PH12014502547A1 - Dosage regimen for a pi-3 kinase inhibitor - Google Patents

Dosage regimen for a pi-3 kinase inhibitor

Info

Publication number
PH12014502547A1
PH12014502547A1 PH12014502547A PH12014502547A PH12014502547A1 PH 12014502547 A1 PH12014502547 A1 PH 12014502547A1 PH 12014502547 A PH12014502547 A PH 12014502547A PH 12014502547 A PH12014502547 A PH 12014502547A PH 12014502547 A1 PH12014502547 A1 PH 12014502547A1
Authority
PH
Philippines
Prior art keywords
dosage regimen
kinase inhibitor
kinase
pi3k
phosphatidylinositol
Prior art date
Application number
PH12014502547A
Other languages
English (en)
Inventor
Hirawat Samit
Massacesi Cristian
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48626588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH12014502547(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PH12014502547A1 publication Critical patent/PH12014502547A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PH12014502547A 2012-05-16 2014-11-14 Dosage regimen for a pi-3 kinase inhibitor PH12014502547A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261647654P 2012-05-16 2012-05-16
PCT/US2013/040877 WO2013173283A1 (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Publications (1)

Publication Number Publication Date
PH12014502547A1 true PH12014502547A1 (en) 2015-01-21

Family

ID=48626588

Family Applications (1)

Application Number Title Priority Date Filing Date
PH12014502547A PH12014502547A1 (en) 2012-05-16 2014-11-14 Dosage regimen for a pi-3 kinase inhibitor

Country Status (19)

Country Link
US (2) US10213432B2 (enExample)
EP (1) EP2849756A1 (enExample)
JP (2) JP6381523B2 (enExample)
KR (1) KR20150009540A (enExample)
CN (1) CN104349779A (enExample)
AU (1) AU2013263043B2 (enExample)
BR (1) BR112014028420A2 (enExample)
CA (1) CA2872526A1 (enExample)
CL (1) CL2014003101A1 (enExample)
HK (1) HK1202435A1 (enExample)
IL (1) IL235567B (enExample)
MX (1) MX360892B (enExample)
NZ (1) NZ700924A (enExample)
PH (1) PH12014502547A1 (enExample)
RU (1) RU2630975C2 (enExample)
SG (2) SG10201608469RA (enExample)
TN (1) TN2014000433A1 (enExample)
WO (1) WO2013173283A1 (enExample)
ZA (1) ZA201407406B (enExample)

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* Cited by examiner, † Cited by third party
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JP6026544B2 (ja) 2011-09-27 2016-11-16 ノバルティス アーゲー 変異体ｉｄｈの阻害剤としての３−ピリミジン−４−イル−オキサゾリジン−２−オン類
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) * 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
GEP201706699B (en) 2013-03-14 2017-07-10 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
CA2930359C (en) 2013-12-06 2022-03-01 Novartis Ag Dosage regimen for an alpha-isoform selective phosphatidylinositol 3-kinase inhibitor
WO2016109426A1 (en) * 2014-12-29 2016-07-07 Verastem, Inc. Oral dosing regimen of a dual mtor and pi3 inhibitor
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WO2018009895A1 (en) * 2016-07-08 2018-01-11 Autotelic Llc Methods for trabedersen dosing by auc

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Also Published As

Publication number Publication date
CA2872526A1 (en) 2013-11-21
HK1202435A1 (en) 2015-10-02
AU2013263043B2 (en) 2016-06-16
IL235567B (en) 2019-08-29
SG11201406550QA (en) 2014-11-27
BR112014028420A2 (pt) 2017-09-19
EP2849756A1 (en) 2015-03-25
JP6381523B2 (ja) 2018-08-29
JP2015517523A (ja) 2015-06-22
TN2014000433A1 (en) 2016-03-30
RU2630975C2 (ru) 2017-09-15
CL2014003101A1 (es) 2015-02-27
US20150141426A1 (en) 2015-05-21
NZ700924A (en) 2016-02-26
CN104349779A (zh) 2015-02-11
KR20150009540A (ko) 2015-01-26
MX360892B (es) 2018-11-20
SG10201608469RA (en) 2016-11-29
JP2018108998A (ja) 2018-07-12
MX2014013904A (es) 2015-01-16
US10213432B2 (en) 2019-02-26
US20190134052A1 (en) 2019-05-09
ZA201407406B (en) 2015-11-25
RU2014150860A (ru) 2016-07-10
IL235567A0 (en) 2015-01-29
AU2013263043A1 (en) 2014-10-30
WO2013173283A1 (en) 2013-11-21

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