PT1357111E - Derivados de 2-piridona com afinidade para receptores de canabinóides do tipo 2 - Google Patents

Derivados de 2-piridona com afinidade para receptores de canabinóides do tipo 2 Download PDF

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Publication number
PT1357111E
PT1357111E PT01272859T PT01272859T PT1357111E PT 1357111 E PT1357111 E PT 1357111E PT 01272859 T PT01272859 T PT 01272859T PT 01272859 T PT01272859 T PT 01272859T PT 1357111 E PT1357111 E PT 1357111E
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Prior art keywords
receptor
affinity
cannabinoid type
alkyl
pyridone derivatives
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PT01272859T
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English (en)
Inventor
Kohji Hanasaki
Yukio Tada
Yasuyoshi Iso
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Shionogi & Co
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Publication of PT1357111E publication Critical patent/PT1357111E/pt

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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PT01272859T 2000-12-28 2001-12-26 Derivados de 2-piridona com afinidade para receptores de canabinóides do tipo 2 PT1357111E (pt)

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CN100575345C (zh) 2009-12-30
US20100081686A1 (en) 2010-04-01
JPWO2002053543A1 (ja) 2004-05-13
KR20060033816A (ko) 2006-04-19
CN1492856A (zh) 2004-04-28
ES2330719T3 (es) 2009-12-15
CA2433158C (en) 2011-05-10
DE60139506D1 (de) 2009-09-17
WO2002053543A1 (fr) 2002-07-11
JP4137636B2 (ja) 2008-08-20
ATE438624T1 (de) 2009-08-15
US20040082619A1 (en) 2004-04-29
US20060052411A1 (en) 2006-03-09
EP1357111A1 (en) 2003-10-29
US8088924B2 (en) 2012-01-03
US7652141B2 (en) 2010-01-26
EP1357111B1 (en) 2009-08-05
EP1357111A4 (en) 2005-10-05
JP2008169217A (ja) 2008-07-24
CY1109514T1 (el) 2014-08-13
BR0116539A (pt) 2003-09-23
KR100828982B1 (ko) 2008-05-14
TWI287004B (en) 2007-09-21
CA2433158A1 (en) 2002-07-11
US6977266B2 (en) 2005-12-20
DK1357111T3 (da) 2009-11-02

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