RU2118527C1 - Фармацевтическая композиция, содержащая алкилсульфонамид-агонист 5ht1, для ректального введения - Google Patents

Фармацевтическая композиция, содержащая алкилсульфонамид-агонист 5ht1, для ректального введения Download PDF

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Publication number
RU2118527C1
RU2118527C1 RU94046069/14A RU94046069A RU2118527C1 RU 2118527 C1 RU2118527 C1 RU 2118527C1 RU 94046069/14 A RU94046069/14 A RU 94046069/14A RU 94046069 A RU94046069 A RU 94046069A RU 2118527 C1 RU2118527 C1 RU 2118527C1
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RU
Russia
Prior art keywords
methyl
active ingredient
indole
composition
composition according
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RU94046069/14A
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English (en)
Russian (ru)
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RU94046069A (ru
Inventor
Мерле Надин (FR)
Мерле Надин
Ришар Изабелль (FR)
Ришар Изабелль
Тиелеман Изабелль (FR)
Тиелеман Изабелль
Original Assignee
Лаборатуар Глаксо С.А.
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Application filed by Лаборатуар Глаксо С.А. filed Critical Лаборатуар Глаксо С.А.
Publication of RU94046069A publication Critical patent/RU94046069A/ru
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Publication of RU2118527C1 publication Critical patent/RU2118527C1/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
RU94046069/14A 1992-05-07 1993-05-03 Фармацевтическая композиция, содержащая алкилсульфонамид-агонист 5ht1, для ректального введения RU2118527C1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions
GB9209882.1 1992-05-07

Publications (2)

Publication Number Publication Date
RU94046069A RU94046069A (ru) 1997-11-27
RU2118527C1 true RU2118527C1 (ru) 1998-09-10

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
RU94046069/14A RU2118527C1 (ru) 1992-05-07 1993-05-03 Фармацевтическая композиция, содержащая алкилсульфонамид-агонист 5ht1, для ректального введения

Country Status (33)

Country Link
US (1) US5705506A (enExample)
EP (1) EP0639072B1 (enExample)
JP (1) JPH07506570A (enExample)
KR (1) KR100253111B1 (enExample)
AT (1) ATE163850T1 (enExample)
AU (1) AU670083B2 (enExample)
BE (1) BE1007024A5 (enExample)
BG (1) BG62120B1 (enExample)
BR (1) BR1100108A (enExample)
CA (1) CA2135179C (enExample)
CH (1) CH685920A5 (enExample)
CY (1) CY2039B1 (enExample)
CZ (1) CZ283512B6 (enExample)
DE (1) DE69317418T2 (enExample)
ES (1) ES2113533T3 (enExample)
FR (1) FR2690847B1 (enExample)
GB (2) GB9209882D0 (enExample)
GR (1) GR3026584T3 (enExample)
HK (1) HK95697A (enExample)
HU (2) HU227338B1 (enExample)
IE (1) IE75203B1 (enExample)
IL (1) IL105468A (enExample)
IT (1) IT1261471B (enExample)
NO (1) NO306700B1 (enExample)
NZ (1) NZ252132A (enExample)
OA (1) OA10109A (enExample)
RO (1) RO112993B1 (enExample)
RU (1) RU2118527C1 (enExample)
SG (1) SG46649A1 (enExample)
TW (1) TW231970B (enExample)
UA (1) UA37206C2 (enExample)
WO (1) WO1993021916A1 (enExample)
ZA (1) ZA933178B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2423360C2 (ru) * 2005-10-14 2011-07-10 Атерсис, Инк. Производные индола как ингибиторы н3-рецептора гистамина для лечения когнитивных расстройств и нарушений сна, ожирения и других расстройств центральной нервной системы

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2434297A (en) * 1996-05-23 1997-12-09 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
ME00189B (me) * 1998-03-26 2011-02-10 Astellas Pharma Inc Preparati sa neprekidnim oslobađanjem
AU3731400A (en) * 1999-03-05 2000-09-21 Trustees Of University Technology Corporation, The Methods and compositions useful in inhibiting apoptosis
SI2124556T1 (sl) 2006-10-09 2015-01-30 Charleston Laboratories, Inc. Farmacevtske sestave
EP3090743A1 (en) 2008-01-09 2016-11-09 Charleston Laboratories, Inc. Pharmaceutical compositions for treating headache and eliminating nausea
CA2767576C (en) 2009-07-08 2020-03-10 Charleston Laboratories Inc. Pharmaceutical compositions comprising an antiemetic and an opioid analgesic
SI2627328T1 (sl) 2010-10-15 2017-01-31 Contera Pharma Aps Kombinacije agonistov receptorjev serotonina za zdravljenje motenj premikanja
CN104411301B (zh) 2012-04-18 2018-02-06 康特拉医药公司 适于改善运动障碍治疗的口服药物配方
CA3055170A1 (en) 2016-03-04 2017-09-08 Charleston Laboratories, Inc. Pharmaceutical compositions
AU2017297718B2 (en) 2016-07-11 2023-06-08 Contera Pharma A/S Pulsatile drug delivery system for treating morning akinesia

