ZA200810350B - 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors - Google Patents

2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors

Info

Publication number
ZA200810350B
ZA200810350B ZA200810350A ZA200810350A ZA200810350B ZA 200810350 B ZA200810350 B ZA 200810350B ZA 200810350 A ZA200810350 A ZA 200810350A ZA 200810350 A ZA200810350 A ZA 200810350A ZA 200810350 B ZA200810350 B ZA 200810350B
Authority
ZA
South Africa
Prior art keywords
amino
substituted
protease inhibitors
hiv protease
benzothiazole sulfonamide
Prior art date
Application number
ZA200810350A
Other languages
English (en)
Inventor
Kock Herman Augustinus De
Tim Hugo Maria Jonckers
Paul Jozef Gabriel Maria Boonants
Stefaan Julien Last
Inge Dierynck
Judith Eva Baumeister
't Klooster Gerben Albert Eleutherius Van
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of ZA200810350B publication Critical patent/ZA200810350B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
ZA200810350A 2006-06-23 2008-12-05 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors ZA200810350B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06116003 2006-06-23

Publications (1)

Publication Number Publication Date
ZA200810350B true ZA200810350B (en) 2010-05-26

Family

ID=37596252

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200810350A ZA200810350B (en) 2006-06-23 2008-12-05 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors

Country Status (31)

Country Link
US (1) US8202887B2 (xx)
EP (1) EP2035432B1 (xx)
JP (1) JP5232776B2 (xx)
KR (1) KR101419320B1 (xx)
CN (1) CN101479275B (xx)
AP (1) AP2069A (xx)
AR (1) AR061619A1 (xx)
AT (1) ATE544769T1 (xx)
AU (1) AU2007262943B2 (xx)
BR (1) BRPI0713487B1 (xx)
CA (1) CA2653233C (xx)
CL (1) CL2007001826A1 (xx)
CY (1) CY1112971T1 (xx)
DK (1) DK2035432T3 (xx)
EA (1) EA016387B1 (xx)
ES (1) ES2381129T3 (xx)
HK (1) HK1125633A1 (xx)
IL (1) IL195381A (xx)
JO (1) JO2841B1 (xx)
MX (1) MX2009000160A (xx)
MY (1) MY146805A (xx)
NZ (1) NZ573286A (xx)
PE (1) PE20080342A1 (xx)
PL (1) PL2035432T3 (xx)
PT (1) PT2035432E (xx)
SI (1) SI2035432T1 (xx)
TW (1) TWI415851B (xx)
UA (1) UA96445C2 (xx)
UY (1) UY30416A1 (xx)
WO (1) WO2007147884A1 (xx)
ZA (1) ZA200810350B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3090B1 (ar) * 2009-12-11 2017-03-15 Janssen Sciences Ireland Uc 5- امينو-4- هيدروكسي-بنتويل اميدات
US9102614B2 (en) 2010-07-02 2015-08-11 Gilead Sciences, Inc. Naphth-2-ylacetic acid derivatives to treat AIDS
AU2011274323B2 (en) 2010-07-02 2015-08-06 Gilead Sciences, Inc. 2 -quinolinyl- acetic acid derivatives as HIV antiviral compounds
US9024038B2 (en) * 2010-12-27 2015-05-05 Purdue Research Foundation Compunds and methods for treating HIV
AP2015008931A0 (en) 2011-04-21 2015-12-31 Gilead Sciences Inc Benzothiazole compounds and their pharmaceutical use
WO2013103738A1 (en) 2012-01-04 2013-07-11 Gilead Sciences, Inc. Napthalene acetic acid derivatives against hiv infection
WO2013103724A1 (en) 2012-01-04 2013-07-11 Gilead Sciences, Inc. 2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids
CA2850881C (en) 2012-04-20 2021-02-16 Gilead Sciences, Inc. Benzothiazol-6-yl acetic acid derivatives and their use for treating an hiv infection
WO2021209563A1 (en) 2020-04-16 2021-10-21 Som Innovation Biotech, S.A. Compounds for use in the treatment of viral infections by respiratory syndrome-related coronavirus

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2275866T3 (es) * 2001-02-14 2007-06-16 Tibotec Pharmaceuticals Ltd. 2-(aminosustituido)-benzotiazol-sulfonamidas de amplio esprecto inhibidoras de la proteasa de vih.
AR037797A1 (es) * 2001-12-12 2004-12-01 Tibotec Pharm Ltd Combinacion de inhibidores de proteasa dependientes del citocromo p450
NZ538488A (en) * 2002-08-02 2007-10-26 Tibotec Pharm Ltd Broadspectrum 2-amino-benzothiazole sulfonamide HIV protease inhibitors
JP2007507469A (ja) * 2003-09-30 2007-03-29 テイボテク・フアーマシユーチカルズ・リミテツド Ｈｃｖ阻害性スルホンアミド

Also Published As

Publication number Publication date
AP2008004679A0 (en) 2008-12-31
IL195381A0 (en) 2009-08-03
CN101479275B (zh) 2012-03-07
KR101419320B1 (ko) 2014-07-14
HK1125633A1 (xx) 2009-08-14
MX2009000160A (es) 2009-01-23
TW200817416A (en) 2008-04-16
WO2007147884A1 (en) 2007-12-27
AU2007262943B2 (en) 2012-04-12
CN101479275A (zh) 2009-07-08
CY1112971T1 (el) 2016-04-13
NZ573286A (en) 2011-09-30
CL2007001826A1 (es) 2008-01-18
AU2007262943A1 (en) 2007-12-27
DK2035432T3 (da) 2012-05-14
AP2069A (en) 2009-12-08
SI2035432T1 (sl) 2012-06-29
EA200970052A1 (ru) 2009-04-28
US8202887B2 (en) 2012-06-19
AR061619A1 (es) 2008-09-10
ATE544769T1 (de) 2012-02-15
ES2381129T3 (es) 2012-05-23
PE20080342A1 (es) 2008-04-25
JP5232776B2 (ja) 2013-07-10
EA016387B1 (ru) 2012-04-30
TWI415851B (zh) 2013-11-21
MY146805A (en) 2012-09-28
BRPI0713487A8 (pt) 2018-01-02
BRPI0713487A2 (xx) 2012-11-13
CA2653233C (en) 2015-09-29
UY30416A1 (es) 2008-01-31
EP2035432A1 (en) 2009-03-18
IL195381A (en) 2013-01-31
PL2035432T3 (pl) 2012-07-31
PT2035432E (pt) 2012-04-24
CA2653233A1 (en) 2007-12-27
UA96445C2 (ru) 2011-11-10
KR20090024257A (ko) 2009-03-06
JP2009541272A (ja) 2009-11-26
JO2841B1 (en) 2014-09-15
BRPI0713487B1 (pt) 2022-07-26
US20090209583A1 (en) 2009-08-20
EP2035432B1 (en) 2012-02-08

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