DK1781683T3 - Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata - Google Patents

Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata

Info

Publication number
DK1781683T3
DK1781683T3 DK05781067.3T DK05781067T DK1781683T3 DK 1781683 T3 DK1781683 T3 DK 1781683T3 DK 05781067 T DK05781067 T DK 05781067T DK 1781683 T3 DK1781683 T3 DK 1781683T3
Authority
DK
Denmark
Prior art keywords
semi
preparation
finished products
vinyl triflates
formula
Prior art date
Application number
DK05781067.3T
Other languages
English (en)
Inventor
Paul Stanley Bury
Original Assignee
Btg Int Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35311370&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1781683(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0418901A external-priority patent/GB0418901D0/en
Priority claimed from GBGB0418900.7A external-priority patent/GB0418900D0/en
Application filed by Btg Int Ltd filed Critical Btg Int Ltd
Application granted granted Critical
Publication of DK1781683T3 publication Critical patent/DK1781683T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
DK05781067.3T 2004-08-24 2005-08-23 Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata DK1781683T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US60355804P 2004-08-24 2004-08-24
GB0418901A GB0418901D0 (en) 2004-08-24 2004-08-24 Synthetic method
GBGB0418900.7A GB0418900D0 (en) 2004-08-24 2004-08-24 Novel salt forms
PCT/GB2005/003283 WO2006021777A1 (en) 2004-08-24 2005-08-23 Process fot the preparation of 17-0-vinyl- triflates as intermediates

Publications (1)

Publication Number Publication Date
DK1781683T3 true DK1781683T3 (da) 2012-02-06

Family

ID=35311370

Family Applications (2)

Application Number Title Priority Date Filing Date
DK11178005T DK2428519T3 (da) 2004-08-24 2005-08-23 Sammensætning til præparation af 17-vinyl-triflater som intermediater
DK05781067.3T DK1781683T3 (da) 2004-08-24 2005-08-23 Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK11178005T DK2428519T3 (da) 2004-08-24 2005-08-23 Sammensætning til præparation af 17-vinyl-triflater som intermediater

Country Status (12)

