RU2696310C1 - Бициклические гетероциклические соединения и их применение в терапии - Google Patents

Бициклические гетероциклические соединения и их применение в терапии Download PDF

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RU2696310C1
RU2696310C1 RU2016129472A RU2016129472A RU2696310C1 RU 2696310 C1 RU2696310 C1 RU 2696310C1 RU 2016129472 A RU2016129472 A RU 2016129472A RU 2016129472 A RU2016129472 A RU 2016129472A RU 2696310 C1 RU2696310 C1 RU 2696310C1
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methyl
compound
pyrrolo
formula
pyridin
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RU2016129472A
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Russian (ru)
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RU2016129472A (ru
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Джанни ЧЕЗЗАРИ
Кристофер Норберт Джонсон
Стивен ГОВАРД
Джеймс Эдвард Харви ДЭЙ
Илдико Мария БАК
Шарлотт Мэри ГРИФФИТС-ДЖОУНЗ
Гордон Саксти
Эмилиано ТАМАНИНИ
Никола Элизабет УИЛШЕР
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Астекс Терапьютикс Лимитед
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Priority claimed from GBGB1322755.8A external-priority patent/GB201322755D0/en
Priority claimed from GB201406986A external-priority patent/GB201406986D0/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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RU2016129472A 2013-12-20 2014-12-19 Бициклические гетероциклические соединения и их применение в терапии RU2696310C1 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB1322755.8A GB201322755D0 (en) 2013-12-20 2013-12-20 Bicyclic heterocycle compounds and their uses in therapy
GB1322755.8 2013-12-20
GB201406986A GB201406986D0 (en) 2014-04-17 2014-04-17 Bicyclic heterocycle compounds and their uses in therapy
GB1406986.8 2014-04-17
PCT/GB2014/053778 WO2015092420A1 (en) 2013-12-20 2014-12-19 Bicyclic heterocycle compounds and their uses in therapy

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RU2016129472A RU2016129472A (ru) 2018-01-25
RU2696310C1 true RU2696310C1 (ru) 2019-08-01

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EP (2) EP3083616B1 (enExample)
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RU (1) RU2696310C1 (enExample)
SA (1) SA516371360B1 (enExample)
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