PL3333173T3 - Sposoby wytwarzania przeciwwirusowych analogów nukleotydów - Google Patents

Sposoby wytwarzania przeciwwirusowych analogów nukleotydów

Info

Publication number
PL3333173T3
PL3333173T3 PL18153951T PL18153951T PL3333173T3 PL 3333173 T3 PL3333173 T3 PL 3333173T3 PL 18153951 T PL18153951 T PL 18153951T PL 18153951 T PL18153951 T PL 18153951T PL 3333173 T3 PL3333173 T3 PL 3333173T3
Authority
PL
Poland
Prior art keywords
methods
nucleotide analogs
preparing anti
viral nucleotide
viral
Prior art date
Application number
PL18153951T
Other languages
English (en)
Inventor
Denise A. Colby
Andrew Anthony Martins
Benjamin James Roberts
Robert William Scott
Nicole S. White
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47297386&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL3333173(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of PL3333173T3 publication Critical patent/PL3333173T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65616Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6509Six-membered rings
    • C07F9/6512Six-membered rings having the nitrogen atoms in positions 1 and 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL18153951T 2012-10-03 2012-10-03 Sposoby wytwarzania przeciwwirusowych analogów nukleotydów PL3333173T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP12798029.0A EP2764002B1 (en) 2012-10-03 2012-10-03 Methods for preparing anti-viral nucleotide analogs
EP18153951.1A EP3333173B1 (en) 2012-10-03 2012-10-03 Methods for preparing anti-viral nucleotide analogs
PCT/US2012/000441 WO2013052094A2 (en) 2011-10-07 2012-10-03 Methods for preparing anti-viral nucleotide analogs
US201161544950P 2014-04-11 2014-04-11

Publications (1)

Publication Number Publication Date
PL3333173T3 true PL3333173T3 (pl) 2019-12-31

Family

ID=47297386

Family Applications (1)

Application Number Title Priority Date Filing Date
PL18153951T PL3333173T3 (pl) 2012-10-03 2012-10-03 Sposoby wytwarzania przeciwwirusowych analogów nukleotydów

Country Status (25)

Country Link
US (4) US8664386B2 (pl)
EP (2) EP3333173B1 (pl)
JP (2) JP6190372B2 (pl)
KR (3) KR102033802B1 (pl)
CN (4) CN107266498B (pl)
AR (1) AR088109A1 (pl)
AU (3) AU2012319172B2 (pl)
BR (2) BR112014011340A2 (pl)
CA (2) CA3042169C (pl)
CL (1) CL2014000827A1 (pl)
CO (1) CO6940431A2 (pl)
CR (1) CR20140204A (pl)
EA (1) EA027086B1 (pl)
EC (1) ECSP14000074A (pl)
ES (2) ES2746859T3 (pl)
HK (1) HK1255222B (pl)
IL (1) IL231879B (pl)
MX (1) MX353064B (pl)
PE (1) PE20141160A1 (pl)
PL (1) PL3333173T3 (pl)
PT (2) PT3333173T (pl)
SI (1) SI3333173T1 (pl)
TW (4) TWI709567B (pl)
UY (1) UY34361A (pl)
WO (1) WO2013052094A2 (pl)

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CN105399771B (zh) * 2014-07-21 2020-11-24 江苏豪森药业集团有限公司 替诺福韦前药晶型及其制备方法和用途
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EP3333173A1 (en) 2018-06-13
KR20140090170A (ko) 2014-07-16
BR112014011340A2 (pt) 2017-06-13
MX353064B (es) 2017-12-19
AU2016228317B2 (en) 2018-07-19
EP3333173B1 (en) 2019-06-26
SI3333173T1 (sl) 2019-08-30
CO6940431A2 (es) 2014-05-09
PE20141160A1 (es) 2014-09-22
US20150291638A1 (en) 2015-10-15
MX2014003952A (es) 2014-08-01
TWI613211B (zh) 2018-02-01
JP2014530809A (ja) 2014-11-20
EP2764002A2 (en) 2014-08-13
US20160311840A1 (en) 2016-10-27
HK1245798A1 (zh) 2018-08-31
EA027086B1 (ru) 2017-06-30
ES2661705T3 (es) 2018-04-03
AU2012319172A1 (en) 2013-05-16
AU2012319172B2 (en) 2014-06-12
CN103842366B (zh) 2017-06-16
NZ624513A (en) 2016-06-24
CA3042169A1 (en) 2013-04-11
KR102139440B1 (ko) 2020-07-29
US20140128602A1 (en) 2014-05-08
CA3042169C (en) 2021-09-07
AU2014215976B2 (en) 2016-06-30
WO2013052094A3 (en) 2013-06-20
US9346841B2 (en) 2016-05-24
PT2764002T (pt) 2018-05-16
KR20200090975A (ko) 2020-07-29
BR102014008928A2 (pt) 2015-12-08
AU2014215976A1 (en) 2014-09-11
KR102033802B1 (ko) 2019-10-17
CA2850466C (en) 2020-07-28
TWI689513B (zh) 2020-04-01
WO2013052094A2 (en) 2013-04-11
EA201490753A1 (ru) 2014-09-30
TWI557133B (zh) 2016-11-11
CN107266498A (zh) 2017-10-20
TWI709567B (zh) 2020-11-11
KR20190086576A (ko) 2019-07-22
CN117343101A (zh) 2024-01-05
CN103842366A (zh) 2014-06-04
EP2764002B1 (en) 2018-02-28
CA2850466A1 (en) 2013-04-11
CN113264959A (zh) 2021-08-17
US8664386B2 (en) 2014-03-04
TW201331218A (zh) 2013-08-01
HK1255222B (en) 2020-07-17
HK1200834A1 (en) 2015-08-14
UY34361A (es) 2013-05-31
CL2014000827A1 (es) 2014-09-05
PT3333173T (pt) 2019-09-10
IL231879B (en) 2019-11-28
CN107266498B (zh) 2023-10-03
AR088109A1 (es) 2014-05-07
TW201716418A (zh) 2017-05-16
CR20140204A (es) 2014-06-03
ES2746859T3 (es) 2020-03-09
JP2017160228A (ja) 2017-09-14
US9676804B2 (en) 2017-06-13
US20130090473A1 (en) 2013-04-11
ECSP14000074A (es) 2016-01-29
TW201811808A (zh) 2018-04-01
BR102014008928B1 (pt) 2022-05-17
AU2016228317A1 (en) 2016-10-06
TW202003531A (zh) 2020-01-16
US9029534B2 (en) 2015-05-12
JP6190372B2 (ja) 2017-08-30

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