PH12013502016A1 - Macrocyclic compound and methods for its production - Google Patents

Macrocyclic compound and methods for its production

Info

Publication number
PH12013502016A1
PH12013502016A1 PH1/2013/502016A PH12013502016A PH12013502016A1 PH 12013502016 A1 PH12013502016 A1 PH 12013502016A1 PH 12013502016 A PH12013502016 A PH 12013502016A PH 12013502016 A1 PH12013502016 A1 PH 12013502016A1
Authority
PH
Philippines
Prior art keywords
production
methods
macrocyclic compound
compound
macrocyclic
Prior art date
Application number
PH1/2013/502016A
Other languages
English (en)
Inventor
Matthew Alan Gregory
Steven James Moss
Barrie Wilkinson
Original Assignee
Neurovive Pharmaceutical Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1105293.3A external-priority patent/GB201105293D0/en
Priority claimed from GBGB1113629.8A external-priority patent/GB201113629D0/en
Priority claimed from GBGB1202060.8A external-priority patent/GB201202060D0/en
Application filed by Neurovive Pharmaceutical Ab filed Critical Neurovive Pharmaceutical Ab
Publication of PH12013502016A1 publication Critical patent/PH12013502016A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06078Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/061,3-Oxazines; Hydrogenated 1,3-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355Non-condensed oxazines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0808Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
PH1/2013/502016A 2011-03-29 2012-03-29 Macrocyclic compound and methods for its production PH12013502016A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB1105293.3A GB201105293D0 (en) 2011-03-29 2011-03-29 Novel compounds and methods for their production
GBGB1113629.8A GB201113629D0 (en) 2011-08-08 2011-08-08 Novel compounds and methods for their production
GBGB1202060.8A GB201202060D0 (en) 2012-02-07 2012-02-07 Novel compounds and methods for their production
PCT/GB2012/050700 WO2012131371A1 (en) 2011-03-29 2012-03-29 Macrocyclic compound and methods for its production

Publications (1)

Publication Number Publication Date
PH12013502016A1 true PH12013502016A1 (en) 2013-12-16

Family

ID=46001313

Family Applications (2)

Application Number Title Priority Date Filing Date
PH1/2013/502000A PH12013502000B1 (en) 2011-03-29 2012-03-29 Macrocyclic compounds and methods for their production
PH1/2013/502016A PH12013502016A1 (en) 2011-03-29 2012-03-29 Macrocyclic compound and methods for its production

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PH1/2013/502000A PH12013502000B1 (en) 2011-03-29 2012-03-29 Macrocyclic compounds and methods for their production

Country Status (29)

Country Link
US (2) US9090657B2 (enExample)
EP (2) EP2691413B1 (enExample)
JP (2) JP6118792B2 (enExample)
KR (2) KR101911484B1 (enExample)
CN (3) CN107417766A (enExample)
AR (1) AR085724A1 (enExample)
AU (2) AU2012235961B2 (enExample)
BR (2) BR112013024974A2 (enExample)
CA (2) CA2830827C (enExample)
CL (2) CL2013002739A1 (enExample)
CY (2) CY1116318T1 (enExample)
DK (2) DK2691413T3 (enExample)
EA (2) EA023907B1 (enExample)
ES (2) ES2533437T3 (enExample)
HR (2) HRP20150187T1 (enExample)
IL (2) IL228508B (enExample)
JO (1) JO3063B1 (enExample)
MX (2) MX345352B (enExample)
MY (2) MY170637A (enExample)
PH (2) PH12013502000B1 (enExample)
PL (2) PL2691413T3 (enExample)
PT (2) PT2691412E (enExample)
RS (2) RS53963B1 (enExample)
SG (2) SG193569A1 (enExample)
SI (2) SI2691412T1 (enExample)
TW (1) TWI525098B (enExample)
UY (1) UY33993A (enExample)
WO (2) WO2012131371A1 (enExample)
ZA (2) ZA201307149B (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2012008873A (es) 2010-02-09 2012-11-22 Biotica Tech Ltd Compuestos a base de sangliferina.
JO3063B1 (ar) * 2011-03-29 2017-03-15 Neurovive Pharmaceutical Ab مركب مبتكر وطرق لانتاجه
CN103130734A (zh) * 2011-12-01 2013-06-05 上海药明康德新药开发有限公司 一种合成1,2-吗啉盐酸盐的方法
CN105695541B (zh) * 2016-03-10 2019-03-15 苏州华赛生物工程技术有限公司 一种抗生素nvp018中间体的分离纯化方法
KR20180036522A (ko) 2016-09-30 2018-04-09 (주)나노믹스 스틸벤 유도체 및 그 제조 방법
AU2017361856A1 (en) * 2016-11-18 2019-05-23 Neurovive Pharmaceutical Ab Use of sanglifehrin macrocyclic analogues as anticancer compounds
CN112410353B (zh) * 2019-08-23 2023-01-24 上海医药工业研究院 一种fkbS基因、含其的基因工程菌及其制备方法和用途
AU2020379734B2 (en) 2019-11-04 2025-11-20 Revolution Medicines, Inc. Ras inhibitors
CN117683049A (zh) 2020-09-15 2024-03-12 锐新医药公司 作为ras抑制剂以治疗癌症的吲哚衍生物
EP4334325A1 (en) 2021-05-05 2024-03-13 Revolution Medicines, Inc. Ras inhibitors for the treatment of cancer
AR127308A1 (es) 2021-10-08 2024-01-10 Revolution Medicines Inc Inhibidores ras
CN115028681B (zh) * 2022-08-11 2022-11-15 中国科学院微生物研究所 一种降解亲环素a的嵌合体化合物及其制备方法与应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR006514A1 (es) 1995-07-04 1999-09-08 Sandoz Ag Un macrolido, sus usos, un proceso para producirlo, un aislado biologicamente puro capaz de producirlo, y una composicion farmaceutica quelo comprende
US6124453A (en) 1995-07-04 2000-09-26 Novartis Ag Macrolides
US20090221598A1 (en) * 2005-06-17 2009-09-03 Kai Lin Use of Sanglifehrin in HCV
EP2124992A2 (en) 2007-01-04 2009-12-02 Debiopharm S.A. Non-immunosuppressive cyclosporin for treatment of ullrich congenital muscular dystrophy
CN101691575B (zh) * 2008-09-24 2013-06-05 中国科学院上海有机化学研究所 一种萨菲菌素的生物合成基因簇
CN102224242B (zh) 2008-09-24 2014-09-24 中国科学院上海有机化学研究所 新基因簇
WO2011098808A1 (en) * 2010-02-09 2011-08-18 Biotica Technology Limited Sanglifehrin based compounds
MX2012008873A (es) * 2010-02-09 2012-11-22 Biotica Tech Ltd Compuestos a base de sangliferina.
WO2011098805A1 (en) * 2010-02-09 2011-08-18 Biotica Technology Limited Sanglifehrin based compounds
WO2012085553A1 (en) * 2010-12-20 2012-06-28 Biotica Technology Limited Sanglifehrin derivatives and methods for their production
JO3063B1 (ar) * 2011-03-29 2017-03-15 Neurovive Pharmaceutical Ab مركب مبتكر وطرق لانتاجه

