RU2020123665A - Преимущественные режимы дозирования g1т38 - Google Patents
Преимущественные режимы дозирования g1т38 Download PDFInfo
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- RU2020123665A RU2020123665A RU2020123665A RU2020123665A RU2020123665A RU 2020123665 A RU2020123665 A RU 2020123665A RU 2020123665 A RU2020123665 A RU 2020123665A RU 2020123665 A RU2020123665 A RU 2020123665A RU 2020123665 A RU2020123665 A RU 2020123665A
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- 238000000034 method Methods 0.000 claims 17
- 239000003814 drug Substances 0.000 claims 14
- 229940124597 therapeutic agent Drugs 0.000 claims 14
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- 150000003839 salts Chemical class 0.000 claims 8
- 230000035772 mutation Effects 0.000 claims 6
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- 150000001875 compounds Chemical class 0.000 claims 4
- -1 elrotinib Chemical compound 0.000 claims 4
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- PDGKHKMBHVFCMG-UHFFFAOYSA-N 2-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]spiro[7,8-dihydropyrazino[5,6]pyrrolo[1,2-d]pyrimidine-9,1'-cyclohexane]-6-one Chemical compound C1CN(C)CCN1C(C=N1)=CC=C1NC1=NC=C(C=C2N3C4(CCCCC4)CNC2=O)C3=N1 PDGKHKMBHVFCMG-UHFFFAOYSA-N 0.000 claims 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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| AU2024205055A1 (en) | 2024-08-15 |
| KR20200108867A (ko) | 2020-09-21 |
| CO2020008825A2 (es) | 2020-07-31 |
| MX2020007312A (es) | 2021-01-08 |
| NZ765617A (en) | 2025-10-31 |
| SG11202005937QA (en) | 2020-07-29 |
| CN111837146B (zh) | 2024-10-15 |
| AU2019205821A1 (en) | 2020-07-09 |
| PE20210121A1 (es) | 2021-01-19 |
| PH12020551050A1 (en) | 2021-08-23 |
| US11357779B2 (en) | 2022-06-14 |
| US20230149406A1 (en) | 2023-05-18 |
| BR112020013915A2 (pt) | 2020-12-01 |
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