PE20080342A1 - Inhibidores de proteasa de hiv de 2-(amino-sustituido)-benzotiazol sulfonamida - Google Patents

Inhibidores de proteasa de hiv de 2-(amino-sustituido)-benzotiazol sulfonamida

Info

Publication number
PE20080342A1
PE20080342A1 PE2007000802A PE2007000802A PE20080342A1 PE 20080342 A1 PE20080342 A1 PE 20080342A1 PE 2007000802 A PE2007000802 A PE 2007000802A PE 2007000802 A PE2007000802 A PE 2007000802A PE 20080342 A1 PE20080342 A1 PE 20080342A1
Authority
PE
Peru
Prior art keywords
amino
protease inhibitors
hiv protease
substituted
benzothiazole sulfonamide
Prior art date
Application number
PE2007000802A
Other languages
English (en)
Spanish (es)
Inventor
Kock Herman Augustinus De
Tim Hugo Maria Jonckers
Paul Jozef Gabriel Maria Boonants
Stefaan Julien Last
Inge Dierynck
T Klooster Gerben Albert Van
Judith Eva Baumeister
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of PE20080342A1 publication Critical patent/PE20080342A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PE2007000802A 2006-06-23 2007-06-22 Inhibidores de proteasa de hiv de 2-(amino-sustituido)-benzotiazol sulfonamida PE20080342A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06116003 2006-06-23

Publications (1)

Publication Number Publication Date
PE20080342A1 true PE20080342A1 (es) 2008-04-25

Family

ID=37596252

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2007000802A PE20080342A1 (es) 2006-06-23 2007-06-22 Inhibidores de proteasa de hiv de 2-(amino-sustituido)-benzotiazol sulfonamida

Country Status (31)

Country Link
US (1) US8202887B2 (US20060241273A1-20061026-C00026.png)
EP (1) EP2035432B1 (US20060241273A1-20061026-C00026.png)
JP (1) JP5232776B2 (US20060241273A1-20061026-C00026.png)
KR (1) KR101419320B1 (US20060241273A1-20061026-C00026.png)
CN (1) CN101479275B (US20060241273A1-20061026-C00026.png)
AP (1) AP2069A (US20060241273A1-20061026-C00026.png)
AR (1) AR061619A1 (US20060241273A1-20061026-C00026.png)
AT (1) ATE544769T1 (US20060241273A1-20061026-C00026.png)
AU (1) AU2007262943B2 (US20060241273A1-20061026-C00026.png)
BR (1) BRPI0713487B1 (US20060241273A1-20061026-C00026.png)
CA (1) CA2653233C (US20060241273A1-20061026-C00026.png)
CL (1) CL2007001826A1 (US20060241273A1-20061026-C00026.png)
CY (1) CY1112971T1 (US20060241273A1-20061026-C00026.png)
DK (1) DK2035432T3 (US20060241273A1-20061026-C00026.png)
EA (1) EA016387B1 (US20060241273A1-20061026-C00026.png)
ES (1) ES2381129T3 (US20060241273A1-20061026-C00026.png)
HK (1) HK1125633A1 (US20060241273A1-20061026-C00026.png)
IL (1) IL195381A (US20060241273A1-20061026-C00026.png)
JO (1) JO2841B1 (US20060241273A1-20061026-C00026.png)
MX (1) MX2009000160A (US20060241273A1-20061026-C00026.png)
MY (1) MY146805A (US20060241273A1-20061026-C00026.png)
NZ (1) NZ573286A (US20060241273A1-20061026-C00026.png)
PE (1) PE20080342A1 (US20060241273A1-20061026-C00026.png)
PL (1) PL2035432T3 (US20060241273A1-20061026-C00026.png)
PT (1) PT2035432E (US20060241273A1-20061026-C00026.png)
SI (1) SI2035432T1 (US20060241273A1-20061026-C00026.png)
TW (1) TWI415851B (US20060241273A1-20061026-C00026.png)
UA (1) UA96445C2 (US20060241273A1-20061026-C00026.png)
UY (1) UY30416A1 (US20060241273A1-20061026-C00026.png)
WO (1) WO2007147884A1 (US20060241273A1-20061026-C00026.png)
ZA (1) ZA200810350B (US20060241273A1-20061026-C00026.png)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3090B1 (ar) 2009-12-11 2017-03-15 Janssen Sciences Ireland Uc 5- امينو-4- هيدروكسي-بنتويل اميدات
MX2012015097A (es) 2010-07-02 2013-05-28 Gilead Sciences Inc Derivados de acido naft-2-ilacetico para tratar sida.
TWI458711B (zh) 2010-07-02 2014-11-01 Gilead Sciences Inc 治療性化合物
US9024038B2 (en) 2010-12-27 2015-05-05 Purdue Research Foundation Compunds and methods for treating HIV
MX2013012266A (es) 2011-04-21 2013-11-22 Gilead Sciences Inc Compuestos de benzotiazol y su uso farmaceutico.
WO2013103738A1 (en) 2012-01-04 2013-07-11 Gilead Sciences, Inc. Napthalene acetic acid derivatives against hiv infection
US9376392B2 (en) 2012-01-04 2016-06-28 Gilead Sciences, Inc. 2-(tert-butoxy)-2-(7-methylquinolin-6-yl) acetic acid derivatives for treating AIDS
SG11201401189WA (en) 2012-04-20 2014-09-26 Gilead Sciences Inc Benzothiazol- 6 -yl acetic acid derivatives and their use for treating an hiv infection
US20230218644A1 (en) 2020-04-16 2023-07-13 Som Innovation Biotech, S.A. Compounds for use in the treatment of viral infections by respiratory syndrome-related coronavirus
US12083099B2 (en) 2020-10-28 2024-09-10 Accencio LLC Methods of treating symptoms of coronavirus infection with viral protease inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE343567T1 (de) 2001-02-14 2006-11-15 Tibotec Pharm Ltd Breitspektrum 2-(substituierte-amino)- benzothiazol-sulfonamide hiv protease inhibitoren
AR037797A1 (es) 2001-12-12 2004-12-01 Tibotec Pharm Ltd Combinacion de inhibidores de proteasa dependientes del citocromo p450
EP1545518A1 (en) * 2002-08-02 2005-06-29 Tibotec Pharmaceuticals Ltd. Broadspectrum 2-amino-benzothiazole sulfonamide hiv protease inhibitors
DE602004010291T2 (de) * 2003-09-30 2008-10-09 Tibotec Pharmaceuticals Ltd. Hcv-hemmende sulfonamide

