RU2079303C1 - Лекарственное средство в виде мази для лечения и/или профилактики кожных болезней и кожных проявлений иммунологически опосредованных заболеваний и способ его получения - Google Patents

Лекарственное средство в виде мази для лечения и/или профилактики кожных болезней и кожных проявлений иммунологически опосредованных заболеваний и способ его получения Download PDF

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Publication number
RU2079303C1
RU2079303C1 SU5001707/14A SU5001707A RU2079303C1 RU 2079303 C1 RU2079303 C1 RU 2079303C1 SU 5001707/14 A SU5001707/14 A SU 5001707/14A SU 5001707 A SU5001707 A SU 5001707A RU 2079303 C1 RU2079303 C1 RU 2079303C1
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Russia
Prior art keywords
group
hydrogen
hydroxy
ointment
compound
Prior art date
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SU5001707/14A
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English (en)
Russian (ru)
Inventor
Асакура Сотоо
Jp]
Мураками Йосио
Канагава Нобуто
Накате Тосиоми
Original Assignee
Фудзисава Фармасьютикалз Ко., Лтд.
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Transplantation (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SU5001707/14A 1990-09-04 1991-09-03 Лекарственное средство в виде мази для лечения и/или профилактики кожных болезней и кожных проявлений иммунологически опосредованных заболеваний и способ его получения RU2079303C1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP23517790 1990-09-04
JP235177/1990 1990-09-04

Publications (1)

Publication Number Publication Date
RU2079303C1 true RU2079303C1 (ru) 1997-05-20

Family

ID=16982211

Family Applications (1)

Application Number Title Priority Date Filing Date
SU5001707/14A RU2079303C1 (ru) 1990-09-04 1991-09-03 Лекарственное средство в виде мази для лечения и/или профилактики кожных болезней и кожных проявлений иммунологически опосредованных заболеваний и способ его получения

Country Status (20)

Country Link
US (1) US5385907A (cg-RX-API-DMAC7.html)
EP (1) EP0474126B1 (cg-RX-API-DMAC7.html)
JP (1) JP2526752B2 (cg-RX-API-DMAC7.html)
KR (1) KR100194240B1 (cg-RX-API-DMAC7.html)
CN (1) CN1069193C (cg-RX-API-DMAC7.html)
AT (1) ATE150304T1 (cg-RX-API-DMAC7.html)
AU (1) AU656145B2 (cg-RX-API-DMAC7.html)
CA (1) CA2050623C (cg-RX-API-DMAC7.html)
DE (1) DE69125230T2 (cg-RX-API-DMAC7.html)
DK (1) DK0474126T3 (cg-RX-API-DMAC7.html)
ES (1) ES2099112T3 (cg-RX-API-DMAC7.html)
GR (1) GR3022883T3 (cg-RX-API-DMAC7.html)
HK (1) HK1000006A1 (cg-RX-API-DMAC7.html)
HU (2) HUT59002A (cg-RX-API-DMAC7.html)
IE (1) IE913085A1 (cg-RX-API-DMAC7.html)
PH (1) PH31282A (cg-RX-API-DMAC7.html)
PT (1) PT98862B (cg-RX-API-DMAC7.html)
RU (1) RU2079303C1 (cg-RX-API-DMAC7.html)
SG (1) SG46547A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA916983B (cg-RX-API-DMAC7.html)

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RU2149635C1 (ru) * 1998-02-27 2000-05-27 Пермская государственная медицинская академия Способ лечения аллергических дерматитов
RU2183113C1 (ru) * 2001-06-28 2002-06-10 Новицкий Юрий Алексеевич Средство-гидросульфат графита и способ лечения больных с доброкачественными и злокачественными опухолями кожи (варианты)
RU2231359C1 (ru) * 2002-12-11 2004-06-27 Государственное образовательное учреждение высшего профессионального образования Московская медицинская академия им. И.М.Сеченова Способ лечения язвенных форм ангиитов кожи
RU2414220C2 (ru) * 2005-10-05 2011-03-20 Мицубиси Танабе Фарма Корпорейшн Средство для лечения дерматита
RU2538680C2 (ru) * 2013-03-12 2015-01-10 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Фармацевтическая композиция для лечения атопического дерматита и способ ее получения
RU2553600C2 (ru) * 2013-05-16 2015-06-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Фармацевтическая композиция для лечения заболеваний кожи

