PE20051168A1 - Benzonitrilos derivados como moduladores de receptores de androgenos - Google Patents

Benzonitrilos derivados como moduladores de receptores de androgenos

Info

Publication number
PE20051168A1
PE20051168A1 PE2005000159A PE2005000159A PE20051168A1 PE 20051168 A1 PE20051168 A1 PE 20051168A1 PE 2005000159 A PE2005000159 A PE 2005000159A PE 2005000159 A PE2005000159 A PE 2005000159A PE 20051168 A1 PE20051168 A1 PE 20051168A1
Authority
PE
Peru
Prior art keywords
haloalkyl
hydroxy
benzonitrile
trifluoromethyl
halogen
Prior art date
Application number
PE2005000159A
Other languages
English (en)
Spanish (es)
Inventor
Lain-Yen Hu
Huangshu Lei
Daniel Yunlong Du
Bruce Allen Lefker
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of PE20051168A1 publication Critical patent/PE20051168A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/49Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/54Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and etherified hydroxy groups bound to the carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/08Antiseborrheics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28Antiandrogens
PE2005000159A 2004-02-13 2005-02-10 Benzonitrilos derivados como moduladores de receptores de androgenos PE20051168A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54473804P 2004-02-13 2004-02-13
US60564704P 2004-08-30 2004-08-30

Publications (1)

Publication Number Publication Date
PE20051168A1 true PE20051168A1 (es) 2006-02-18

Family

ID=34890476

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2005000159A PE20051168A1 (es) 2004-02-13 2005-02-10 Benzonitrilos derivados como moduladores de receptores de androgenos

Country Status (20)

Country Link
US (1) US7576128B2 (US07576128-20090818-C00030.png)
EP (1) EP1716110A1 (US07576128-20090818-C00030.png)
JP (1) JP3997255B2 (US07576128-20090818-C00030.png)
KR (1) KR100783255B1 (US07576128-20090818-C00030.png)
AP (1) AP2006003700A0 (US07576128-20090818-C00030.png)
AR (1) AR047606A1 (US07576128-20090818-C00030.png)
AU (1) AU2005214167B2 (US07576128-20090818-C00030.png)
BR (1) BRPI0507670A (US07576128-20090818-C00030.png)
CA (1) CA2554696C (US07576128-20090818-C00030.png)
CR (1) CR8555A (US07576128-20090818-C00030.png)
EA (1) EA009902B1 (US07576128-20090818-C00030.png)
EC (1) ECSP066761A (US07576128-20090818-C00030.png)
IL (1) IL176935A0 (US07576128-20090818-C00030.png)
MA (1) MA28361A1 (US07576128-20090818-C00030.png)
NO (1) NO20064053L (US07576128-20090818-C00030.png)
PA (1) PA8623501A1 (US07576128-20090818-C00030.png)
PE (1) PE20051168A1 (US07576128-20090818-C00030.png)
TW (1) TW200534842A (US07576128-20090818-C00030.png)
UY (1) UY28746A1 (US07576128-20090818-C00030.png)
WO (1) WO2005080320A1 (US07576128-20090818-C00030.png)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7507860B2 (en) 2004-04-13 2009-03-24 Pfizer Inc. Androgen modulators
WO2005102990A1 (en) 2004-04-22 2005-11-03 Warner-Lambert Company Llc Androgen modulators
BRPI0513020A (pt) 2004-07-08 2008-04-22 Warner Lambert Co moduladores de andrÈgenio, seus usos, composição farmacêutica, formulação farmacêutica tópica e artigo de fabricação
WO2006018732A1 (en) * 2004-08-18 2006-02-23 Warner-Lambert Company Llc Androgen modulators
ES2302229T3 (es) * 2004-08-31 2008-07-01 Warner-Lambert Company Llc Moduladores de androgenos.
TW200724139A (en) 2005-05-05 2007-07-01 Warner Lambert Co Androgen modulators
TW200708499A (en) * 2005-06-22 2007-03-01 Warner Lambert Co Process for producing ethers
WO2007007149A1 (en) * 2005-07-12 2007-01-18 Warner-Lambert Company Llc Androgen modulators
US20090170886A1 (en) * 2005-08-08 2009-07-02 Pfizer Inc Androgen modulators
EP3108879A1 (en) 2015-06-25 2016-12-28 Cassiopea S.p.A. High concentration formulation
US20210292335A1 (en) * 2018-08-07 2021-09-23 Emory University Heterocyclic Flavone Derivatives, Compositions, and Methods Related Thereto

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Also Published As

Publication number Publication date
KR100783255B1 (ko) 2007-12-06
EA009902B1 (ru) 2008-04-28
CA2554696C (en) 2009-06-30
ECSP066761A (es) 2006-11-16
JP3997255B2 (ja) 2007-10-24
KR20060116223A (ko) 2006-11-14
MA28361A1 (fr) 2006-12-01
EA200601267A1 (ru) 2006-12-29
TW200534842A (en) 2005-11-01
US7576128B2 (en) 2009-08-18
US20050182132A1 (en) 2005-08-18
JP2007522199A (ja) 2007-08-09
AP2006003700A0 (en) 2006-08-31
UY28746A1 (es) 2005-09-30
CR8555A (es) 2006-10-17
AU2005214167A1 (en) 2005-09-01
BRPI0507670A (pt) 2007-07-17
AU2005214167B2 (en) 2008-08-07
CA2554696A1 (en) 2005-09-01
NO20064053L (no) 2006-11-08
EP1716110A1 (en) 2006-11-02
IL176935A0 (en) 2006-12-10
AR047606A1 (es) 2006-01-25
WO2005080320A1 (en) 2005-09-01
PA8623501A1 (es) 2005-08-30

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