Country Link
US (2) US8236946B2 (da)
EP (2) EP1781683B1 (da)
JP (1) JP5199667B2 (da)
AT (1) ATE533775T1 (da)
CY (1) CY1112283T1 (da)
DK (2) DK2428519T3 (da)
ES (2) ES2377074T3 (da)
HK (1) HK1167658A1 (da)
PL (2) PL2428519T3 (da)
PT (2) PT1781683E (da)
SI (2) SI1781683T1 (da)
WO (1) WO2006021777A1 (da)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102030798B (zh) * 2010-12-17 2012-10-17 深圳万乐药业有限公司 一种醋酸阿比特龙的纯化方法
PL2766381T3 (pl) * 2011-10-10 2016-12-30 Sposób wytwarzania steroidów podstawionych w pozycji 17
CN103172690B (zh) * 2011-12-23 2016-08-24 重庆医药工业研究院有限责任公司 醋酸阿比特龙及其中间体的制备方法
EP2607371A1 (en) 2011-12-23 2013-06-26 Crystal Pharma, S.A.U. Processes for the preparation of abiraterone and related compouds
CN103193849B (zh) * 2012-01-04 2016-05-04 连云港润众制药有限公司 一种高纯度醋酸阿比特龙的制备方法
CN103254265B (zh) 2012-02-21 2016-07-13 上海希迈医药科技有限公司 醋酸阿比特龙三氟乙酸盐及其制备方法和应用
US9511152B2 (en) * 2012-04-05 2016-12-06 The Board Of Regents Of The University Of Texas System Multicolored pH-activatable fluorescence nanoplatform
WO2014009434A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Self-microemulsifying drug delivery system of abiraterone or abiraterone acetate
WO2014009437A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Oxidation stability of abiraterone acetate
WO2014009436A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Nanosuspension of abiraterone acetate
EP2877482A4 (en) * 2012-07-25 2016-04-06 Mapi Pharma Ltd PROCESS AND INTERMEDIATES USED IN THE PREPARATION OF ABIRATERONE ACETATE
CN102816200B (zh) * 2012-09-05 2015-04-15 中山大学 一种醋酸阿比特龙的制备方法
ITMI20121788A1 (it) 2012-10-22 2014-04-23 Olon Spa Procedimento per la purificazione di abiraterone acetato
EP2917225A1 (en) 2012-11-09 2015-09-16 Synthon BV Process for making abiraterone-3-acetate
WO2014071983A1 (en) 2012-11-09 2014-05-15 Synthon Bv Process for making the 17-triflate intermediate of abiraterone-3-acetate
WO2014075978A1 (en) 2012-11-16 2014-05-22 Synthon B.V. Process for the production of abiraterone-3-acetate involving an enol trliflation reaction in the presence of an alkoxy-pyridine compound
CA2895356A1 (en) 2012-12-19 2014-06-26 Bayer Pharma Aktiengesellschaft Combination comprising radium-223 for the treatment of cancer
WO2014102833A2 (en) * 2012-12-31 2014-07-03 Hetero Research Foundation Process for abiraterone acetate
ES2612780T3 (es) 2013-04-19 2017-05-18 Zach System Proceso para producir una forma sólida de acetato de abiraterona
CN103242410B (zh) * 2013-05-09 2015-08-26 苏州明锐医药科技有限公司 醋酸阿比特龙的制备方法
JP2016527213A (ja) * 2013-06-24 2016-09-08 サン・ファーマシューティカル・インダストリーズ・リミテッドＳｕｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌ Ｉｎｄｕｓｔｒｉｅｓ Ｌｔｄ． アビラテロン酢酸エステルの製造方法
CN105377871B (zh) * 2013-06-28 2017-06-06 台湾神隆股份有限公司 阿比特龙及其中间体的制备方法
ES2663469T3 (es) 2013-07-29 2018-04-12 Industriale Chimica S.R.L. Proceso para la preparación de abiraterona y acetato de abiraterona
ITMI20131861A1 (it) * 2013-11-08 2015-05-09 Ind Chimica Srl Processo per la preparazione di abiraterone e abiraterone acetato
EP2890705B1 (en) 2013-07-29 2016-04-13 Industriale Chimica S.R.L. Process for the preparation of abiraterone or abiraterone acetate
CN104418930B (zh) * 2013-08-23 2018-01-12 四川海思科制药有限公司 一种高纯度醋酸乌利司他
ES2741505T3 (es) 2014-01-28 2020-02-11 Olon Spa Procedimiento para la preparación de acetato de abiraterona y sus productos intermedios
CN103965282B (zh) * 2014-04-21 2016-01-20 武汉百科药物开发有限公司 一种醋酸阿比特龙的制备方法
US9315541B2 (en) * 2014-05-20 2016-04-19 Olon S.P.A. Process for the preparation of unsaturated trifluoromethanesulfonate steroid derivatives
WO2016001208A1 (en) 2014-06-30 2016-01-07 Galenicum Health S.L. Stable pharmaceutical compositions in the form of immediate release tablets
CZ2014475A3 (cs) 2014-07-09 2016-01-20 Zentiva, K.S. Způsob přípravy Abirateron acetátu o vysoké čistotě aplikovatelný v průmyslovém měřítku
CN105622703B (zh) * 2014-11-05 2019-09-27 兰州大学 一种制备醋酸阿比特龙的方法
CN104447934B (zh) * 2014-12-08 2017-03-15 深圳科兴生物工程有限公司 一种醋酸阿比特龙的纯化方法
HU231297B1 (hu) 2018-07-31 2022-09-28 Richter Gedeon Nyrt Stabil gyógyszerkészítmények és eljárás az előállításukra
CN112812147A (zh) * 2019-11-15 2021-05-18 江苏佳尔科药业集团股份有限公司 一种醋酸阿比特龙的合成方法及其中间体
EP3944860A1 (en) 2020-07-30 2022-02-02 Galenicum Health S.L.U. Abiraterone for use in a method of treating cancer

