TNSN86135A1 - Procede de preparation de nouveaux derives bicycliques du catechol - Google Patents

Procede de preparation de nouveaux derives bicycliques du catechol

Info

Publication number
TNSN86135A1
TNSN86135A1 TNTNSN86135A TNSN86135A TNSN86135A1 TN SN86135 A1 TNSN86135 A1 TN SN86135A1 TN TNSN86135 A TNTNSN86135 A TN TNSN86135A TN SN86135 A TNSN86135 A TN SN86135A TN SN86135 A1 TNSN86135 A1 TN SN86135A1
Authority
TN
Tunisia
Prior art keywords
preparation
catechol
bicyclic derivatives
new bicyclic
formula
Prior art date
Application number
TNTNSN86135A
Other languages
English (en)
Inventor
Follet Michel
Bonato Marc
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of TNSN86135A1 publication Critical patent/TNSN86135A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/06—Benzothiopyrans; Hydrogenated benzothiopyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10—Sulfides; Sulfoxides; Sulfones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Steroid Compounds (AREA)

Abstract

LA PRESENTE INVENTION CONCERNE UN PROCEDE DE PREPARATION DES DERIVES BICYCLIQUES DU CATECHOL REPONDANT A L'UNE DES FORMULES GENERALES I ET II. DANS LESQUELLES R1, R2, R3 ET Z REPRESENTENT DIFFERENTS SUBSTITUANTS, CONSISTANT A FAIRE REAGIR UN COMPOSE DE FORMULE III. DANS LAQUELLE R1 ET R2 ONT LES MEMES SIGNIFICATIONS QUE CI-DESSUS SUR UN ACIDE OU UN ESTER PROPIONIQUE OU BUTYRIQUE DE FORMULE IV. DANS LAQUELLE R3 A LA MEME SIGNIFICATION QUE CI-DESSUS
TNTNSN86135A 1985-09-26 1986-09-26 Procede de preparation de nouveaux derives bicycliques du catechol TNSN86135A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858523776A GB8523776D0 (en) 1985-09-26 1985-09-26 Catechol derivatives

Publications (1)

Publication Number Publication Date
TNSN86135A1 true TNSN86135A1 (fr) 1990-01-01

Family

ID=10585770

Family Applications (2)

Application Number Title Priority Date Filing Date
TNTNSN86134A TNSN86134A1 (fr) 1985-09-26 1986-09-26 Procede de preparation de nouveaux derives du catechol
TNTNSN86135A TNSN86135A1 (fr) 1985-09-26 1986-09-26 Procede de preparation de nouveaux derives bicycliques du catechol

Family Applications Before (1)

Application Number Title Priority Date Filing Date
TNTNSN86134A TNSN86134A1 (fr) 1985-09-26 1986-09-26 Procede de preparation de nouveaux derives du catechol

Country Status (28)

Country Link
US (2) US4699919A (fr)
JP (2) JPS6284055A (fr)
AR (2) AR242559A1 (fr)
AT (2) AT396469B (fr)
BE (2) BE905433A (fr)
CA (2) CA1318686C (fr)
CH (2) CH668421A5 (fr)
DE (2) DE3632824A1 (fr)
DK (2) DK165115C (fr)
DZ (2) DZ990A1 (fr)
ES (2) ES2001705A6 (fr)
FI (2) FI84480C (fr)
FR (4) FR2587702B1 (fr)
GB (3) GB8523776D0 (fr)
HK (2) HK91289A (fr)
IE (2) IE59479B1 (fr)
IT (2) IT1235760B (fr)
LU (2) LU86591A1 (fr)
MA (2) MA20779A1 (fr)
MY (2) MY103521A (fr)
NL (2) NL189410C (fr)
NO (2) NO165238C (fr)
OA (2) OA08417A (fr)
PT (2) PT83436B (fr)
SE (2) SE467053B (fr)
SG (1) SG65889G (fr)
TN (2) TNSN86134A1 (fr)
ZA (2) ZA866905B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4927629A (en) * 1987-12-17 1990-05-22 Huntington Medical Research Institutes Relaxation of smooth vascular muscle
AU1520699A (en) 1997-11-07 1999-05-31 Johns Hopkins University, The Methods for treatment of disorders of cardiac contractility
CN102159203A (zh) * 2008-07-23 2011-08-17 麻省理工学院 组蛋白脱乙酰酶1(hdac1)的活化防范dna损伤和增加神经元存活
ES2719266T3 (es) 2011-07-22 2019-07-09 Massachusetts Inst Technology Activadores de histona desacetilasas de clase I (HDACS), y usos de los mismos

