TN2014000433A1 - Dosage regimen for a pi-3 kinase inhibitor - Google Patents

Dosage regimen for a pi-3 kinase inhibitor

Info

Publication number
TN2014000433A1
TN2014000433A1 TN2014000433A TN2014000433A TN2014000433A1 TN 2014000433 A1 TN2014000433 A1 TN 2014000433A1 TN 2014000433 A TN2014000433 A TN 2014000433A TN 2014000433 A TN2014000433 A TN 2014000433A TN 2014000433 A1 TN2014000433 A1 TN 2014000433A1
Authority
TN
Tunisia
Prior art keywords
dosage regimen
kinase inhibitor
kinase
pi3k
phosphatidylinositol
Prior art date
Application number
TN2014000433A
Other languages
English (en)
French (fr)
Inventor
Samit Hirawat
Cristian Massacesi
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48626588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2014000433(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of TN2014000433A1 publication Critical patent/TN2014000433A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TN2014000433A 2012-05-16 2014-10-17 Dosage regimen for a pi-3 kinase inhibitor TN2014000433A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261647654P 2012-05-16 2012-05-16
PCT/US2013/040877 WO2013173283A1 (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Publications (1)

Publication Number Publication Date
TN2014000433A1 true TN2014000433A1 (en) 2016-03-30

Family

ID=48626588

Family Applications (1)

Application Number Title Priority Date Filing Date
TN2014000433A TN2014000433A1 (en) 2012-05-16 2014-10-17 Dosage regimen for a pi-3 kinase inhibitor

Country Status (19)

Country Link
US (2) US10213432B2 (enExample)
EP (1) EP2849756A1 (enExample)
JP (2) JP6381523B2 (enExample)
KR (1) KR20150009540A (enExample)
CN (1) CN104349779A (enExample)
AU (1) AU2013263043B2 (enExample)
BR (1) BR112014028420A2 (enExample)
CA (1) CA2872526A1 (enExample)
CL (1) CL2014003101A1 (enExample)
HK (1) HK1202435A1 (enExample)
IL (1) IL235567B (enExample)
MX (1) MX360892B (enExample)
NZ (1) NZ700924A (enExample)
PH (1) PH12014502547A1 (enExample)
RU (1) RU2630975C2 (enExample)
SG (2) SG10201608469RA (enExample)
TN (1) TN2014000433A1 (enExample)
WO (1) WO2013173283A1 (enExample)
ZA (1) ZA201407406B (enExample)

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* Cited by examiner, † Cited by third party
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JP6026544B2 (ja) 2011-09-27 2016-11-16 ノバルティス アーゲー 変異体ｉｄｈの阻害剤としての３−ピリミジン−４−イル−オキサゾリジン−２−オン類
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WO2014141104A1 (en) 2013-03-14 2014-09-18 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
WO2015083101A1 (en) 2013-12-06 2015-06-11 Novartis Ag Dosage regimen for an alpha-isoform selective phosphatidylinositol 3-kinase inhibitor
WO2016109426A1 (en) * 2014-12-29 2016-07-07 Verastem, Inc. Oral dosing regimen of a dual mtor and pi3 inhibitor
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WO2018009895A1 (en) * 2016-07-08 2018-01-11 Autotelic Llc Methods for trabedersen dosing by auc

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Also Published As

Publication number Publication date
JP6381523B2 (ja) 2018-08-29
US10213432B2 (en) 2019-02-26
IL235567A0 (en) 2015-01-29
EP2849756A1 (en) 2015-03-25
KR20150009540A (ko) 2015-01-26
NZ700924A (en) 2016-02-26
WO2013173283A1 (en) 2013-11-21
HK1202435A1 (en) 2015-10-02
SG10201608469RA (en) 2016-11-29
MX360892B (es) 2018-11-20
CA2872526A1 (en) 2013-11-21
JP2018108998A (ja) 2018-07-12
US20150141426A1 (en) 2015-05-21
ZA201407406B (en) 2015-11-25
RU2630975C2 (ru) 2017-09-15
IL235567B (en) 2019-08-29
MX2014013904A (es) 2015-01-16
AU2013263043A1 (en) 2014-10-30
AU2013263043B2 (en) 2016-06-16
JP2015517523A (ja) 2015-06-22
CN104349779A (zh) 2015-02-11
US20190134052A1 (en) 2019-05-09
PH12014502547A1 (en) 2015-01-21
BR112014028420A2 (pt) 2017-09-19
SG11201406550QA (en) 2014-11-27
CL2014003101A1 (es) 2015-02-27
RU2014150860A (ru) 2016-07-10

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