SK281195B6 - Spôsob výroby (s)-3-amino-1-substituovaných pyrolidínov a medziprodukty na uvedený spôsob - Google Patents

Spôsob výroby (s)-3-amino-1-substituovaných pyrolidínov a medziprodukty na uvedený spôsob Download PDF

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Publication number
SK281195B6
SK281195B6 SK1298-94A SK129894A SK281195B6 SK 281195 B6 SK281195 B6 SK 281195B6 SK 129894 A SK129894 A SK 129894A SK 281195 B6 SK281195 B6 SK 281195B6
Authority
SK
Slovakia
Prior art keywords
formula
alkyl
compound
amino
defined above
Prior art date
Application number
SK1298-94A
Other languages
English (en)
Slovak (sk)
Other versions
SK129894A3 (en
Inventor
Tung Van Le
F. Gregory Spence
James Norton Wemple
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of SK129894A3 publication Critical patent/SK129894A3/sk
Publication of SK281195B6 publication Critical patent/SK281195B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D203/22—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SK1298-94A 1992-04-27 1993-04-16 Spôsob výroby (s)-3-amino-1-substituovaných pyrolidínov a medziprodukty na uvedený spôsob SK281195B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/874,657 US5177217A (en) 1992-04-27 1992-04-27 Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines
PCT/US1993/003646 WO1993022283A1 (en) 1992-04-27 1993-04-16 Process for the manufacture of (s)-3-amino-1-substituted-pyrrolidines

Publications (2)

Publication Number Publication Date
SK129894A3 SK129894A3 (en) 1995-05-10
SK281195B6 true SK281195B6 (sk) 2001-01-18

Family

ID=25364272

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1298-94A SK281195B6 (sk) 1992-04-27 1993-04-16 Spôsob výroby (s)-3-amino-1-substituovaných pyrolidínov a medziprodukty na uvedený spôsob

Country Status (20)

Country Link
US (1) US5177217A (el)
EP (2) EP0911322A3 (el)
JP (1) JP3264928B2 (el)
KR (1) KR950701316A (el)
AT (1) ATE181549T1 (el)
AU (1) AU666736B2 (el)
CA (1) CA2133091C (el)
CZ (1) CZ285593B6 (el)
DE (1) DE69325452T2 (el)
DK (1) DK0638068T3 (el)
ES (1) ES2135477T3 (el)
FI (1) FI106122B (el)
GR (1) GR3031149T3 (el)
HU (1) HU220603B1 (el)
MX (1) MX9302414A (el)
NO (1) NO300969B1 (el)
NZ (1) NZ252850A (el)
RU (1) RU2101279C1 (el)
SK (1) SK281195B6 (el)
WO (1) WO1993022283A1 (el)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5177217A (en) * 1992-04-27 1993-01-05 Warner-Lambert Company Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines
EP1138672A1 (en) * 1998-01-12 2001-10-04 Basilea Pharmaceutica AG Process for the preparation of 3-amino-pyrrolidine derivatives
US5977381A (en) * 1998-01-12 1999-11-02 Hoffmann-La Roche Inc. Process for making 3-amino-pyrolidine derivatives
EP1125922A1 (en) 1998-11-02 2001-08-22 Welfide Corporation Pyrrolidine compounds and medicinal utilization thereof
US6531594B2 (en) 2000-08-24 2003-03-11 Mitsubishi Chemical Corporation Process for producing 1H-3-aminopyrrolidine and derivatives thereof
WO2003082815A1 (fr) 2002-03-29 2003-10-09 Kaneka Corporation Procede d'amelioration de la purete optique de 1-benzyl-3- aminopyrrolidine et sel utilise dans ce procede
EP1676837A4 (en) * 2003-10-08 2008-09-10 Teijin Pharma Ltd METHOD FOR PRODUCING AN AMINOPYRROLIDINE DERIVATIVE AND AN INTERMEDIATE COMPOUND
TW200630337A (en) 2004-10-14 2006-09-01 Euro Celtique Sa Piperidinyl compounds and the use thereof
US8247442B2 (en) 2006-03-29 2012-08-21 Purdue Pharma L.P. Benzenesulfonamide compounds and their use
WO2007118854A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and the use thereof
US8791264B2 (en) 2006-04-13 2014-07-29 Purdue Pharma L.P. Benzenesulfonamide compounds and their use as blockers of calcium channels
US8399486B2 (en) 2007-04-09 2013-03-19 Purdue Pharma L.P. Benzenesulfonyl compounds and the use thereof
WO2009040659A2 (en) 2007-09-28 2009-04-02 Purdue Pharma L.P. Benzenesulfonamide compounds and the use thereof
CN111620802A (zh) * 2020-06-18 2020-09-04 山西千岫制药有限公司 一种头孢托罗中间体(r)-1-苄基-3-氨基吡咯烷的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4785119A (en) * 1985-10-11 1988-11-15 Tokyo Kasei Kogyo Co., Ltd. 3-aminopyrrolidine compound and process for preparation thereof
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4859776A (en) * 1988-03-11 1989-08-22 Abbott Laboratories (S)-7-(3-aminopyrrolidin-1-yl)-1-(ortho, para-difluorophenyl)-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid and method for its preparation
JP2995704B2 (ja) * 1989-02-17 1999-12-27 東京化成工業株式会社 光学活性な１ｈ−３−アミノピロリジン化合物の製造法
US4916141A (en) * 1989-03-28 1990-04-10 Warner-Lambert Company (S)-7-(3-amino-1-pyrrolidinyl)-1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid
CA2036516A1 (en) * 1990-02-19 1991-08-20 Yoshikazu Asahina Optically active 8-methoxyouinolonecarboxylic acid derivatives, their preparative processes and their intermediates
US5177217A (en) * 1992-04-27 1993-01-05 Warner-Lambert Company Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines

Also Published As

Publication number Publication date
EP0638068B1 (en) 1999-06-23
CA2133091A1 (en) 1993-11-11
CZ285593B6 (cs) 1999-09-15
KR950701316A (ko) 1995-03-23
NZ252850A (en) 1996-10-28
MX9302414A (es) 1993-10-01
US5177217A (en) 1993-01-05
JP3264928B2 (ja) 2002-03-11
AU4289993A (en) 1993-11-29
EP0911322A2 (en) 1999-04-28
NO300969B1 (no) 1997-08-25
FI945000A0 (fi) 1994-10-24
EP0638068A1 (en) 1995-02-15
EP0911322A3 (en) 2001-06-13
GR3031149T3 (en) 1999-12-31
AU666736B2 (en) 1996-02-22
NO944075D0 (no) 1994-10-26
NO944075L (no) 1994-12-27
SK129894A3 (en) 1995-05-10
RU2101279C1 (ru) 1998-01-10
RU94046013A (ru) 1996-10-10
FI106122B (fi) 2000-11-30
HU220603B1 (hu) 2002-03-28
DE69325452D1 (de) 1999-07-29
HUT70218A (en) 1995-09-28
FI945000A (fi) 1994-10-24
CA2133091C (en) 2005-01-04
DK0638068T3 (da) 1999-11-22
JPH07506110A (ja) 1995-07-06
ATE181549T1 (de) 1999-07-15
ES2135477T3 (es) 1999-11-01
WO1993022283A1 (en) 1993-11-11
CZ257694A3 (en) 1995-10-18
DE69325452T2 (de) 2000-05-18

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