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2549118A (en) * 1949-10-05 1951-04-17 Us Rubber Co Vulcanized rubber and method of preserving same
CH301691A (de) * 1951-08-07 1954-09-15 Cilag Ag Verfahren zur Herstellung eines neuen aromatischen Thioäthers.
CH301688A (de) * 1951-08-07 1954-09-15 Cilag Ag Verfahren zur Herstellung eines neuen aromatischen Thioäthers.
CH301687A (de) * 1951-08-07 1954-09-15 Cilag Ag Verfahren zur Herstellung eines neuen aromatischen Thioäthers.
US3148997A (en) * 1963-01-04 1964-09-15 Dow Chemical Co Catechol compounds in improving clays and clay-containing materials
US3282979A (en) * 1963-06-17 1966-11-01 Dow Chemical Co Phenolic thioethers
US3274257A (en) * 1963-06-17 1966-09-20 Dow Chemical Co Synthesis of (alkylthio) phenols
GB1362782A (en) * 1970-08-26 1974-08-07 Fisons Ltd Tetrazole derivatives
US3751483A (en) * 1971-10-13 1973-08-07 Crown Zellerbach Corp Phenolic thioethers and process for preparing same
GB1428110A (en) * 1972-05-30 1976-03-17 Reckitt & Colmann Prod Ltd Pharmaceutical antihypertensive and vasodilator compositions
JPS506340A (fr) * 1973-05-16 1975-01-23
DE2644591A1 (de) * 1976-10-02 1978-04-06 Bayer Ag Verfahren zur herstellung von arylsulfoniumsalzen
AU548253B2 (en) * 1981-05-11 1985-12-05 Pierre Fabre S.A. Benzoxepine derivatives and sulphur and nitrogen analogues thereof
US4661505A (en) * 1982-11-03 1987-04-28 Eli Lilly And Company Leukotriene antagonists
JPS60260532A (ja) * 1984-06-07 1985-12-23 Yamanouchi Pharmaceut Co Ltd 新規カテコ−ル誘導体
US4785004A (en) * 1985-12-23 1988-11-15 Ciba-Geigy Corporation Aromatic thioethers

Also Published As

Publication number Publication date
AR241702A1 (es) 1992-11-30
GB8623075D0 (en) 1986-10-29
BE905432A (fr) 1987-03-16
US4699919A (en) 1987-10-13
GB2189782B (en) 1989-04-12
DK457386A (da) 1987-03-27
FR2587699B1 (fr) 1988-11-10
ES2001705A6 (es) 1988-06-01
GB8623074D0 (en) 1986-10-29
ZA866906B (en) 1987-04-29
BE905433A (fr) 1987-03-16
NL8602383A (nl) 1987-04-16
NL189410B (nl) 1992-11-02
IE59479B1 (en) 1994-03-09
IE862532L (en) 1987-03-26
FR2587703A1 (fr) 1987-03-27
IT1235761B (it) 1992-09-28
PT83436A (en) 1986-10-01
SE467053B (sv) 1992-05-18
NO863834D0 (no) 1986-09-25
DK168334B1 (da) 1994-03-14
JPS6284055A (ja) 1987-04-17
DZ991A1 (fr) 2004-09-13
MA20779A1 (fr) 1987-04-01
NL8602382A (nl) 1987-04-16
CA1278299C (fr) 1990-12-27
FI863742A0 (fi) 1986-09-16
GB2181431B (en) 1989-09-20
JPS6284080A (ja) 1987-04-17
AR242559A1 (es) 1993-04-30
GB2181431A (en) 1987-04-23
TNSN86134A1 (fr) 1990-01-01
CH668261A5 (fr) 1988-12-15
CA1318686C (fr) 1993-06-01
IT8621836A0 (it) 1986-09-26
DK165115B (da) 1992-10-12
FI863743A0 (fi) 1986-09-16
FI84480C (fi) 1991-12-10
OA08417A (fr) 1988-06-30
FR2587702A1 (fr) 1987-03-27
LU86590A1 (fr) 1987-01-22
MY103521A (en) 1993-07-31
NO863835D0 (no) 1986-09-25
NO170415C (no) 1992-10-14
FR2587698B1 (fr) 1989-04-28
FR2587703B1 (fr) 1988-11-04
NO165238B (no) 1990-10-08
MY105863A (en) 1995-02-28
MA20780A1 (fr) 1987-04-01
JPH0482129B2 (fr) 1992-12-25
DE3632841A1 (de) 1987-04-02
IE59478B1 (en) 1994-03-09
OA08416A (fr) 1988-06-30
IE862533L (en) 1987-03-26
PT83437B (pt) 1988-07-29
IT1235760B (it) 1992-09-28
AT402070B (de) 1997-01-27
NO165238C (no) 1991-01-16
GB2189782A (en) 1987-11-04
HK91289A (en) 1989-11-24
HK46190A (en) 1990-06-22
FI87646C (fi) 1993-02-10
CH668421A5 (fr) 1988-12-30
SE8603793D0 (sv) 1986-09-10
FI84480B (fi) 1991-08-30
PT83437A (en) 1986-10-01
FI87646B (fi) 1992-10-30
NO170415B (no) 1992-07-06
SE8603792L (sv) 1987-03-27
DK165115C (da) 1993-03-01
FI863743A (fi) 1987-03-27
SE464522B (sv) 1991-05-06
FR2587698A1 (fr) 1987-03-27
DK457386D0 (da) 1986-09-25
IT8621837A0 (it) 1986-09-26
FR2587699A1 (fr) 1987-03-27
DE3632824A1 (de) 1987-04-02
DK457486D0 (da) 1986-09-25
DE3632824C2 (fr) 1992-04-30
DZ990A1 (fr) 2004-09-13
US5013756A (en) 1991-05-07
NO863834L (no) 1987-03-27
SG65889G (en) 1990-01-26
NO863835L (no) 1987-03-27
DK457486A (da) 1987-03-27
ATA257386A (de) 1993-01-15
ES2001440A6 (es) 1988-05-16
LU86591A1 (fr) 1987-01-22
ATA257486A (de) 1996-06-15
SE8603792D0 (sv) 1986-09-10
NL189334C (nl) 1993-03-16
AT396469B (de) 1993-09-27
DE3632841C2 (fr) 1992-06-11
FR2587702B1 (fr) 1988-11-04
GB8523776D0 (en) 1985-10-30
FI863742A (fi) 1987-03-27
JPH0417956B2 (fr) 1992-03-26
NL189410C (nl) 1993-04-01
SE8603793L (sv) 1987-03-27
PT83436B (pt) 1988-07-29
ZA866905B (en) 1987-04-29

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