TR199900712T2 - 1H-Pirido$3,4-b]indol-4-karboksamid t�revleri, haz�rlanmalar� ve terapide uygulanmas�. - Google Patents

1H-Pirido$3,4-b]indol-4-karboksamid t�revleri, haz�rlanmalar� ve terapide uygulanmas�.

Info

Publication number
TR199900712T2
TR199900712T2 TR1999/00712T TR9900712T TR199900712T2 TR 199900712 T2 TR199900712 T2 TR 199900712T2 TR 1999/00712 T TR1999/00712 T TR 1999/00712T TR 9900712 T TR9900712 T TR 9900712T TR 199900712 T2 TR199900712 T2 TR 199900712T2
Authority
TR
Turkey
Prior art keywords
group
therapy
alkyl
pirido
indole
Prior art date
Application number
TR1999/00712T
Other languages
English (en)
Turkish (tr)
Inventor
Evanno Yannick
Sevrin Mireille
Maloizel Christian
Legalloudec Odette
George Pascal
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of TR199900712T2 publication Critical patent/TR199900712T2/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
TR1999/00712T 1996-10-08 1997-10-03 1H-Pirido$3,4-b]indol-4-karboksamid t�revleri, haz�rlanmalar� ve terapide uygulanmas�. TR199900712T2 (xx)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9612229A FR2754262B1 (fr) 1996-10-08 1996-10-08 Derives de 1h-pyrido[3,4-b]indole-4-carboxamide, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
TR199900712T2 true TR199900712T2 (xx) 1999-06-21

Family

ID=9496449

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1999/00712T TR199900712T2 (xx) 1996-10-08 1997-10-03 1H-Pirido$3,4-b]indol-4-karboksamid t�revleri, haz�rlanmalar� ve terapide uygulanmas�.

Country Status (33)

Country Link
US (1) US6075021A (et)
EP (1) EP0934319B1 (et)
JP (1) JP4227197B2 (et)
KR (1) KR100488095B1 (et)
CN (1) CN1089765C (et)
AR (1) AR009112A1 (et)
AT (1) ATE218567T1 (et)
AU (1) AU721102B2 (et)
BG (1) BG63751B1 (et)
BR (1) BR9711879A (et)
CA (1) CA2266376A1 (et)
CO (1) CO4910141A1 (et)
CY (1) CY2291B1 (et)
CZ (1) CZ298906B6 (et)
DE (1) DE69713124T2 (et)
DK (1) DK0934319T3 (et)
EE (1) EE03830B1 (et)
ES (1) ES2178008T3 (et)
FR (1) FR2754262B1 (et)
HK (1) HK1023338A1 (et)
HU (1) HUP9904623A3 (et)
IL (1) IL129018A0 (et)
NO (1) NO311938B1 (et)
NZ (1) NZ334708A (et)
PL (1) PL188244B1 (et)
PT (1) PT934319E (et)
RU (1) RU2180904C2 (et)
SK (1) SK282970B6 (et)
TR (1) TR199900712T2 (et)
TW (1) TW461889B (et)
UA (1) UA57037C2 (et)
WO (1) WO1998015552A1 (et)
ZA (1) ZA978970B (et)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2766823B1 (fr) 1997-07-30 1999-10-08 Synthelabo Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique
FR2788776B1 (fr) 1999-01-26 2001-02-23 Synthelabo Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique
FR2788696B1 (fr) * 1999-01-26 2004-03-05 Synthelabo Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central
FR2811990A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo DERIVES DE 1-(4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b]INDOLE-1 -CARBONYL)PIPERAZINE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2811897A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo UTILISATION DE DERIVES DE PYRIDAZINO[4,5-b]INDOLE-1- ACETAMIDE POUR LA PREPARATION DE MEDICAMENTS DESTINES AU TRAITEMENT DES DYSFONCTIONNEMENTS DES RECEPTEURS DE TYPE PERIPHERIQUE AUX BENZODIAZEPINES
FR2833953B1 (fr) * 2001-12-21 2004-12-03 Sanofi Synthelabo DERIVES DE 3-HETEROARYL-3,5-DIHYDRO-4-OXO-4H-PYRIDAZINO [4,5-b]INDOLE-1-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2838124B1 (fr) * 2002-04-03 2004-05-28 Sanofi Synthelabo Derives de 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino [4,5-b]indole-1-acetamide, leur preparation et leur application en therapeutique
PA8586801A1 (es) * 2002-10-31 2005-02-04 Pfizer Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
JP2006516606A (ja) * 2003-01-27 2006-07-06 ファイザー インコーポレイテッド Ｈｉｖインテグラーゼインヒビター、医薬組成物、およびそれらの使用
JP2007534738A (ja) * 2004-04-26 2007-11-29 ファイザー・インク Ｈｉｖインテグラーゼ酵素の阻害剤
BRPI0510319A (pt) * 2004-04-26 2007-10-16 Pfizer inibidores da enzima integrase de hiv
CA2606861C (en) * 2005-05-05 2012-08-07 Sanofi-Aventis U.S. Llc Stable nanoparticle formulations
AP2008004400A0 (en) * 2005-10-07 2008-04-30 Pfizer Prod Inc Inhibitors of HIV integrase enzyme
UA95788C2 (en) 2005-12-15 2011-09-12 Ф. Хоффманн-Ля Рош Аг Fused pyrrole derivatives
PT2029572E (pt) * 2006-06-05 2011-02-09 Novartis Ag Compostos orgânicos
CN1946120B (zh) * 2006-10-20 2010-05-12 华为技术有限公司 实现话单关联的方法及系统
KR100688448B1 (ko) * 2006-12-06 2007-03-02 (주)경진건축사사무소 건축물 내부 조적구조