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4207851A1 (de) * 1992-03-12 1993-09-16 Bayer Ag Mittel und verfahren zur ausruestung von textilien
CA2132449C (en) * 1992-03-31 2002-09-10 Susan E. Barrie 17 - substituted steroids useful in cancer treatment
US5338875A (en) 1992-11-19 1994-08-16 Merck & Co., Inc. Boron containing intermediates useful in the preparation of carbapenems
NZ273367A (en) 1993-09-30 1997-07-27 British Tech Group Preparation of 3<beta>-hydroxy (or lower acyloxy)-16,17-ene-17-(2-pyridyl)-substituted steroids using a palladium complex catalysed cross coupling reaction
US5466770A (en) * 1994-05-26 1995-11-14 Minnesota Mining And Manufacturing Company Fluorine-efficient oil- and water-repellent compositions
JP3982012B2 (ja) * 1997-01-30 2007-09-26 ダイキン工業株式会社 新規組成物および処理剤
US5994334A (en) 1997-02-05 1999-11-30 University Of Maryland Androgen synthesis inhibitors
JP3399286B2 (ja) * 1997-04-11 2003-04-21 ダイキン工業株式会社 防汚加工剤組成物
JPH10316719A (ja) * 1997-05-20 1998-12-02 Daikin Ind Ltd 新規重合体およびそれを含む防汚加工剤組成物
US6059868A (en) * 1998-10-29 2000-05-09 Hewlett-Packard Company Ink-jet inks with improved performance
JP4457497B2 (ja) * 1998-12-22 2010-04-28 ダイキン工業株式会社 撥水撥油剤水性分散液
JP2000212549A (ja) * 1999-01-25 2000-08-02 Asahi Glass Co Ltd 撥水撥油剤組成物およびその製造方法
US6274060B1 (en) * 1999-02-04 2001-08-14 Daikin Industries, Ltd. Water- and oil-repellent
EP1338637A4 (en) * 2000-09-21 2008-03-05 Daikin Ind Ltd AQUEOUS DISPERSION OF WATER AND OLEOFUGE OF ITS MANUFACTURING PROCESS
WO2002064696A1 (fr) * 2001-01-30 2002-08-22 Daikin Industries, Ltd. Composition hydrofuge et oléofuge, procédé de fabrication et utilisation
US7217760B2 (en) * 2001-03-09 2007-05-15 Daikin Industries, Ltd. Water-and-oil repellant composition with improved suitability for cold cure
KR100889714B1 (ko) * 2001-04-13 2009-03-23 아사히 가라스 가부시키가이샤 발수발유제 조성물
WO2003062347A1 (fr) * 2002-01-21 2003-07-31 Daikin Industries, Ltd. Dispersion aqueuse impermeabilisante eau et huile
AU2003244320A1 (en) * 2002-06-20 2004-01-06 Kyowa Hakko Kogyo Co., Ltd. Process for production of vinyl perfluoroalkanesulfonate derivatives
WO2004035708A1 (ja) * 2002-10-15 2004-04-29 Asahi Glass Company, Limited 撥水撥油剤組成物
GB0418900D0 (en) * 2004-08-24 2004-09-29 Btg Int Ltd Novel salt forms

