce procede et leurs applications
BRPI0412734A (pt) * 2003-07-17 2006-09-26 Tibotec Pharm Ltd processo para preparação de partìculas que contêm um antiviral
FR2857591B1 (fr) * 2003-07-17 2007-11-02 Ethypharm Sa Particules comprenant un principe actif sous forme de co-precipite
FR2883179B1 (fr) 2005-03-18 2009-04-17 Ethypharm Sa Comprime enrobe
JP5435946B2 (ja) 2005-08-22 2014-03-05 ジョンズ ホプキンス ユニバーシティ 疾患を処置するためのヘッジホッグ経路アンタゴニスト
CN101283984B (zh) * 2007-04-12 2010-05-26 永胜药品工业股份有限公司 高生物使用率的经杀真菌剂和聚合物涂覆的核心微粒状物
US11304960B2 (en) 2009-01-08 2022-04-19 Chandrashekar Giliyar Steroidal compositions
EP2542222A2 (de) * 2010-03-05 2013-01-09 Basf Se Schmelzüberzogene arzneiformen
US9034858B2 (en) 2010-11-30 2015-05-19 Lipocine Inc. High-strength testosterone undecanoate compositions
US9358241B2 (en) 2010-11-30 2016-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US20120148675A1 (en) 2010-12-10 2012-06-14 Basawaraj Chickmath Testosterone undecanoate compositions
US9498485B2 (en) 2014-08-28 2016-11-22 Lipocine Inc. Bioavailable solid state (17-β)-hydroxy-4-androsten-3-one esters
US20170246187A1 (en) 2014-08-28 2017-08-31 Lipocine Inc. (17-ß)-3-OXOANDROST-4-EN-17-YL TRIDECANOATE COMPOSITIONS AND METHODS OF THEIR PREPARATION AND USE
MA40982A (fr) * 2014-11-19 2017-09-26 Biogen Ma Inc Formulation de bille pharmaceutique comprenant du fumarate de diméthyle
RU2017141029A (ru) * 2015-05-25 2019-06-25 Сан Фармасьютикал Индастриз Лимитед Фармацевтическая пероральная композиция изотретиноина для применения один раз в сутки
AU2017310506B2 (en) 2016-08-11 2019-11-21 Dmk Pharmaceuticals Corporation Drug compositions
WO2018098501A1 (en) 2016-11-28 2018-05-31 Lipocine Inc. Oral testosterone undecanoate therapy
US11564910B2 (en) 2017-12-08 2023-01-31 Adamis Pharmaceuticals Corporation Drug compositions
WO2019208801A1 (ja) * 2018-04-27 2019-10-31 凸版印刷株式会社 徐放性複合粒子、徐放性複合粒子の製造方法、乾燥粉体及び壁紙
WO2023118082A1 (en) * 2021-12-22 2023-06-29 Palau Pharma, S.L.U. Multiparticulate albaconazole composition

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Also Published As

Publication number Publication date
HUP0103708A2 (hu) 2002-02-28
ES2194480T3 (es) 2003-11-16
YU3901A (sh) 2003-08-29
NZ509886A (en) 2002-09-27
HUP0103708A3 (en) 2002-07-29
JP2002521323A (ja) 2002-07-16
KR20010070990A (ko) 2001-07-28
NO320054B1 (no) 2005-10-17
BG65187B1 (bg) 2007-06-29
ATE234077T1 (de) 2003-03-15
ZA200101293B (en) 2001-08-21
HRP20010128B1 (en) 2003-12-31
PL194740B1 (pl) 2007-06-29
CA2337509A1 (en) 2000-02-03
NO20010289L (no) 2001-03-07
US6737082B1 (en) 2004-05-18
EP1103252B1 (en) 2003-03-12
ES2157731B1 (es) 2002-05-01
IL140910A (en) 2004-03-28
EE200100041A (et) 2002-06-17
PT1103252E (pt) 2003-07-31
DK1103252T3 (da) 2003-07-14
HRP20010128A2 (en) 2002-12-31
DE69905905D1 (de) 2003-04-17
BG105282A (en) 2001-11-30
RU2209628C2 (ru) 2003-08-10
DE69905905T2 (de) 2004-03-04
KR100572135B1 (ko) 2006-04-19
NO20010289D0 (no) 2001-01-17
AU4782199A (en) 2000-02-14
ES2157731A1 (es) 2001-08-16
SK283279B6 (sk) 2003-05-02
IL140910A0 (en) 2002-02-10
CZ291938B6 (cs) 2003-06-18
MEP26708A (en) 2010-06-10
MXPA01000681A (es) 2002-04-24
AU750730B2 (en) 2002-07-25
HK1037531A1 (en) 2002-02-15
EP1103252A1 (en) 2001-05-30
PL345625A1 (en) 2002-01-02
UA64009C2 (en) 2004-02-16
EE04415B1 (et) 2005-02-15
CZ2001175A3 (en) 2001-05-16
WO2000004881A1 (es) 2000-02-03
SK862001A3 (en) 2001-08-06
JP4190732B2 (ja) 2008-12-03
BR9912300A (pt) 2001-04-17
RS50063B (sr) 2009-01-22
HU228895B1 (en) 2013-06-28
CA2337509C (en) 2005-12-27

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