PE20121118A1 - Compuestos de haloalquil heteroaril benzamida - Google Patents

Compuestos de haloalquil heteroaril benzamida

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Publication number
PE20121118A1
PE20121118A1 PE2011001963A PE2011001963A PE20121118A1 PE 20121118 A1 PE20121118 A1 PE 20121118A1 PE 2011001963 A PE2011001963 A PE 2011001963A PE 2011001963 A PE2011001963 A PE 2011001963A PE 20121118 A1 PE20121118 A1 PE 20121118A1
Authority
PE
Peru
Prior art keywords
benzamide compounds
haloalkyl heteroaryl
haloalkyl
heteroaryl benzamide
compounds
Prior art date
Application number
PE2011001963A
Other languages
English (en)
Inventor
Jean-Francois Rossignol
J Edward Semple
Original Assignee
Romark Lab Lc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43069021&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20121118(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Romark Lab Lc filed Critical Romark Lab Lc
Publication of PE20121118A1 publication Critical patent/PE20121118A1/es

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/22—Viral peptide or viral protein
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Abstract

REFERIDA A UN COMPUESTO DE FORMULA I, DONDE R1 A R5 SON CADA UNO H, CN, NO2, F, CL, BR, OH, ALQULO, ENTRE OTROS; R6 ES HALOALQUILO, PERHALOALQUILO, HALOALCOXI, PERHALOALCOXI, ENTRE OTROS; W, X, e Y SON CADA UNO S, O, N, NR9, ENTRE OTROS; R9 ES H, F, Cl, ALQUILO, ARILO, HETEROARILO, ENTRE OTROS. SON COMPUESTOS PREFERIDOS: A, B. DICHOS COMPUESTOS SON UTILES EN EL TRATAMIENTO DE INFECCION POR EL VIRUS DE LA HEPATITIS C
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