Also Published As

Publication number Publication date
JP2008510781A (ja) 2008-04-10
US8389714B2 (en) 2013-03-05
SI1781683T1 (sl) 2012-06-29
SI2428519T1 (sl) 2015-07-31
US20070282109A1 (en) 2007-12-06
US8236946B2 (en) 2012-08-07
PT2428519E (pt) 2015-04-29
US20110288288A1 (en) 2011-11-24
ATE533775T1 (de) 2011-12-15
EP2428519B1 (en) 2015-01-21
DK2428519T3 (da) 2015-04-13
WO2006021777A1 (en) 2006-03-02
EP1781683A1 (en) 2007-05-09
EP2428519A2 (en) 2012-03-14
ES2377074T3 (es) 2012-03-22
EP1781683B1 (en) 2011-11-16
HK1167658A1 (en) 2012-12-07
JP5199667B2 (ja) 2013-05-15
PT1781683E (pt) 2012-02-13
EP2428519A3 (en) 2014-01-15
CY1112283T1 (el) 2015-12-09
PL2428519T3 (pl) 2015-09-30
ES2534587T3 (es) 2015-04-24
PL1781683T3 (pl) 2012-04-30

Similar Documents

Publication Publication Date Title
DK1781683T3 (da) Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata
RS51341B (en) INTERMEDIATE COMPOUNDS FOR THE TRANS-5-CHLOR-2-METHYL-2,3A, 12B-TETRAHYDRO-1H-DIBENZE [2,3; 6,7] OXEPINO [4,5-C] Pyrrole
ATE497957T1 (de) Pyridinderivate als fungizide verbindungen
BRPI0516911A (pt) método para a preparação de um composto e composto de anilina
DK1740544T3 (da) 2 pyridinylcycloalkylcarboxamidderivater, der er egnede som fungicider
BRPI0411268C8 (pt) Processo para a preparação de compostos 3-aril butil-amina substituído
EA200701470A1 (ru) Способы получения производных 4-(фенокси-5-метилпиримидин-4-илокси)пиперидин-1-карбоновой кислоты и родственных соединений
IS7978A (is) Aðferð til að framleiða súr viðbótarsölt af fjölsýrðum basískum samböndum
DK1907396T3 (da) Fremgangsmåde til fremstilling af 4-beta-amino-4&#39;-demethyl-4-deoxypodophyllotoxin
BR0308345A (pt) Processo para derivados de ácido trans-4-amino-1-cicloexanocarboxìlico
NO20040388L (no) Fremgangsmåte for fremstilling av beraprost og salter derav, samt forbindelser som er mellomprodukter i fremgangsmåten
EA200700767A1 (ru) Способ получения пиразолов
DE602006014001D1 (de) Herstellung von 2-aminothiazol-5-carbonsäurederivaten
BR0315112A (pt) Sal de adição ácido, e, processo para a preparação de um composto
DE502006005865D1 (de) Herstellung von 1,7` -dimethyl-2` -propyl-2,5` -bi-1h-benzimidazol
DE602006015458D1 (de) Verfahren zur herstellung eines carbonsäureamidderivats
EA200500688A1 (ru) Новый способ получения синтетических промежуточных соединений для пестицидов
DK1272480T3 (da) Fremgangsmåde til fremstilling af spirocycliske tetronsyrederivater
WO2007143014A3 (en) Methods for preparing glutamic acid derivatives and intermediates thereof
NO330965B1 (no) Fremgangsmate for fremstilling av substituerte imidazolderivater, mellomprodukter anvendt i fremgangsmaten samt fremgangsmate for fremstilling av mellomprodukt
BRPI0400141A (pt) Composição de incenso inseticida, e emulsão e processo para produção da mesma
CY1106126T1 (el) Μεθοδος δια την παρασκευην ενωσεων 2-(4-αλκυλο-1-πιπepαζινυλο)-βενζαλδεϋδης και-βενζυλιδενυλιου δια νουκλεοφιλικης αρωματικης υποκαταστασεως 2-φθοροβενζαλδεϋδης δια 4-αλκυλο-1-πιπepαζινης, εις υδωρ ως διαλυτην
DE602007012989D1 (de) Verfahren zur Herstellung von Entacapon
ATE522499T1 (de) Verfahren zur herstellung von tamsulosin und seinen derivaten
BR0205408A (pt) Método de produção de um composto de 2,6-diclorofenol