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JPH06345646A (ja) * 1993-06-08 1994-12-20 Fujisawa Pharmaceut Co Ltd ローション剤
AU735106B2 (en) * 1994-10-26 2001-06-28 Novartis Ag Pharmaceutical compositions
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DE19549794B4 (de) * 1994-10-26 2009-07-30 Novartis Ag Pharmazeutische Zusammensetzungen
JP4155593B2 (ja) * 1994-10-26 2008-09-24 ノバルティス・アクチエンゲゼルシャフト 医薬組成物
GB2327610B (en) * 1994-11-04 1999-06-02 Novartis Ag Macrolide compositions
AR004480A1 (es) * 1995-04-06 1998-12-16 Amico Derin C D Compuestos de ascomicina que poseen actividad antiinflamatoria, pro cedimiento para prepararlos, uso de dichos compuestos para preparar agentesfarmaceuticos y composiciones farmaceuticas que los incluyen
US5993787A (en) * 1996-09-13 1999-11-30 Johnson & Johnson Consumer Products, Inc. Composition base for topical therapeutic and cosmetic preparations
AU5340298A (en) * 1996-12-27 1998-07-31 Takeda Chemical Industries Ltd. Stabilized tricyclic compound
TW450810B (en) * 1997-02-20 2001-08-21 Fujisawa Pharmaceutical Co Macrolides antibiotic pharmaceutical composition for preventing and treating skin diseases
GB9723669D0 (en) * 1997-11-07 1998-01-07 Univ Aberdeen Skin penetration enhancing components
TR200003108T2 (tr) * 1998-04-27 2001-02-21 Fujisawa Pharmaceutical Co., Ltd. İlaç kompozisyonları
GB9817064D0 (en) * 1998-08-05 1998-10-07 Fujisawa Pharmaceutical Co New use
US6307049B1 (en) 1998-09-30 2001-10-23 The Procter & Gamble Co. Heterocyclic 2-substituted ketoamides
US6300341B1 (en) 1998-09-30 2001-10-09 The Procter & Gamble Co. 2-substituted heterocyclic sulfonamides
GB9826656D0 (en) 1998-12-03 1999-01-27 Novartis Ag Organic compounds
AUPR529701A0 (en) * 2001-05-28 2001-06-21 Fujisawa Pharmaceutical Co., Ltd. Pharmaceutical composition
WO2003004098A1 (en) 2001-07-06 2003-01-16 Sucampo Ag Composition for topical administration comprising an interleukin-2 inhibitor and an antimicrobial agent
AR038628A1 (es) * 2002-03-04 2005-01-19 Novartis Ag Composicion oftalmica
CN1674868B (zh) * 2002-07-23 2010-09-29 诺瓦提斯公司 包含药物、软膏基质和增溶剂/分散剂的眼用软膏剂组合物
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AU2005274574B2 (en) * 2004-08-18 2011-03-17 Ace Aps Cosmetic and pharmaceutical compositions comprising ACE inhibitors and/or angiotensin II receptor antagonists
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CN101119730A (zh) * 2005-02-14 2008-02-06 大正制药株式会社 软膏剂
JPWO2006098353A1 (ja) * 2005-03-15 2008-08-28 協和醗酵工業株式会社 外用剤
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CN102176913B (zh) * 2008-10-08 2014-08-13 高田制药株式会社 外用的他克莫司制剂
JP2010132607A (ja) * 2008-12-05 2010-06-17 Taisho Pharm Ind Ltd アトピー性皮膚炎治療用軟膏剤
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CN102885761B (zh) * 2012-09-24 2015-08-05 浙江万晟药业有限公司 一种制备他克莫司软膏的方法
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JP6932180B2 (ja) 2016-04-04 2021-09-08 エムシー2・セラピューティクス・リミテッドMC2 Therapeutics Limited タクロリムスを含む局所組成物
CN105769752B (zh) * 2016-04-08 2018-12-11 湖北人福成田药业有限公司 制备他克莫司软膏的方法及他克莫司软膏
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Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2149635C1 (ru) * 1998-02-27 2000-05-27 Пермская государственная медицинская академия Способ лечения аллергических дерматитов
RU2183113C1 (ru) * 2001-06-28 2002-06-10 Новицкий Юрий Алексеевич Средство-гидросульфат графита и способ лечения больных с доброкачественными и злокачественными опухолями кожи (варианты)
RU2231359C1 (ru) * 2002-12-11 2004-06-27 Государственное образовательное учреждение высшего профессионального образования Московская медицинская академия им. И.М.Сеченова Способ лечения язвенных форм ангиитов кожи
RU2414220C2 (ru) * 2005-10-05 2011-03-20 Мицубиси Танабе Фарма Корпорейшн Средство для лечения дерматита
RU2538680C2 (ru) * 2013-03-12 2015-01-10 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Фармацевтическая композиция для лечения атопического дерматита и способ ее получения
RU2553600C2 (ru) * 2013-05-16 2015-06-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Фармацевтическая композиция для лечения заболеваний кожи

Also Published As

Publication number Publication date
JP2526752B2 (ja) 1996-08-21
ATE150304T1 (de) 1997-04-15
DK0474126T3 (cg-RX-API-DMAC7.html) 1997-04-07
PT98862A (pt) 1992-08-31
CA2050623C (en) 2002-02-05
AU656145B2 (en) 1995-01-27
ZA916983B (en) 1992-05-27
IE913085A1 (en) 1992-03-11
HUT59002A (en) 1992-04-28
DE69125230D1 (de) 1997-04-24
JPH0517481A (ja) 1993-01-26
PT98862B (pt) 1999-02-26
KR100194240B1 (ko) 1999-06-15
DE69125230T2 (de) 1997-07-10
CA2050623A1 (en) 1992-03-05
GR3022883T3 (en) 1997-06-30
CN1059468A (zh) 1992-03-18
KR920005987A (ko) 1992-04-27
PH31282A (en) 1998-07-06
SG46547A1 (en) 1998-02-20
EP0474126B1 (en) 1997-03-19
HU211470A9 (en) 1995-11-28
HK1000006A1 (en) 1997-10-03
EP0474126A1 (en) 1992-03-11
ES2099112T3 (es) 1997-05-16
US5385907A (en) 1995-01-31
AU8351591A (en) 1992-03-12
CN1069193C (zh) 2001-08-08

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