DK0638068T3 - Fremgangsmåde til fremstilling af (S)-3-amino-1-substitueret-pyrrolidiner - Google Patents
Fremgangsmåde til fremstilling af (S)-3-amino-1-substitueret-pyrrolidinerInfo
- Publication number
- DK0638068T3 DK0638068T3 DK93912301T DK93912301T DK0638068T3 DK 0638068 T3 DK0638068 T3 DK 0638068T3 DK 93912301 T DK93912301 T DK 93912301T DK 93912301 T DK93912301 T DK 93912301T DK 0638068 T3 DK0638068 T3 DK 0638068T3
- Authority
- DK
- Denmark
- Prior art keywords
- pyrrolidines
- amino
- substituted
- preparation
- propionylaminoü
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/14—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D203/22—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/874,657 US5177217A (en) | 1992-04-27 | 1992-04-27 | Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines |
PCT/US1993/003646 WO1993022283A1 (en) | 1992-04-27 | 1993-04-16 | Process for the manufacture of (s)-3-amino-1-substituted-pyrrolidines |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0638068T3 true DK0638068T3 (da) | 1999-11-22 |
Family
ID=25364272
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK93912301T DK0638068T3 (da) | 1992-04-27 | 1993-04-16 | Fremgangsmåde til fremstilling af (S)-3-amino-1-substitueret-pyrrolidiner |
Country Status (20)
Country | Link |
---|---|
US (1) | US5177217A (da) |
EP (2) | EP0638068B1 (da) |
JP (1) | JP3264928B2 (da) |
KR (1) | KR950701316A (da) |
AT (1) | ATE181549T1 (da) |
AU (1) | AU666736B2 (da) |
CA (1) | CA2133091C (da) |
CZ (1) | CZ285593B6 (da) |
DE (1) | DE69325452T2 (da) |
DK (1) | DK0638068T3 (da) |
ES (1) | ES2135477T3 (da) |
FI (1) | FI106122B (da) |
GR (1) | GR3031149T3 (da) |
HU (1) | HU220603B1 (da) |
MX (1) | MX9302414A (da) |
NO (1) | NO300969B1 (da) |
NZ (1) | NZ252850A (da) |
RU (1) | RU2101279C1 (da) |
SK (1) | SK281195B6 (da) |
WO (1) | WO1993022283A1 (da) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5177217A (en) * | 1992-04-27 | 1993-01-05 | Warner-Lambert Company | Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines |
EP1138672A1 (en) * | 1998-01-12 | 2001-10-04 | Basilea Pharmaceutica AG | Process for the preparation of 3-amino-pyrrolidine derivatives |
US5977381A (en) * | 1998-01-12 | 1999-11-02 | Hoffmann-La Roche Inc. | Process for making 3-amino-pyrolidine derivatives |
EP1125922A1 (en) | 1998-11-02 | 2001-08-22 | Welfide Corporation | Pyrrolidine compounds and medicinal utilization thereof |
US6531594B2 (en) | 2000-08-24 | 2003-03-11 | Mitsubishi Chemical Corporation | Process for producing 1H-3-aminopyrrolidine and derivatives thereof |
JP4481659B2 (ja) | 2002-03-29 | 2010-06-16 | 株式会社カネカ | 1−ベンジル−3−アミノピロリジンの光学純度向上方法及びそれに用いられる塩 |
BRPI0415018A (pt) * | 2003-10-08 | 2006-11-28 | Teijin Pharma Ltd | métodos para a produção de derivados de aminopirrolidina e de antranilamida, e, composto |
TW200630337A (en) | 2004-10-14 | 2006-09-01 | Euro Celtique Sa | Piperidinyl compounds and the use thereof |
US8247442B2 (en) | 2006-03-29 | 2012-08-21 | Purdue Pharma L.P. | Benzenesulfonamide compounds and their use |
TW200815353A (en) | 2006-04-13 | 2008-04-01 | Euro Celtique Sa | Benzenesulfonamide compounds and their use |
