PT2336132E - Derivado de morfolinopurina - Google Patents

Derivado de morfolinopurina Download PDF

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Publication number
PT2336132E
PT2336132E PT98205792T PT09820579T PT2336132E PT 2336132 E PT2336132 E PT 2336132E PT 98205792 T PT98205792 T PT 98205792T PT 09820579 T PT09820579 T PT 09820579T PT 2336132 E PT2336132 E PT 2336132E
Authority
PT
Portugal
Prior art keywords
morpholinopurine
derivative
morpholinopurine derivative
Prior art date
Application number
PT98205792T
Other languages
English (en)
Portuguese (pt)
Inventor
Takashi Odagiri
Kiyoshi Nakayama
Masaki Setoguchi
Yuichi Tominaga
Masanori Saitou
Kazuyuki Sugita
Original Assignee
Daiichi Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co Ltd filed Critical Daiichi Sankyo Co Ltd
Publication of PT2336132E publication Critical patent/PT2336132E/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT98205792T 2008-10-14 2009-10-13 Derivado de morfolinopurina PT2336132E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2008264797 2008-10-14
JP2009121690 2009-05-20

Publications (1)

Publication Number Publication Date
PT2336132E true PT2336132E (pt) 2014-04-02

Family

ID=42106564

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98205792T PT2336132E (pt) 2008-10-14 2009-10-13 Derivado de morfolinopurina

Country Status (21)

Country Link
US (2) US8097622B2 (cg-RX-API-DMAC10.html)
EP (1) EP2336132B1 (cg-RX-API-DMAC10.html)
JP (1) JP5090423B2 (cg-RX-API-DMAC10.html)
KR (1) KR101614976B1 (cg-RX-API-DMAC10.html)
CN (1) CN102245607B (cg-RX-API-DMAC10.html)
AU (1) AU2009304789B2 (cg-RX-API-DMAC10.html)
BR (1) BRPI0920199A2 (cg-RX-API-DMAC10.html)
CA (1) CA2740471C (cg-RX-API-DMAC10.html)
CO (1) CO6362009A2 (cg-RX-API-DMAC10.html)
DK (1) DK2336132T3 (cg-RX-API-DMAC10.html)
ES (1) ES2452541T3 (cg-RX-API-DMAC10.html)
IL (1) IL212278A (cg-RX-API-DMAC10.html)
MX (1) MX2011003490A (cg-RX-API-DMAC10.html)
MY (1) MY156456A (cg-RX-API-DMAC10.html)
NZ (1) NZ592761A (cg-RX-API-DMAC10.html)
PL (1) PL2336132T3 (cg-RX-API-DMAC10.html)
PT (1) PT2336132E (cg-RX-API-DMAC10.html)
RU (1) RU2490269C2 (cg-RX-API-DMAC10.html)
TW (1) TWI378933B (cg-RX-API-DMAC10.html)
WO (1) WO2010044401A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201102449B (cg-RX-API-DMAC10.html)

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TWI837231B (zh) 2018-11-29 2024-04-01 日商第一三共股份有限公司 含有ｅｚｈ１／２雙重抑制劑之醫藥組合及其用途
CN113368114B (zh) * 2020-03-10 2022-04-22 四川大学 一种吗啉嘧啶类化合物的抗肿瘤应用
JP2024511996A (ja) * 2021-03-17 2024-03-18 タンゴ セラピューティクス， インコーポレイテッド 抗がん剤としてのプリン誘導体

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Also Published As

Publication number Publication date
PL2336132T3 (pl) 2014-06-30
RU2011119525A (ru) 2012-11-27
CN102245607A (zh) 2011-11-16
CA2740471A1 (en) 2010-04-22
IL212278A (en) 2016-07-31
DK2336132T3 (da) 2014-04-07
JP5090423B2 (ja) 2012-12-05
RU2490269C2 (ru) 2013-08-20
NZ592761A (en) 2012-05-25
US20100130492A1 (en) 2010-05-27
JP2011001339A (ja) 2011-01-06
CA2740471C (en) 2013-09-17
MY156456A (en) 2016-02-26
EP2336132B1 (en) 2014-01-01
US20120071476A1 (en) 2012-03-22
ES2452541T3 (es) 2014-04-01
US8097622B2 (en) 2012-01-17
BRPI0920199A2 (pt) 2019-09-24
WO2010044401A1 (ja) 2010-04-22
EP2336132A1 (en) 2011-06-22
CO6362009A2 (es) 2012-01-20
TW201018690A (en) 2010-05-16
CN102245607B (zh) 2014-07-02
KR20110067038A (ko) 2011-06-20
KR101614976B1 (ko) 2016-04-22
ZA201102449B (en) 2011-12-28
AU2009304789A1 (en) 2010-04-22
MX2011003490A (es) 2011-04-21
HK1158189A1 (en) 2012-07-13
EP2336132A4 (en) 2012-03-21
IL212278A0 (en) 2011-06-30
AU2009304789B2 (en) 2012-04-05
TWI378933B (en) 2012-12-11
US8309546B2 (en) 2012-11-13

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