SG182187A1 - 5-heteroaryl substituted indazoles as kinase inhibitors - Google Patents
5-heteroaryl substituted indazoles as kinase inhibitors Download PDFInfo
- Publication number
- SG182187A1 SG182187A1 SG2012043113A SG2012043113A SG182187A1 SG 182187 A1 SG182187 A1 SG 182187A1 SG 2012043113 A SG2012043113 A SG 2012043113A SG 2012043113 A SG2012043113 A SG 2012043113A SG 182187 A1 SG182187 A1 SG 182187A1
- Authority
- SG
- Singapore
- Prior art keywords
- indazol
- benzyl
- triazol
- carboxamide
- indazole
- Prior art date
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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Applications Claiming Priority (1)
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US8546404B2 (en) | 2005-12-13 | 2013-10-01 | Merck Sharp & Dohme | Compounds that are ERK inhibitors |
EP1984331B1 (en) | 2006-02-16 | 2010-10-20 | Schering Corporation | Pyrrolidine derivatives as erk inhibitors |
US8648069B2 (en) * | 2007-06-08 | 2014-02-11 | Abbvie Inc. | 5-substituted indazoles as kinase inhibitors |
US20110301155A1 (en) * | 2007-06-19 | 2011-12-08 | Tsuneo Yasuma | Indazole compounds for activating glucokinase |
AU2008276512A1 (en) | 2007-07-17 | 2009-01-22 | Amgen Inc. | Thiadiazole modulators of PKB |
AU2008276521B2 (en) | 2007-07-17 | 2011-11-03 | Amgen Inc. | Heterocyclic modulators of PKB |
JPWO2009028543A1 (ja) * | 2007-08-30 | 2010-12-02 | 武田薬品工業株式会社 | 置換ピラゾール誘導体 |
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2009
- 2009-11-24 IL IL202318A patent/IL202318A0/en unknown
- 2009-12-04 ZA ZA2009/08624A patent/ZA200908624B/en unknown
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2013
- 2013-12-25 JP JP2013266989A patent/JP2014074057A/ja active Pending
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EP2167491A1 (en) | 2010-03-31 |
CA2689117A1 (en) | 2008-12-18 |
JP2010529137A (ja) | 2010-08-26 |
KR20100032886A (ko) | 2010-03-26 |
JP2014074057A (ja) | 2014-04-24 |
RU2009149696A (ru) | 2011-07-20 |
RU2487873C2 (ru) | 2013-07-20 |
CN101790526A (zh) | 2010-07-28 |
MX2009013213A (es) | 2010-03-30 |
JP5451602B2 (ja) | 2014-03-26 |
WO2008154241A1 (en) | 2008-12-18 |
ZA200908624B (en) | 2015-08-26 |
AU2008262038A1 (en) | 2008-12-18 |
IL202318A0 (en) | 2010-06-30 |
BRPI0811065A2 (pt) | 2014-12-02 |
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