ZA200908624B - 5-heteroaryl substituted indazoles as kinase inhibitors - Google Patents
5-heteroaryl substituted indazoles as kinase inhibitorsInfo
- Publication number
- ZA200908624B ZA200908624B ZA2009/08624A ZA200908624A ZA200908624B ZA 200908624 B ZA200908624 B ZA 200908624B ZA 2009/08624 A ZA2009/08624 A ZA 2009/08624A ZA 200908624 A ZA200908624 A ZA 200908624A ZA 200908624 B ZA200908624 B ZA 200908624B
- Authority
- ZA
- South Africa
- Prior art keywords
- kinase inhibitors
- heteroaryl substituted
- substituted indazoles
- indazoles
- heteroaryl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Public Health (AREA)
- Engineering & Computer Science (AREA)
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- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
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- Endocrinology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Pulmonology (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Communicable Diseases (AREA)
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- Psychology (AREA)
- Dermatology (AREA)
- Gynecology & Obstetrics (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US93396007P | 2007-06-08 | 2007-06-08 | |
PCT/US2008/065727 WO2008154241A1 (en) | 2007-06-08 | 2008-06-04 | 5-heteroaryl substituted indazoles as kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA200908624B true ZA200908624B (en) | 2015-08-26 |
Family
ID=39951673
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA2009/08624A ZA200908624B (en) | 2007-06-08 | 2009-12-04 | 5-heteroaryl substituted indazoles as kinase inhibitors |
Country Status (13)
Country | Link |
---|---|
EP (1) | EP2167491A1 (en) |
JP (2) | JP5451602B2 (en) |
KR (1) | KR20100032886A (en) |
CN (1) | CN101790526A (en) |
AU (1) | AU2008262038A1 (en) |
BR (1) | BRPI0811065A2 (en) |
CA (1) | CA2689117A1 (en) |
IL (1) | IL202318A0 (en) |
MX (1) | MX2009013213A (en) |
RU (1) | RU2487873C2 (en) |
SG (1) | SG182187A1 (en) |
WO (1) | WO2008154241A1 (en) |
ZA (1) | ZA200908624B (en) |
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EP2157859A4 (en) * | 2007-06-19 | 2011-01-12 | Takeda Pharmaceutical | Indazole compounds for activating glucokinase |
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US7919504B2 (en) | 2007-07-17 | 2011-04-05 | Amgen Inc. | Thiadiazole modulators of PKB |
EP2194045A4 (en) * | 2007-08-30 | 2011-09-21 | Takeda Pharmaceutical | Substituted pyrazole derivative |
RU2525389C2 (en) | 2008-02-21 | 2014-08-10 | Мерк Шарп И Доум Корп. | Compounds which are erk inhibitors |
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ES2548141T3 (en) * | 2008-11-20 | 2015-10-14 | Glaxosmithkline Llc | Chemical compounds |
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CN102675286B (en) * | 2011-03-07 | 2015-08-19 | 中国科学院上海药物研究所 | One class indazole compounds and preparation method thereof, purposes and pharmaceutical composition |
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KR20140130124A (en) * | 2012-02-21 | 2014-11-07 | 아지엔드 키미쉐 리유나이트 안젤리니 프란체스코 에이.씨.알.에이.에프. 에스.피.에이 | 1H-Indazole-3-Carboxamide Compounds as Glycogen Synthase Kinase 3 Beta Inhibitors |
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KR20100032886A (en) | 2010-03-26 |
EP2167491A1 (en) | 2010-03-31 |
MX2009013213A (en) | 2010-03-30 |
SG182187A1 (en) | 2012-07-30 |
BRPI0811065A2 (en) | 2014-12-02 |
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