SK99799A3 - Use of central cannabinoid receptor antagonists for regulating appetence - Google Patents

Use of central cannabinoid receptor antagonists for regulating appetence Download PDF

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Publication number
SK99799A3
SK99799A3 SK997-99A SK99799A SK99799A3 SK 99799 A3 SK99799 A3 SK 99799A3 SK 99799 A SK99799 A SK 99799A SK 99799 A3 SK99799 A3 SK 99799A3
Authority
SK
Slovakia
Prior art keywords
group
alkyl
substituted
phenyl
hydrogen
Prior art date
Application number
SK997-99A
Other languages
English (en)
Slovak (sk)
Inventor
Jeanne Maruani
Philippe Soubrie
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of SK99799A3 publication Critical patent/SK99799A3/sk

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
SK997-99A 1997-01-28 1998-01-28 Use of central cannabinoid receptor antagonists for regulating appetence SK99799A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9700870A FR2758723B1 (fr) 1997-01-28 1997-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
PCT/FR1998/000154 WO1998032441A1 (fr) 1997-01-28 1998-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour reguler l'appetance

Publications (1)

Publication Number Publication Date
SK99799A3 true SK99799A3 (en) 2000-06-12

Family

ID=9503028

Family Applications (1)

Application Number Title Priority Date Filing Date
SK997-99A SK99799A3 (en) 1997-01-28 1998-01-28 Use of central cannabinoid receptor antagonists for regulating appetence

Country Status (32)

Country Link
US (3) US6344474B1 (ar)
EP (2) EP0969835B1 (ar)
JP (1) JP3676383B2 (ar)
AR (1) AR011776A1 (ar)
AT (1) ATE358480T1 (ar)
AU (1) AU6219398A (ar)
BR (1) BR9806801A (ar)
CA (1) CA2278661A1 (ar)
DE (1) DE69837473T2 (ar)
DK (1) DK0969835T3 (ar)
DZ (1) DZ2405A1 (ar)
EE (1) EE04630B1 (ar)
ES (1) ES2285760T3 (ar)
FR (1) FR2758723B1 (ar)
GT (1) GT199800021A (ar)
HK (1) HK1022829A1 (ar)
HR (1) HRP980042A2 (ar)
ID (1) ID22216A (ar)
IS (1) IS5113A (ar)
LV (1) LV12354B (ar)
ME (1) MEP26508A (ar)
MY (1) MY117251A (ar)
NO (1) NO323696B1 (ar)
PT (1) PT969835E (ar)
RS (1) RS49830B (ar)
SA (1) SA98181113B1 (ar)
SK (1) SK99799A3 (ar)
TR (1) TR199901721T2 (ar)
TW (1) TW450808B (ar)
UY (1) UY24847A1 (ar)
WO (1) WO1998032441A1 (ar)
ZA (1) ZA98691B (ar)

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EP1795194A2 (fr) 2007-06-13
ATE358480T1 (de) 2007-04-15
BR9806801A (pt) 2000-05-16
SA98181113B1 (ar) 2006-06-25
EP0969835B1 (fr) 2007-04-04
RS49830B (sr) 2008-08-07
ZA98691B (en) 1998-08-05
IS5113A (is) 1999-07-12
EP1795194A3 (fr) 2008-04-30
EE04630B1 (et) 2006-06-15
US6344474B1 (en) 2002-02-05
UY24847A1 (es) 1998-04-21
HK1022829A1 (en) 2000-08-25
JP2001501971A (ja) 2001-02-13
MY117251A (en) 2004-06-30
DE69837473T2 (de) 2007-12-13
JP3676383B2 (ja) 2005-07-27
ES2285760T3 (es) 2007-11-16
LV12354A (lv) 1999-10-20
NO323696B1 (no) 2007-06-25
AU6219398A (en) 1998-08-18
TR199901721T2 (xx) 1999-10-21
AR011776A1 (es) 2000-09-13
CA2278661A1 (en) 1998-07-30
LV12354B (en) 2000-02-20
US20020128302A1 (en) 2002-09-12
DE69837473D1 (de) 2007-05-16
GT199800021A (es) 1999-07-22
WO1998032441A1 (fr) 1998-07-30
YU35099A (sh) 2002-08-12
FR2758723A1 (fr) 1998-07-31
EP0969835A1 (fr) 2000-01-12
DK0969835T3 (da) 2007-08-06
DZ2405A1 (fr) 2003-01-04
NO993634D0 (no) 1999-07-27
PT969835E (pt) 2007-07-12
US20050026986A1 (en) 2005-02-03
MEP26508A (en) 2010-06-10
HRP980042A2 (en) 1998-10-31
ID22216A (id) 1999-09-16
NO993634L (no) 1999-09-27
FR2758723B1 (fr) 1999-04-23
EE9900304A (et) 2000-02-15
TW450808B (en) 2001-08-21

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