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2724384B1 (fr) * 1994-09-14 1999-04-16 Cemaf Nouveaux derives de la 3,4-dihydro beta-carboline agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament

Also Published As

Publication number Publication date
JP4227197B2 (ja) 2009-02-18
KR100488095B1 (ko) 2005-05-09
UA57037C2 (uk) 2003-06-16
BG103301A (en) 2000-05-31
FR2754262B1 (fr) 1998-10-30
NO311938B1 (no) 2002-02-18
AU721102B2 (en) 2000-06-22
JP2001508403A (ja) 2001-06-26
CN1089765C (zh) 2002-08-28
DE69713124D1 (de) 2002-07-11
HUP9904623A2 (hu) 2000-06-28
SK282970B6 (sk) 2003-01-09
CO4910141A1 (es) 2000-04-24
PT934319E (pt) 2002-10-31
ZA978970B (en) 1998-04-20
DK0934319T3 (da) 2002-09-30
ATE218567T1 (de) 2002-06-15
EE03830B1 (et) 2002-08-15
RU2180904C2 (ru) 2002-03-27
CZ119399A3 (cs) 1999-07-14
NO991624L (no) 1999-06-07
KR20000048992A (ko) 2000-07-25
AR009112A1 (es) 2000-03-08
CZ298906B6 (cs) 2008-03-12
HUP9904623A3 (en) 2001-03-28
CY2291B1 (en) 2003-07-04
NO991624D0 (no) 1999-04-06
BG63751B1 (bg) 2002-11-29
SK45199A3 (en) 2000-02-14
BR9711879A (pt) 1999-08-24
CA2266376A1 (en) 1998-04-16
PL188244B1 (pl) 2005-01-31
HK1023338A1 (en) 2000-09-08
EP0934319A1 (fr) 1999-08-11
WO1998015552A1 (fr) 1998-04-16
FR2754262A1 (fr) 1998-04-10
DE69713124T2 (de) 2003-01-30
US6075021A (en) 2000-06-13
PL332643A1 (en) 1999-09-27
CN1233248A (zh) 1999-10-27
IL129018A0 (en) 2000-02-17
NZ334708A (en) 2000-10-27
EE9900155A (et) 1999-12-15
ES2178008T3 (es) 2002-12-16
EP0934319B1 (fr) 2002-06-05
TW461889B (en) 2001-11-01
AU4559497A (en) 1998-05-05