WO2007118854A1 (en) | 2006-04-13 | 2007-10-25 | Euro-Celtique S.A. | Benzenesulfonamide compounds and the use thereof |
WO2008124118A1 (en) | 2007-04-09 | 2008-10-16 | Purdue Pharma L.P. | Benzenesulfonyl compounds and the use therof |
US8765736B2 (en) | 2007-09-28 | 2014-07-01 | Purdue Pharma L.P. | Benzenesulfonamide compounds and the use thereof |
CN111620802A (zh) * | 2020-06-18 | 2020-09-04 | 山西千岫制药有限公司 | 一种头孢托罗中间体(r)-1-苄基-3-氨基吡咯烷的制备方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4785119A (en) * | 1985-10-11 | 1988-11-15 | Tokyo Kasei Kogyo Co., Ltd. | 3-aminopyrrolidine compound and process for preparation thereof |
US4851418A (en) * | 1987-08-21 | 1989-07-25 | Warner-Lambert Company | Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent |
US4859776A (en) * | 1988-03-11 | 1989-08-22 | Abbott Laboratories | (S)-7-(3-aminopyrrolidin-1-yl)-1-(ortho, para-difluorophenyl)-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid and method for its preparation |
JP2995704B2 (ja) * | 1989-02-17 | 1999-12-27 | 東京化成工業株式会社 | 光学活性な1h−3−アミノピロリジン化合物の製造法 |
US4916141A (en) * | 1989-03-28 | 1990-04-10 | Warner-Lambert Company | (S)-7-(3-amino-1-pyrrolidinyl)-1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid |
HU208005B (en) * | 1990-02-19 | 1993-07-28 | Kyorin Seiyaku Kk | Process for producing optically active 8-methoxy-quinolone-carboxylic acid derivatives and pharmaceutical compositions containing them |
US5177217A (en) * | 1992-04-27 | 1993-01-05 | Warner-Lambert Company | Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines |
-
1992
- 1992-04-27 US US07/874,657 patent/US5177217A/en not_active Expired - Lifetime
-
1993
- 1993-04-16 CZ CZ942576A patent/CZ285593B6/cs not_active IP Right Cessation
- 1993-04-16 SK SK1298-94A patent/SK281195B6/sk unknown
- 1993-04-16 DK DK93912301T patent/DK0638068T3/da active
- 1993-04-16 CA CA002133091A patent/CA2133091C/en not_active Expired - Fee Related
- 1993-04-16 DE DE69325452T patent/DE69325452T2/de not_active Expired - Fee Related
- 1993-04-16 HU HU9403083A patent/HU220603B1/hu not_active IP Right Cessation
- 1993-04-16 KR KR1019940703802A patent/KR950701316A/ko active IP Right Grant
- 1993-04-16 RU RU94046013/04A patent/RU2101279C1/ru not_active IP Right Cessation
- 1993-04-16 WO PCT/US1993/003646 patent/WO1993022283A1/en active IP Right Grant
- 1993-04-16 ES ES93912301T patent/ES2135477T3/es not_active Expired - Lifetime
- 1993-04-16 NZ NZ252850A patent/NZ252850A/en unknown
- 1993-04-16 AT AT93912301T patent/ATE181549T1/de not_active IP Right Cessation
- 1993-04-16 JP JP51932393A patent/JP3264928B2/ja not_active Expired - Fee Related
- 1993-04-16 AU AU42899/93A patent/AU666736B2/en not_active Ceased
- 1993-04-16 EP EP93912301A patent/EP0638068B1/en not_active Expired - Lifetime
- 1993-04-16 EP EP98121092A patent/EP0911322A3/en not_active Ceased
- 1993-04-26 MX MX9302414A patent/MX9302414A/es not_active IP Right Cessation
-
1994
- 1994-10-24 FI FI945000A patent/FI106122B/fi not_active IP Right Cessation
- 1994-10-26 NO NO944075A patent/NO300969B1/no not_active IP Right Cessation
-
1999