Also Published As

Publication number Publication date
JP5232776B2 (ja) 2013-07-10
JO2841B1 (en) 2014-09-15
CL2007001826A1 (es) 2008-01-18
BRPI0713487A2 (US20060241273A1-20061026-C00026.png) 2012-11-13
BRPI0713487A8 (pt) 2018-01-02
WO2007147884A1 (en) 2007-12-27
CN101479275A (zh) 2009-07-08
EA200970052A1 (ru) 2009-04-28
JP2009541272A (ja) 2009-11-26
AR061619A1 (es) 2008-09-10
DK2035432T3 (da) 2012-05-14
EP2035432A1 (en) 2009-03-18
US20090209583A1 (en) 2009-08-20
PL2035432T3 (pl) 2012-07-31
SI2035432T1 (sl) 2012-06-29
CN101479275B (zh) 2012-03-07
HK1125633A1 (US20060241273A1-20061026-C00026.png) 2009-08-14
IL195381A0 (en) 2009-08-03
PT2035432E (pt) 2012-04-24
MX2009000160A (es) 2009-01-23
AP2069A (en) 2009-12-08
EA016387B1 (ru) 2012-04-30
CA2653233C (en) 2015-09-29
TWI415851B (zh) 2013-11-21
ATE544769T1 (de) 2012-02-15
AP2008004679A0 (en) 2008-12-31
AU2007262943A1 (en) 2007-12-27
CY1112971T1 (el) 2016-04-13
AU2007262943B2 (en) 2012-04-12
KR101419320B1 (ko) 2014-07-14
MY146805A (en) 2012-09-28
IL195381A (en) 2013-01-31
BRPI0713487B1 (pt) 2022-07-26
US8202887B2 (en) 2012-06-19
KR20090024257A (ko) 2009-03-06
CA2653233A1 (en) 2007-12-27
NZ573286A (en) 2011-09-30
ES2381129T3 (es) 2012-05-23
ZA200810350B (en) 2010-05-26
EP2035432B1 (en) 2012-02-08
UA96445C2 (ru) 2011-11-10
TW200817416A (en) 2008-04-16
UY30416A1 (es) 2008-01-31

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