RS57331B1 - Inhibitori demetilaze za lsd1 zasnovani na arilciklopropilaminu i njihova medicinska upotreba - Google Patents

Inhibitori demetilaze za lsd1 zasnovani na arilciklopropilaminu i njihova medicinska upotreba

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Publication number
RS57331B1
RS57331B1 RS20180684A RSP20180684A RS57331B1 RS 57331 B1 RS57331 B1 RS 57331B1 RS 20180684 A RS20180684 A RS 20180684A RS P20180684 A RSP20180684 A RS P20180684A RS 57331 B1 RS57331 B1 RS 57331B1
Authority
RS
Serbia
Prior art keywords
arylcyclopropylamine
lsd1
medical use
demethylase inhibitors
based demethylase
Prior art date
Application number
RS20180684A
Other languages
English (en)
Inventor
Muñoz Alberto Ortega
Matthew Colin Thor Fyfe
Pedemonte Marc Martinell
FERNANDEZ DE LA CUESTA Iñigo TIRAPU
Maria De Los Ángeles Estiarte-Martínez
Original Assignee
Oryzon Genomics Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oryzon Genomics Sa filed Critical Oryzon Genomics Sa
Publication of RS57331B1 publication Critical patent/RS57331B1/sr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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