- 1999-09-02 GR GR990402237T patent/GR3031149T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
CZ285593B6 (cs) | 1999-09-15 |
AU4289993A (en) | 1993-11-29 |
NO300969B1 (no) | 1997-08-25 |
GR3031149T3 (en) | 1999-12-31 |
CA2133091A1 (en) | 1993-11-11 |
ATE181549T1 (de) | 1999-07-15 |
EP0638068B1 (en) | 1999-06-23 |
HUT70218A (en) | 1995-09-28 |
NO944075D0 (no) | 1994-10-26 |
AU666736B2 (en) | 1996-02-22 |
JP3264928B2 (ja) | 2002-03-11 |
NZ252850A (en) | 1996-10-28 |
RU2101279C1 (ru) | 1998-01-10 |
KR950701316A (ko) | 1995-03-23 |
ES2135477T3 (es) | 1999-11-01 |
DE69325452T2 (de) | 2000-05-18 |
US5177217A (en) | 1993-01-05 |
HU220603B1 (hu) | 2002-03-28 |
EP0638068A1 (en) | 1995-02-15 |
FI945000A (fi) | 1994-10-24 |
FI106122B (fi) | 2000-11-30 |
EP0911322A3 (en) | 2001-06-13 |
DE69325452D1 (de) | 1999-07-29 |
MX9302414A (es) | 1993-10-01 |
WO1993022283A1 (en) | 1993-11-11 |
FI945000A0 (fi) | 1994-10-24 |
JPH07506110A (ja) | 1995-07-06 |
NO944075L (no) | 1994-12-27 |
SK129894A3 (en) | 1995-05-10 |
RU94046013A (ru) | 1996-10-10 |
EP0911322A2 (en) | 1999-04-28 |
SK281195B6 (sk) | 2001-01-18 |
CZ257694A3 (en) | 1995-10-18 |
CA2133091C (en) | 2005-01-04 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ID30373A (id) | PARAHERKUAMIDA ANTIPARASIT (Pecahan P-962086) | |
DE69133397D1 (de) | Benzoylderivate | |
NO881697D0 (no) | Verktoeyenhet, verktoeydeler og fremgangsmaate for sammensetting av delene. | |
DK0758904T3 (da) | Fremgangsmåder og sammensætninger til behandling af glomerulonephritis | |
ZA919629B (en) | Novel 4-arylpiperazines and 4-arylpiperidines | |
EP0528858A4 (en) | Inhibitors of dipeptidyl-aminopeptidase type iv | |
ATE243694T1 (de) | 4-mercaptoacetylamino-(2)benzazepinon(3)- derivate, und verwendung als enkephalinase- inhibitoren | |
DK0638068T3 (da) | Fremgangsmåde til fremstilling af (S)-3-amino-1-substitueret-pyrrolidiner | |
DK0545511T3 (da) | Fremgangsmåde til fremstilling af mono-N-substiuerede tetraazamakrocycler | |
ATE103594T1 (de) | Fucosidase-inhibitoren. | |
ES2042726T3 (es) | Beta-alquilmelatoninas. | |
NO903338L (no) | Fremgangsmaate for mikrobiologisk fremstilling av l-carnitin. | |
DK0648738T3 (da) | Fremgangsmåde til fremstilling af acetoacetarylamider | |
DK192890D0 (da) | 24r-scumnol, fremgangsmaade til fremstilling heraf samt anvendelse af samme | |
DK0635490T3 (da) | Fremgangsmåde til fremstilling af N-ethylcarbazol | |
FI892051A (fi) | Foerfarande foer framstaellning av 5-klor-3-klorsulfonyl-2-tiofencarbonsyraestrar. | |
DK0730861T3 (da) | Anvendelse af 6,7-substituerede 2-aminotetraliner til fremstilling af farmaceutiske præparater, der er nyttige til behandli | |
ES2051953T3 (es) | Derivados isomeros de trimetilbiciclo(4,3,0)nonano. | |
FI913414A (fi) | Foerfarande foer framstaellning av 2-hydroxi-3-halogen-5-nitropyridiner. | |
DK0582977T3 (da) | Fremgangsmåde til fremstilling af 1,3-dialkyl-5-hydroxyoxindoler og etherderivater deraf | |
TR27159A (tr) | Sübstitüe edilmis 2 -fenil-5-(3-fenoksifelin (1,1,1-trifloropentanlari hazirlamaya mahsus yöntem ve aramaddeler. | |
IT8902129A0 (it) | Esalatore rosa. | |
DK319189D0 (da) | Fremgangsmaade til nedbrydning af uklarhedsdannende vinproteiner |