PH24345A - Novel heteroaryl alkanediphosphonic acids and pharmaceutical compositions containing said compounds - Google Patents

Novel heteroaryl alkanediphosphonic acids and pharmaceutical compositions containing said compounds

Info

Publication number
PH24345A
PH24345A PH36100A PH36100A PH24345A PH 24345 A PH24345 A PH 24345A PH 36100 A PH36100 A PH 36100A PH 36100 A PH36100 A PH 36100A PH 24345 A PH24345 A PH 24345A
Authority
PH
Philippines
Prior art keywords
halogen
compounds
substituted
acids
phosphono group
Prior art date
Application number
PH36100A
Other languages
English (en)
Inventor
Knut A Jaeggi
Leo Widler
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4280350&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH24345(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of PH24345A publication Critical patent/PH24345A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
    • C07F9/6539—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/65031—Five-membered rings having the nitrogen atoms in the positions 1 and 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nutrition Science (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Control Of El Displays (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Glass Compositions (AREA)
PH36100A 1986-11-21 1987-11-20 Novel heteroaryl alkanediphosphonic acids and pharmaceutical compositions containing said compounds PH24345A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH466686 1986-11-21

Publications (1)

Publication Number Publication Date
PH24345A true PH24345A (en) 1990-06-13

Family

ID=4280350

Family Applications (1)

Application Number Title Priority Date Filing Date
PH36100A PH24345A (en) 1986-11-21 1987-11-20 Novel heteroaryl alkanediphosphonic acids and pharmaceutical compositions containing said compounds

Country Status (27)

Country Link
US (1) US4939130A (da)
EP (1) EP0275821B1 (da)
JP (1) JP2744238B2 (da)
KR (1) KR960010752B1 (da)
AT (1) ATE72816T1 (da)
AU (1) AU607722B2 (da)
CA (1) CA1338937C (da)
CY (1) CY1827A (da)
DD (1) DD270533A5 (da)
DE (2) DE10199052I1 (da)
DK (1) DK174098B1 (da)
ES (1) ES2038692T4 (da)
FI (1) FI87570C (da)
GR (1) GR3003895T3 (da)
HK (1) HK114894A (da)
HU (1) HU199150B (da)
IE (1) IE59816B1 (da)
IL (1) IL84497A (da)
LU (1) LU90838I2 (da)
MX (1) MX9427A (da)
NL (1) NL300058I2 (da)
NO (2) NO173446C (da)
NZ (1) NZ222610A (da)
PH (1) PH24345A (da)
PT (1) PT86167B (da)
SG (1) SG92194G (da)
ZA (1) ZA878698B (da)

Families Citing this family (149)

* Cited by examiner, † Cited by third party
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US5753634A (en) * 1992-05-29 1998-05-19 The Procter & Gamble Company Quaternary nitrogen containing phosphonate compounds, pharmaceutical compostions, and methods for treating abnormal calcium and phosphate metabolism
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US9795622B2 (en) 2012-05-14 2017-10-24 Antecip Bioventures Ii Llc Neridronic acid for treating pain associated with a joint
US9820999B2 (en) 2012-05-14 2017-11-21 Antecip Bioventures Ii Llc Neridronic acid for treating complex regional pain syndrome
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HUT46330A (en) 1988-10-28
SG92194G (en) 1995-04-28
KR960010752B1 (ko) 1996-08-08
ES2038692T3 (es) 1993-08-01
ZA878698B (en) 1988-05-23
HK114894A (en) 1994-10-27
NO2001015I2 (no) 2004-10-11
FI87570C (fi) 1993-01-25
PT86167B (pt) 1990-08-31
IE873148L (en) 1988-05-21
GR3003895T3 (da) 1993-03-16
DE3776880D1 (de) 1992-04-02
JPS63150291A (ja) 1988-06-22
NO874856L (no) 1988-05-24
JP2744238B2 (ja) 1998-04-28
NL300058I1 (nl) 2001-12-01
EP0275821B1 (de) 1992-02-26
IL84497A0 (en) 1988-04-29
FI875096A7 (fi) 1988-05-22
NO173446B (no) 1993-09-06
MX9427A (es) 1993-12-01
DK609587D0 (da) 1987-11-20
IL84497A (en) 1994-10-21
FI87570B (fi) 1992-10-15
HU199150B (en) 1990-01-29
CA1338937C (en) 1997-02-25
PT86167A (en) 1987-12-01
NO173446C (no) 1993-12-15
DE10199052I1 (de) 2002-01-10
LU90838I2 (fr) 2001-11-19
AU607722B2 (en) 1991-03-14
EP0275821A1 (de) 1988-07-27
AU8145387A (en) 1988-05-26
ATE72816T1 (de) 1992-03-15
DK609587A (da) 1988-05-22
FI875096A0 (fi) 1987-11-18
IE59816B1 (en) 1994-04-06
NO874856D0 (no) 1987-11-20
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NL300058I2 (nl) 2002-02-01
NZ222610A (en) 1990-09-26
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KR880006204A (ko) 1988-07-22
US4939130A (en) 1990-07-03
DK174098B1 (da) 2002-06-17
DD270533A5 (de) 1989-08-02

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