SI1781683T1 - Postopek za pripravo 17-vinil-triflatov kot intermediatov - Google Patents

Postopek za pripravo 17-vinil-triflatov kot intermediatov

Info

Publication number
SI1781683T1
SI1781683T1 SI200531462T SI200531462T SI1781683T1 SI 1781683 T1 SI1781683 T1 SI 1781683T1 SI 200531462 T SI200531462 T SI 200531462T SI 200531462 T SI200531462 T SI 200531462T SI 1781683 T1 SI1781683 T1 SI 1781683T1
Authority
SI
Slovenia
Prior art keywords
triflates
intermediates
vinyl
preparation
formula
Prior art date
Application number
SI200531462T
Other languages
English (en)
Inventor
Paul Stanley Safc Pharma Bury
Original Assignee
Btg Int Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35311370&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1781683(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0418900.7A external-priority patent/GB0418900D0/en
Priority claimed from GB0418901A external-priority patent/GB0418901D0/en
Application filed by Btg Int Ltd filed Critical Btg Int Ltd
Publication of SI1781683T1 publication Critical patent/SI1781683T1/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyridine Compounds (AREA)
SI200531462T 2004-08-24 2005-08-23 Postopek za pripravo 17-vinil-triflatov kot intermediatov SI1781683T1 (sl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US60355804P 2004-08-24 2004-08-24
GBGB0418900.7A GB0418900D0 (en) 2004-08-24 2004-08-24 Novel salt forms
GB0418901A GB0418901D0 (en) 2004-08-24 2004-08-24 Synthetic method
EP05781067A EP1781683B1 (en) 2004-08-24 2005-08-23 Process for the preparation of 17-vinyl- triflates as intermediates
PCT/GB2005/003283 WO2006021777A1 (en) 2004-08-24 2005-08-23 Process fot the preparation of 17-0-vinyl- triflates as intermediates

Publications (1)

Publication Number Publication Date
SI1781683T1 true SI1781683T1 (sl) 2012-06-29

Family

ID=35311370

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200531462T SI1781683T1 (sl) 2004-08-24 2005-08-23 Postopek za pripravo 17-vinil-triflatov kot intermediatov
SI200531956T SI2428519T1 (sl) 2004-08-24 2005-08-23 Sestavek za pripravo 17-vinil-triflatov kot intermediatov

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200531956T SI2428519T1 (sl) 2004-08-24 2005-08-23 Sestavek za pripravo 17-vinil-triflatov kot intermediatov

Country Status (12)

Country Link
US (2) US8236946B2 (sl)
EP (2) EP2428519B1 (sl)
JP (1) JP5199667B2 (sl)
AT (1) ATE533775T1 (sl)
CY (1) CY1112283T1 (sl)
DK (2) DK2428519T3 (sl)
ES (2) ES2534587T3 (sl)
HK (1) HK1167658A1 (sl)
PL (2) PL1781683T3 (sl)
PT (2) PT1781683E (sl)
SI (2) SI1781683T1 (sl)
WO (1) WO2006021777A1 (sl)