Family Cites Families (12)

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SE454777B (sv) * 1980-08-12 1988-05-30 Glaxo Group Ltd 5-substituerade 3-aminoalkyl-1h-indoler, forfarande for framstellning av dessa och en farmaceutisk komposition for behandling av migren
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
GB8332435D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
IT1181741B (it) * 1984-12-04 1987-09-30 Glaxo Group Ltd Derivati di indolo,procedimento per prepararli e composizioni farmaceutiche che li contengono
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
US4833153A (en) * 1985-11-08 1989-05-23 Glaxo Group Limited Indole derivatives
AU611469B2 (en) * 1987-08-13 1991-06-13 Glaxo Group Limited Indole derivatives
PT97888B (pt) * 1990-06-07 1998-12-31 Zeneca Ltd Processo para a preparacao de compostos heterociclicos derivados de indol e de composicoes farmaceuticas que os contem

Non-Patent Citations (1)

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Title
US, 5037845 А (Glaxo groop Limited), 06.08.91, A 61 K 31/40. EP, 0303507 А2 (Glaxo Groop Limited),15.02.89, A 61 K 31/445. SU, 1498386 А3 (Глексо Групп лимитед), C 07 D 209/16, 30.07.89. *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2423360C2 (ru) * 2005-10-14 2011-07-10 Атерсис, Инк. Производные индола как ингибиторы н3-рецептора гистамина для лечения когнитивных расстройств и нарушений сна, ожирения и других расстройств центральной нервной системы

Also Published As

Publication number Publication date
HU211638A9 (en) 1995-12-28
HK95697A (en) 1997-08-08
EP0639072B1 (en) 1998-03-11
ITRM930286A0 (it) 1993-05-06
RO112993B1 (ro) 1998-03-30
GB9209882D0 (en) 1992-06-24
IL105468A0 (en) 1993-08-18
AU670083B2 (en) 1996-07-04
EP0639072A1 (en) 1995-02-22
WO1993021916A1 (en) 1993-11-11
ITRM930286A1 (it) 1994-11-06
ZA933178B (en) 1994-01-10
HUT71418A (en) 1995-11-28
TW231970B (enExample) 1994-10-11
CH685920A5 (fr) 1995-11-15
GB9309209D0 (en) 1993-06-16
ATE163850T1 (de) 1998-03-15
NO944214L (no) 1994-11-07
OA10109A (en) 1996-12-18
KR100253111B1 (en) 2000-07-01
BE1007024A5 (fr) 1995-02-21
AU4064093A (en) 1993-11-29
DE69317418T2 (de) 1998-07-30
SG46649A1 (en) 1998-02-20
UA37206C2 (uk) 2001-05-15
FR2690847A1 (fr) 1993-11-12
BG62120B1 (bg) 1999-03-31
CA2135179A1 (en) 1993-11-11
GR3026584T3 (en) 1998-07-31
US5705506A (en) 1998-01-06
JPH07506570A (ja) 1995-07-20
IE930339A1 (en) 1993-11-17
NO306700B1 (no) 1999-12-13
CZ283512B6 (cs) 1998-04-15
HU227338B1 (en) 2011-04-28
DE69317418D1 (de) 1998-04-16
IE75203B1 (en) 1997-08-27
BR1100108A (pt) 1999-12-07
NZ252132A (en) 1996-09-25
GB2266665A (en) 1993-11-10
GB2266665B (en) 1996-05-22
CA2135179C (en) 2000-12-05
ES2113533T3 (es) 1998-05-01
NO944214D0 (no) 1994-11-04
CZ272394A3 (en) 1995-10-18
IL105468A (en) 1998-09-24
FR2690847B1 (fr) 1995-06-09
BG99167A (bg) 1995-06-30
IT1261471B (it) 1996-05-23
CY2039B1 (en) 1998-04-30

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Effective date: 20040504