SG10201505606QA - Compounds and methods for kinase modulation, and indications therefor - Google Patents
Compounds and methods for kinase modulation, and indications thereforInfo
- Publication number
- SG10201505606QA SG10201505606QA SG10201505606QA SG10201505606QA SG10201505606QA SG 10201505606Q A SG10201505606Q A SG 10201505606QA SG 10201505606Q A SG10201505606Q A SG 10201505606QA SG 10201505606Q A SG10201505606Q A SG 10201505606QA SG 10201505606Q A SG10201505606Q A SG 10201505606QA
- Authority
- SG
- Singapore
- Prior art keywords
- compounds
- methods
- kinase modulation
- indications therefor
- indications
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P9/00—Drugs for disorders of the cardiovascular system
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Oncology (AREA)
- Obesity (AREA)
- Vascular Medicine (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Transplantation (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32662610P | 2010-04-21 | 2010-04-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG10201505606QA true SG10201505606QA (en) | 2015-08-28 |
Family
ID=44816304
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG10201505606QA SG10201505606QA (en) | 2010-04-21 | 2011-04-20 | Compounds and methods for kinase modulation, and indications therefor |
SG2012076584A SG184874A1 (en) | 2010-04-21 | 2011-04-20 | Compounds and methods for kinase modulation, and indications therefor |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG2012076584A SG184874A1 (en) | 2010-04-21 | 2011-04-20 | Compounds and methods for kinase modulation, and indications therefor |
Country Status (37)
Country | Link |
---|---|
US (3) | US8901118B2 (de) |
EP (1) | EP2560972B1 (de) |
JP (2) | JP5808793B2 (de) |
KR (1) | KR101799126B1 (de) |
CN (1) | CN102947305B (de) |
AR (2) | AR080940A1 (de) |
AU (1) | AU2011242778B2 (de) |
BR (1) | BR112012026927A2 (de) |
CA (1) | CA2796998C (de) |
CL (1) | CL2012002937A1 (de) |
CO (1) | CO6620045A2 (de) |
CR (1) | CR20120536A (de) |
CY (1) | CY1120554T1 (de) |
DK (1) | DK2560972T3 (de) |
EA (1) | EA028105B1 (de) |
EC (1) | ECSP12012245A (de) |
ES (1) | ES2641643T3 (de) |
GE (1) | GEP20156251B (de) |
HR (1) | HRP20171660T1 (de) |
HU (1) | HUE036461T2 (de) |
IL (1) | IL222498A (de) |
LT (1) | LT2560972T (de) |
MA (1) | MA34229B1 (de) |
MX (1) | MX336056B (de) |
MY (1) | MY160780A (de) |
NZ (2) | NZ703538A (de) |
PE (1) | PE20130240A1 (de) |
PL (1) | PL2560972T3 (de) |
PT (1) | PT2560972T (de) |
RS (1) | RS56588B1 (de) |
SG (2) | SG10201505606QA (de) |
SI (1) | SI2560972T1 (de) |
TW (2) | TWI619713B (de) |
UA (1) | UA109128C2 (de) |
UY (1) | UY33346A (de) |
WO (1) | WO2011133637A2 (de) |
ZA (1) | ZA201207898B (de) |
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PT2350075E (pt) | 2008-09-22 | 2014-06-09 | Array Biopharma Inc | Compostos imidazo[1,2b]piridazina substituídos como inibidores da trk cinase |
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EP2694509B1 (de) | 2011-04-05 | 2016-05-18 | Pfizer Limited | Pyrrolo[2,3-d]pyrimidinderivate als inhibitoren von tropomyosin-verwandten kinasen |
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