TNSN03113A1 - Sels consistant en tartrates de 5,8,14 - triazatetracyclo [10.3.1. 02, 11, 04,9] - hexadeca - 2 (11),3,5,7,9 - pentaene.et compositions pharmaceutiques le contenant. - Google Patents

Sels consistant en tartrates de 5,8,14 - triazatetracyclo [10.3.1. 02, 11, 04,9] - hexadeca - 2 (11),3,5,7,9 - pentaene.et compositions pharmaceutiques le contenant.

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Publication number
TNSN03113A1
TNSN03113A1 TNPCT/IB2002/001437A TNSN03113A TNSN03113A1 TN SN03113 A1 TNSN03113 A1 TN SN03113A1 TN SN03113 A TNSN03113 A TN SN03113A TN SN03113 A1 TNSN03113 A1 TN SN03113A1
Authority
TN
Tunisia
Prior art keywords
tartrate
triazatetracyclo
pentaene
hexadeca
polymorphic forms
Prior art date
Application number
TNPCT/IB2002/001437A
Other languages
English (en)
Inventor
David Everett Bogle
Peter Robert Rose
Glenn Robert Williams
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23117845&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TNSN03113(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN03113A1 publication Critical patent/TNSN03113A1/fr

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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
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Abstract

LA PRESENTE INVENTION CONCERNE DES SELS CONSISTNT EN TARTRATE DE 5,8,14-TRIAZATETRACYCLO[10.3.1.02,11.04,9]-HEXADECA-2(11),3,5,7,9-PENTAENE DE FORMULE (1), ET DES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT. LA PRESENTE INVENTION CONCERNE EN PARTICULIER LE SEL CONSISTANT EN L-TARTRATE, AINSI QUE LES DIFFERENTES FORMES POLYMORPHES DU SEL CONSISTANT EN L -TARTRATE, COMPRENANT DEUX FORMES POLYMORPHES ANHYDRES DISTINCTES (APPELES DANS LE PRESENT MEMOIRE FORMES A ET B) ET UNE FORME POLYMORPHE HYDRATE (APPELES DANS LE PRESENT MEMOIRE FORME C). EN OUTRE, LA PRESENTE INVENTION CONCERNE EGALEMENT EGALEMENT LE SEL CONSISTANT EN D-TARTRATE DE 5,8,14-TRIAZATETRACYCLO[10.3.02,11.04,9]- HEXADECA-2(11),3,5,7,9-PENTAENE ET SES DIFFERENTES FORMES POLYMORPHES, AINSI QUE SON SEL CONSISTANT EN D,L TARTRATE DE CE COMPOSE ET SES FORMES POLYMORPHES, ET LE SEL CONSISTANT EN MESO-TARTRATE DE CE COMPOSE ET SES FORMES POLYMORPHES.
TNPCT/IB2002/001437A 2001-05-14 2003-07-08 Sels consistant en tartrates de 5,8,14 - triazatetracyclo [10.3.1. 02, 11, 04,9] - hexadeca - 2 (11),3,5,7,9 - pentaene.et compositions pharmaceutiques le contenant. TNSN03113A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29086101P 2001-05-14 2001-05-14

Publications (1)

Publication Number Publication Date
TNSN03113A1 true TNSN03113A1 (fr) 2005-12-23

Family

ID=23117845

Family Applications (1)

Application Number Title Priority Date Filing Date
TNPCT/IB2002/001437A TNSN03113A1 (fr) 2001-05-14 2003-07-08 Sels consistant en tartrates de 5,8,14 - triazatetracyclo [10.3.1. 02, 11, 04,9] - hexadeca - 2 (11),3,5,7,9 - pentaene.et compositions pharmaceutiques le contenant.

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US (2) US6890927B2 (fr)
EP (1) EP1392307B1 (fr)
JP (1) JP3779682B2 (fr)
KR (1) KR100551184B1 (fr)
CN (1) CN100370987C (fr)
AP (1) AP1473A (fr)
AR (1) AR033635A1 (fr)
AT (1) ATE302607T1 (fr)
AU (1) AU2002253482B2 (fr)
BG (1) BG66408B1 (fr)
BR (1) BR0209605A (fr)
CA (1) CA2447405C (fr)
CR (1) CR7080A (fr)
CZ (1) CZ304763B6 (fr)
DE (1) DE60205742T2 (fr)
DK (1) DK1392307T3 (fr)
DO (1) DOP2002000392A (fr)
EA (1) EA005528B1 (fr)
EC (2) ECSP034850A (fr)
EE (1) EE05441B1 (fr)
EG (1) EG24228A (fr)
ES (1) ES2246396T3 (fr)
GE (1) GEP20053712B (fr)
GT (1) GT200200084A (fr)
HK (1) HK1062645A1 (fr)
HR (1) HRP20030910B1 (fr)
HU (1) HU229867B1 (fr)
IL (2) IL157933A0 (fr)
IS (1) IS2217B (fr)
MA (1) MA27020A1 (fr)
ME (1) ME00466B (fr)
MX (1) MXPA03010364A (fr)
MY (1) MY127807A (fr)
NO (1) NO326148B1 (fr)
NZ (1) NZ528210A (fr)
OA (1) OA12599A (fr)
PA (1) PA8545101A1 (fr)
PE (1) PE20021065A1 (fr)
PL (1) PL214876B1 (fr)
PT (1) PT1392307E (fr)
RS (1) RS50814B (fr)
SI (1) SI1392307T1 (fr)
SK (1) SK287170B6 (fr)
TN (1) TNSN03113A1 (fr)
TW (1) TWI262078B (fr)
UA (1) UA73422C2 (fr)
WO (1) WO2002092089A1 (fr)
ZA (1) ZA200307235B (fr)

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CN113980020B (zh) * 2021-11-22 2023-05-09 浙江车头制药股份有限公司 一种酒石酸伐尼克兰晶型的制备方法
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