BR0209605A - Sais tartarato de 5,8,14-triazatetraciclo[10.3.1.0.²,¹¹.04,9]-hexadeca-2(11), 3,5,7,9-pentaeno - Google Patents

Sais tartarato de 5,8,14-triazatetraciclo[10.3.1.0.²,¹¹.04,9]-hexadeca-2(11), 3,5,7,9-pentaeno

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Publication number
BR0209605A
BR0209605A BR0209605-6A BR0209605A BR0209605A BR 0209605 A BR0209605 A BR 0209605A BR 0209605 A BR0209605 A BR 0209605A BR 0209605 A BR0209605 A BR 0209605A
Authority
BR
Brazil
Prior art keywords
hexadeca
polymorphs
pentaene
triazatetracyclo
salts
Prior art date
Application number
BR0209605-6A
Other languages
English (en)
Inventor
David Everett Bogle
Peter Robert Rose
Glenn Robert Williams
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23117845&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0209605(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BR0209605A publication Critical patent/BR0209605A/pt

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

"SAIS TARTARATO DE 5,8,14-TRIAZATETRACICLO [10.3.1 .0^ 2,11^.0^ 4,9^]-HEXADECA-2(11),3,5,7,9-PENTAENO". A presente invenção refere-se aos sais tartarato de 5,8,14triazatetraciclo[10.3.1.0^ 2,11^.0^ 4,9^]-hexadeca-2(11),3,5,7,9-pentaeno de fórmula (1): e suas composições farmacêuticas. Em particular a presente invenção refere-se ao sal L-tartarato, e ainda aos vários polimorfos do sal L-tartarato, incluindo dois polimorfos anidros distintos (aqui referidos como Formas A e B) e um polimorfo hidrato (aqui referido como Forma C). Além disso, a presente invenção também refere-se ao sal D-tartarato de 5,8,14-triazatetraciclo [10.3.1 .0^ 2,11^.0^ 4,9^]-hexadeca-2(11),3,5,7,9-pentaeno e aos seus vários polimorfos; bem como ao sal D,L-tartarato e aos seus polimorfos, e ao sal mesotartarato e aos seus polimorfos.
BR0209605-6A 2001-05-14 2002-04-26 Sais tartarato de 5,8,14-triazatetraciclo[10.3.1.0.²,¹¹.04,9]-hexadeca-2(11), 3,5,7,9-pentaeno BR0209605A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29086101P 2001-05-14 2001-05-14
PCT/IB2002/001437 WO2002092089A1 (en) 2001-05-14 2002-04-26 Tartrate salts of 5,8,14-triazatetracyclo {10.3.1.0?2,11.04,9¿}-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
BR0209605A true BR0209605A (pt) 2004-03-23

Family

ID=23117845

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0209605-6A BR0209605A (pt) 2001-05-14 2002-04-26 Sais tartarato de 5,8,14-triazatetraciclo[10.3.1.0.²,¹¹.04,9]-hexadeca-2(11), 3,5,7,9-pentaeno

Country Status (48)

Country Link
US (2) US6890927B2 (pt)
EP (1) EP1392307B1 (pt)
JP (1) JP3779682B2 (pt)
KR (1) KR100551184B1 (pt)
CN (1) CN100370987C (pt)
AP (1) AP1473A (pt)
AR (1) AR033635A1 (pt)
AT (1) ATE302607T1 (pt)
AU (1) AU2002253482B2 (pt)
BG (1) BG66408B1 (pt)
BR (1) BR0209605A (pt)
CA (1) CA2447405C (pt)
CR (1) CR7080A (pt)
CZ (1) CZ304763B6 (pt)
DE (1) DE60205742T2 (pt)
DK (1) DK1392307T3 (pt)
DO (1) DOP2002000392A (pt)
EA (1) EA005528B1 (pt)
EC (2) ECSP034849A (pt)
EE (1) EE05441B1 (pt)
EG (1) EG24228A (pt)
ES (1) ES2246396T3 (pt)
GE (1) GEP20053712B (pt)
GT (1) GT200200084A (pt)
HK (1) HK1062645A1 (pt)
HR (1) HRP20030910B1 (pt)
HU (1) HU229867B1 (pt)
IL (2) IL157933A0 (pt)
IS (1) IS2217B (pt)
MA (1) MA27020A1 (pt)
ME (1) ME00466B (pt)
MX (1) MXPA03010364A (pt)
MY (1) MY127807A (pt)
NO (1) NO326148B1 (pt)
NZ (1) NZ528210A (pt)
OA (1) OA12599A (pt)
PA (1) PA8545101A1 (pt)
PE (1) PE20021065A1 (pt)
PL (1) PL214876B1 (pt)
PT (1) PT1392307E (pt)
RS (1) RS50814B (pt)
SI (1) SI1392307T1 (pt)
SK (1) SK287170B6 (pt)
TN (1) TNSN03113A1 (pt)
TW (1) TWI262078B (pt)
UA (1) UA73422C2 (pt)
WO (1) WO2002092089A1 (pt)
ZA (1) ZA200307235B (pt)

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IL137937A0 (en) * 1999-08-27 2001-10-31 Pfizer Prod Inc A pharmaceutical composition for the prevention and treatment of nicotine addiction in a mammal
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