Also Published As

Publication number Publication date
WO2012131377A1 (en) 2012-10-04
IL228508B (en) 2018-01-31
AU2012235961A1 (en) 2013-10-10
CL2013002740A1 (es) 2014-07-11
CN103619869A (zh) 2014-03-05
KR20140057481A (ko) 2014-05-13
UY33993A (es) 2012-10-31
MX345351B (es) 2017-01-26
MY170637A (en) 2019-08-21
JP2014510746A (ja) 2014-05-01
HK1189237A1 (en) 2014-05-30
PL2691412T3 (pl) 2015-08-31
AU2012235880A1 (en) 2013-10-17
SI2691412T1 (sl) 2015-05-29
US20120251581A1 (en) 2012-10-04
EP2691413A1 (en) 2014-02-05
CA2830831C (en) 2020-03-10
HRP20150184T1 (hr) 2015-05-08
EA201391396A1 (ru) 2014-02-28
IL228508A0 (en) 2013-12-31
SG193569A1 (en) 2013-11-29
KR20140071958A (ko) 2014-06-12
CN103619869B (zh) 2015-11-25
RS53963B1 (sr) 2015-08-31
AU2012235961B2 (en) 2016-09-01
DK2691413T3 (en) 2015-04-07
CA2830831A1 (en) 2012-10-04
DK2691412T3 (en) 2015-04-07
JP2014514290A (ja) 2014-06-19
MY170618A (en) 2019-08-21
US20140038885A1 (en) 2014-02-06
TW201300398A (zh) 2013-01-01
MX345352B (es) 2017-01-26
EA023907B1 (ru) 2016-07-29
HRP20150187T1 (xx) 2015-06-05
RS53964B1 (sr) 2015-08-31
IL228509B (en) 2018-02-28
SG193568A1 (en) 2013-11-29
PH12013502000A1 (en) 2013-12-02
CL2013002739A1 (es) 2014-07-11
BR112013024965A2 (pt) 2017-04-18
ES2533437T3 (es) 2015-04-10
MX2013011051A (es) 2014-03-13
ES2533438T3 (es) 2015-04-10
AU2012235880B2 (en) 2016-11-17
EP2691412B1 (en) 2014-12-24
JP6118793B2 (ja) 2017-04-26
CY1116186T1 (el) 2017-02-08
EA201391399A1 (ru) 2014-02-28
EA023848B1 (ru) 2016-07-29
CN103635484B (zh) 2017-05-10
HK1189236A1 (en) 2014-05-30
KR101868084B1 (ko) 2018-06-18
JO3063B1 (ar) 2017-03-15
JP6118792B2 (ja) 2017-04-26
AR085724A1 (es) 2013-10-23
PH12013502000B1 (en) 2018-08-10
PT2691413E (pt) 2015-03-25
CN107417766A (zh) 2017-12-01
IL228509A0 (en) 2013-12-31
US9090657B2 (en) 2015-07-28
PL2691413T3 (pl) 2015-05-29
EP2691412A1 (en) 2014-02-05
TWI525098B (zh) 2016-03-11
CA2830827C (en) 2020-03-10
WO2012131371A1 (en) 2012-10-04
SI2691413T1 (sl) 2015-05-29
ZA201307149B (en) 2015-04-29
BR112013024974A2 (pt) 2016-09-06
ZA201307231B (en) 2015-05-27
KR101911484B1 (ko) 2018-10-24
US9139613B2 (en) 2015-09-22
MX2013011043A (es) 2014-04-25
EP2691413B1 (en) 2014-12-24
PT2691412E (pt) 2015-03-25
CY1116318T1 (el) 2017-02-08
CN103635484A (zh) 2014-03-12
CA2830827A1 (en) 2012-10-04

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