Similar Documents

Publication Publication Date Title
TR199900712T2 (xx) 1H-Pirido$3,4-b]indol-4-karboksamid t�revleri, haz�rlanmalar� ve terapide uygulanmas�.
TW328086B (en) Biphenylamides, compositions comprising them and the preparation and use thereof
TR199800464T1 (xx) Serotonin antagonistleri olarak kinolein-2(1H)-on t�revleri
IL133825A0 (en) Substituted 6-phenylphenanthridines, medicaments containing same and use thereof
HUP9901820A2 (hu) 4-Amino-pirimidin-származékok, ezeket tartalmazó gyógyszerkészítmények, alkalmazásuk és eljárás előállításukra
IL122855A0 (en) 7H-pyrrolo [2,3-d] pyrimidine derivatives their preparation and pharmaceutical compositions containing them
HUP0004807A2 (hu) Vérlemezkéből származó növekedési faktort és/vagy P56lck tirozin kinázokat gátló hatású kinolin- és kinoxalin-vegyületek, alkalmazásuk gyógyászati készítmények előállítására és a vegyületeket tartalmazó gyógyászati készítmények
TR199800780T2 (xx) Kayna�m�� tropan t�revleri, haz�rlan��lar� ve kullan�mlar�.
ATE179698T1 (de) Pyrrolidin- und oxazolidin derivate , ihre herstellung und ihre verwendung als thrombocyten- aggregations-hemmer
IS5352A (is) Ný efnasambönd
IL133824A0 (en) Tetrazole derivatives, medicaments containing same and use thereof
HUP9903948A2 (hu) Tachikinin antagonista 1-(1,2-diszubsztituált piperidinil)-4-(kondenzált imidazolil)-piperidin-származékok, előállításuk és alkalmazásuk
HUP0001865A2 (hu) Amino-pirimidin-származékok, alkalmazásuk, eljárás előállításukra és az ezeket tartalmazó gyógyszerkészítmények
TR199902367T2 (xx) 16-Hidroksi-11-(ikameli fenil)-estra-4,9-dien t�revleri.
AU2797695A (en) Thiazolidine derivatives, their preparation and drugs containing same
AU681688B2 (en) Imidazo(1,2-a)pyrazine-4-one, preparation thereof and drugs containing same
CA2298522A1 (en) 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b]-indole-1-acetamide derivatives, their preparation and their application in therapy
HUP0101469A2 (hu) 5-[(2-Imidazolidinilidén)-amino]-benzimidazol-származékok, előállításuk és alkalmazásuk javított metabolikus stabilitású alfa-adrenoceptor agonistákként
TR199902115T2 (xx) 2,3- Dihidrofuro (3,2-b) piridiun t�revleri, haz�rlan��lar� ve terapide uygulanmalar�.
ATE225335T1 (de) Amide derivate als 5-ht1a liganden
TR199900634T2 (xx) N-(Benzotiazol-2-il) Piperidin-1-etanamin t�revleri, haz�rlanmalar� ve terapide uygulanmas�.
TR199902600T2 (xx) 5-HT4 Resept�r ligandlar� olarak 5-aril-3-(8-azabisayklo $3.2.1]okt-3-il)-1,3,4-okzadiazol-2(3h)-on t�revleri.
DK0772615T3 (da) Imidazo[1,2-a]indeno[1,2-e]pyrazin-2-carboxylsyrederivater, fremstilling af disse forbindelser og lægemidler indeholdende d
TR200000057T2 (tr) 6-pirolidin-2-ilpirindinler, hazırlanmaları ve terapötik uygulamaları.
MY133140A (en) N-substituted azabicycloheptane derivatives, their preparation and use