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CN102030798B (zh) * 2010-12-17 2012-10-17 深圳万乐药业有限公司 一种醋酸阿比特龙的纯化方法
ES2590753T3 (es) 2011-10-10 2016-11-23 Zach System Proceso para la preparación de esteroides 17-sustituidos
EP2607371A1 (en) 2011-12-23 2013-06-26 Crystal Pharma, S.A.U. Processes for the preparation of abiraterone and related compouds
CN103172690B (zh) * 2011-12-23 2016-08-24 重庆医药工业研究院有限责任公司 醋酸阿比特龙及其中间体的制备方法
CN105461777B (zh) * 2012-01-04 2017-07-18 连云港润众制药有限公司 一种醋酸阿比特龙的纯化方法
CN103254265B (zh) 2012-02-21 2016-07-13 上海希迈医药科技有限公司 醋酸阿比特龙三氟乙酸盐及其制备方法和应用
US9511152B2 (en) * 2012-04-05 2016-12-06 The Board Of Regents Of The University Of Texas System Multicolored pH-activatable fluorescence nanoplatform
WO2014009437A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Oxidation stability of abiraterone acetate
WO2014009434A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Self-microemulsifying drug delivery system of abiraterone or abiraterone acetate
WO2014009436A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Nanosuspension of abiraterone acetate
WO2014016830A1 (en) * 2012-07-25 2014-01-30 Mapi Pharma Ltd. Process and intermediates for the preparation of abiraterone acetate
CN102816200B (zh) * 2012-09-05 2015-04-15 中山大学 一种醋酸阿比特龙的制备方法
ITMI20121788A1 (it) 2012-10-22 2014-04-23 Olon Spa Procedimento per la purificazione di abiraterone acetato
WO2014071983A1 (en) 2012-11-09 2014-05-15 Synthon Bv Process for making the 17-triflate intermediate of abiraterone-3-acetate
CA2890589A1 (en) 2012-11-09 2014-05-15 Synthon Bv Process for making abiraterone-3-acetate
WO2014075978A1 (en) 2012-11-16 2014-05-22 Synthon B.V. Process for the production of abiraterone-3-acetate involving an enol trliflation reaction in the presence of an alkoxy-pyridine compound
WO2014095833A1 (en) 2012-12-19 2014-06-26 Bayer Pharma Aktiengesellschaft Combination comprising radium-223 for the treatment of cancer
WO2014102833A2 (en) * 2012-12-31 2014-07-03 Hetero Research Foundation Process for abiraterone acetate
EP2792682B1 (en) 2013-04-19 2016-11-09 Zach System Process for producing a solid form of abiraterone acetate
CN103242410B (zh) * 2013-05-09 2015-08-26 苏州明锐医药科技有限公司 醋酸阿比特龙的制备方法
WO2014207762A1 (en) * 2013-06-24 2014-12-31 Sun Pharmaceutical Industries Ltd. Process for preparation of abiraterone acetate
ES2705579T3 (es) * 2013-06-28 2019-03-26 Scinopharm Taiwan Ltd Procedimiento de preparación de abiraterona e intermedios de la misma
EP3027638B1 (en) 2013-07-29 2017-12-27 Industriale Chimica S.R.L. Process for the preparation of abiraterone and abiraterone acetate
ES2581317T3 (es) 2013-07-29 2016-09-05 Industriale Chimica S.R.L. Proceso de preparación de abiraterona o acetato de abiraterona
ITMI20131861A1 (it) * 2013-11-08 2015-05-09 Ind Chimica Srl Processo per la preparazione di abiraterone e abiraterone acetato
CN104418930B (zh) * 2013-08-23 2018-01-12 四川海思科制药有限公司 一种高纯度醋酸乌利司他
US9556219B2 (en) 2014-01-28 2017-01-31 Olon S.P.A. Procedure for the preparation of abiraterone acetate and intermediates thereof
CN103965282B (zh) * 2014-04-21 2016-01-20 武汉百科药物开发有限公司 一种醋酸阿比特龙的制备方法
US9315541B2 (en) 2014-05-20 2016-04-19 Olon S.P.A. Process for the preparation of unsaturated trifluoromethanesulfonate steroid derivatives
WO2016001208A1 (en) 2014-06-30 2016-01-07 Galenicum Health S.L. Stable pharmaceutical compositions in the form of immediate release tablets
CZ2014475A3 (cs) 2014-07-09 2016-01-20 Zentiva, K.S. Způsob přípravy Abirateron acetátu o vysoké čistotě aplikovatelný v průmyslovém měřítku
CN105622703B (zh) * 2014-11-05 2019-09-27 兰州大学 一种制备醋酸阿比特龙的方法
CN104447934B (zh) * 2014-12-08 2017-03-15 深圳科兴生物工程有限公司 一种醋酸阿比特龙的纯化方法
HU231297B1 (hu) 2018-07-31 2022-09-28 Richter Gedeon Nyrt Stabil gyógyszerkészítmények és eljárás az előállításukra
CN112812147A (zh) * 2019-11-15 2021-05-18 江苏佳尔科药业集团股份有限公司 一种醋酸阿比特龙的合成方法及其中间体
EP3944860A1 (en) 2020-07-30 2022-02-02 Galenicum Health S.L.U. Abiraterone for use in a method of treating cancer

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GB0418900D0 (en) * 2004-08-24 2004-09-29 Btg Int Ltd Novel salt forms

Also Published As

Publication number Publication date
EP2428519A2 (en) 2012-03-14
JP5199667B2 (ja) 2013-05-15
PL1781683T3 (pl) 2012-04-30
EP2428519B1 (en) 2015-01-21
HK1167658A1 (en) 2012-12-07
ES2377074T3 (es) 2012-03-22
PT1781683E (pt) 2012-02-13
EP1781683B1 (en) 2011-11-16
JP2008510781A (ja) 2008-04-10
PL2428519T3 (pl) 2015-09-30
US8236946B2 (en) 2012-08-07
US20110288288A1 (en) 2011-11-24
CY1112283T1 (el) 2015-12-09
WO2006021777A1 (en) 2006-03-02
EP1781683A1 (en) 2007-05-09
DK1781683T3 (da) 2012-02-06
US8389714B2 (en) 2013-03-05
DK2428519T3 (en) 2015-04-13
SI2428519T1 (sl) 2015-07-31
US20070282109A1 (en) 2007-12-06
EP2428519A3 (en) 2014-01-15
ATE533775T1 (de) 2011-12-15
ES2534587T3 (es) 2015-04-24
PT2428519E (pt) 2015-04-29

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