ATE438624T1 - 2-pyridonderivate mit affinität für den cannabinoid-typ-2-rezeptor - Google Patents

2-pyridonderivate mit affinität für den cannabinoid-typ-2-rezeptor

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Publication number
ATE438624T1
ATE438624T1 AT01272859T AT01272859T ATE438624T1 AT E438624 T1 ATE438624 T1 AT E438624T1 AT 01272859 T AT01272859 T AT 01272859T AT 01272859 T AT01272859 T AT 01272859T AT E438624 T1 ATE438624 T1 AT E438624T1
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Austria
Prior art keywords
receptor
affinity
cannabinoid type
alkyl
pyridone derivatives
Prior art date
Application number
AT01272859T
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English (en)
Inventor
Yukio Tada
Yasuyoshi Iso
Kohji Hanasaki
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Shionogi & Co
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Publication of ATE438624T1 publication Critical patent/ATE438624T1/de

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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AT01272859T 2000-12-28 2001-12-26 2-pyridonderivate mit affinität für den cannabinoid-typ-2-rezeptor ATE438624T1 (de)

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CA2433158C (en) 2011-05-10
EP1357111B1 (de) 2009-08-05
DE60139506D1 (de) 2009-09-17
CA2433158A1 (en) 2002-07-11
TWI287004B (en) 2007-09-21
EP1357111A1 (de) 2003-10-29
KR20030070082A (ko) 2003-08-27
KR20060033816A (ko) 2006-04-19
US7652141B2 (en) 2010-01-26
BR0116539A (pt) 2003-09-23
KR100828982B1 (ko) 2008-05-14
JP4137636B2 (ja) 2008-08-20
EP1357111A4 (de) 2005-10-05
US20060052411A1 (en) 2006-03-09
JPWO2002053543A1 (ja) 2004-05-13
JP2008169217A (ja) 2008-07-24
US20040082619A1 (en) 2004-04-29
CN1492856A (zh) 2004-04-28
PT1357111E (pt) 2009-10-20
US8088924B2 (en) 2012-01-03
CY1109514T1 (el) 2014-08-13
WO2002053543A1 (fr) 2002-07-11
US20100081686A1 (en) 2010-04-01
DK1357111T3 (da) 2009-11-02
ES2330719T3 (es) 2009-12-15
US6977266B2 (en) 2005-12-20
CN100575345C (zh) 2009-12-30

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