CA2872526A1 - Dosage regimen for a pi-3 kinase inhibitor - Google Patents
Dosage regimen for a pi-3 kinase inhibitor Download PDFInfo
- Publication number
- CA2872526A1 CA2872526A1 CA2872526A CA2872526A CA2872526A1 CA 2872526 A1 CA2872526 A1 CA 2872526A1 CA 2872526 A CA2872526 A CA 2872526A CA 2872526 A CA2872526 A CA 2872526A CA 2872526 A1 CA2872526 A1 CA 2872526A1
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- Prior art keywords
- substituted
- pharmaceutically acceptable
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Classifications
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US201261647654P | 2012-05-16 | 2012-05-16 | |
| US61/647,654 | 2012-05-16 | ||
| PCT/US2013/040877 WO2013173283A1 (en) | 2012-05-16 | 2013-05-14 | Dosage regimen for a pi-3 kinase inhibitor |
Publications (1)
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|---|---|
| CA2872526A1 true CA2872526A1 (en) | 2013-11-21 |
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| CA2872526A Abandoned CA2872526A1 (en) | 2012-05-16 | 2013-05-14 | Dosage regimen for a pi-3 kinase inhibitor |
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| CL (1) | CL2014003101A1 (enExample) |
| HK (1) | HK1202435A1 (enExample) |
| IL (1) | IL235567B (enExample) |
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| TN (1) | TN2014000433A1 (enExample) |
| WO (1) | WO2013173283A1 (enExample) |
| ZA (1) | ZA201407406B (enExample) |
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| JP6026544B2 (ja) | 2011-09-27 | 2016-11-16 | ノバルティス アーゲー | 変異体ｉｄｈの阻害剤としての３−ピリミジン−４−イル−オキサゾリジン−２−オン類 |
| UY34632A (es) | 2012-02-24 | 2013-05-31 | Novartis Ag | Compuestos de oxazolidin- 2- ona y usos de los mismos |
| US9296733B2 (en) | 2012-11-12 | 2016-03-29 | Novartis Ag | Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases |
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-
2013
- 2013-05-14 EP EP13729120.9A patent/EP2849756A1/en not_active Withdrawn
- 2013-05-14 CA CA2872526A patent/CA2872526A1/en not_active Abandoned
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- 2013-05-14 HK HK15103031.8A patent/HK1202435A1/xx unknown
- 2013-05-14 US US14/400,444 patent/US10213432B2/en active Active
- 2013-05-14 BR BR112014028420A patent/BR112014028420A2/pt not_active Application Discontinuation
- 2013-05-14 RU RU2014150860A patent/RU2630975C2/ru not_active IP Right Cessation
- 2013-05-14 WO PCT/US2013/040877 patent/WO2013173283A1/en not_active Ceased
- 2013-05-14 JP JP2015512735A patent/JP6381523B2/ja not_active Expired - Fee Related
- 2013-05-14 CN CN201380025377.6A patent/CN104349779A/zh active Pending
- 2013-05-14 SG SG10201608469RA patent/SG10201608469RA/en unknown
- 2013-05-14 KR KR1020147031775A patent/KR20150009540A/ko not_active Ceased
- 2013-05-14 NZ NZ700924A patent/NZ700924A/en not_active IP Right Cessation
- 2013-05-14 MX MX2014013904A patent/MX360892B/es active IP Right Grant
- 2013-05-14 AU AU2013263043A patent/AU2013263043B2/en not_active Ceased
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2014
- 2014-10-13 ZA ZA2014/07406A patent/ZA201407406B/en unknown
- 2014-10-17 TN TN2014000433A patent/TN2014000433A1/fr unknown
- 2014-11-06 IL IL235567A patent/IL235567B/en not_active IP Right Cessation
- 2014-11-14 PH PH12014502547A patent/PH12014502547A1/en unknown
- 2014-11-14 CL CL2014003101A patent/CL2014003101A1/es unknown
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2018
- 2018-01-12 JP JP2018003680A patent/JP2018108998A/ja active Pending
- 2018-12-21 US US16/230,737 patent/US20190134052A1/en not_active Abandoned
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| CN104349779A (zh) | 2015-02-11 |
| US20150141426A1 (en) | 2015-05-21 |
| JP2015517523A (ja) | 2015-06-22 |
| BR112014028420A2 (pt) | 2017-09-19 |
| AU2013263043B2 (en) | 2016-06-16 |
| WO2013173283A1 (en) | 2013-11-21 |
| ZA201407406B (en) | 2015-11-25 |
| IL235567A0 (en) | 2015-01-29 |
| RU2014150860A (ru) | 2016-07-10 |
| JP2018108998A (ja) | 2018-07-12 |
| JP6381523B2 (ja) | 2018-08-29 |
| MX2014013904A (es) | 2015-01-16 |
| TN2014000433A1 (en) | 2016-03-30 |
| NZ700924A (en) | 2016-02-26 |
| IL235567B (en) | 2019-08-29 |
| CL2014003101A1 (es) | 2015-02-27 |
| SG11201406550QA (en) | 2014-11-27 |
| AU2013263043A1 (en) | 2014-10-30 |
| RU2630975C2 (ru) | 2017-09-15 |
| US20190134052A1 (en) | 2019-05-09 |
| HK1202435A1 (en) | 2015-10-02 |
| EP2849756A1 (en) | 2015-03-25 |
| PH12014502547A1 (en) | 2015-01-21 |
| SG10201608469RA (en) | 2016-11-29 |
| MX360892B (es) | 2018-11-20 |
| US10213432B2 (en) | 2019-02-26 |
| KR20150009540A (ko) | 2015-01-26 |
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