OA11706A - Calcium (3S) tetrahydro-3-furaranyl (1S,2R)-3-[[(4-aminophenyl)sulfony](isobutyl) amino]-1-benzyl-2-(phosphonooxy)propylcarbamate. - Google Patents

Calcium (3S) tetrahydro-3-furaranyl (1S,2R)-3-[[(4-aminophenyl)sulfony](isobutyl) amino]-1-benzyl-2-(phosphonooxy)propylcarbamate. Download PDF

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Publication number
OA11706A
OA11706A OA1200100016A OA1200100016A OA11706A OA 11706 A OA11706 A OA 11706A OA 1200100016 A OA1200100016 A OA 1200100016A OA 1200100016 A OA1200100016 A OA 1200100016A OA 11706 A OA11706 A OA 11706A
Authority
OA
OAPI
Prior art keywords
compound
formula
preparation
calcium
water
Prior art date
Application number
OA1200100016A
Other languages
English (en)
French (fr)
Inventor
Ian Gordon Armitage
Andrew David Searle
Hardev Singh
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of OA11706A publication Critical patent/OA11706A/fr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • C07F9/65515Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a five-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/665Phosphorus compounds having oxygen as a ring hetero atom, e.g. fosfomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
OA1200100016A 1998-07-18 1999-07-15 Calcium (3S) tetrahydro-3-furaranyl (1S,2R)-3-[[(4-aminophenyl)sulfony](isobutyl) amino]-1-benzyl-2-(phosphonooxy)propylcarbamate. OA11706A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9815567.4A GB9815567D0 (en) 1998-07-18 1998-07-18 Antiviral compound

Publications (1)

Publication Number Publication Date
OA11706A true OA11706A (en) 2005-01-13

Family

ID=10835689

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200100016A OA11706A (en) 1998-07-18 1999-07-15 Calcium (3S) tetrahydro-3-furaranyl (1S,2R)-3-[[(4-aminophenyl)sulfony](isobutyl) amino]-1-benzyl-2-(phosphonooxy)propylcarbamate.

Country Status (47)

Country Link
US (3) US6514953B1 (es)
EP (2) EP1240903A3 (es)
JP (1) JP3437553B2 (es)
KR (1) KR100694721B1 (es)
CN (1) CN1188422C (es)
AP (1) AP2001002039A0 (es)
AR (1) AR019388A1 (es)
AT (1) ATE229964T1 (es)
AU (1) AU766056B2 (es)
BG (1) BG105253A (es)
BR (1) BRPI9912156B8 (es)
CA (1) CA2337857C (es)
CO (1) CO5090836A1 (es)
CZ (1) CZ300447B6 (es)
DE (1) DE69904600T2 (es)
DK (1) DK1098898T3 (es)
DZ (1) DZ2845A1 (es)
EA (1) EA003191B1 (es)
EE (1) EE200100038A (es)
ES (1) ES2189450T3 (es)
GB (1) GB9815567D0 (es)
GC (1) GC0000105A (es)
GE (1) GEP20033030B (es)
GT (1) GT199900111A (es)
HR (1) HRP20010046A2 (es)
HU (1) HU229700B1 (es)
ID (1) ID28070A (es)
IL (1) IL140824A (es)
IS (1) IS5808A (es)
JO (1) JO2114B1 (es)
MA (1) MA26660A1 (es)
MY (1) MY122323A (es)
NO (1) NO329676B1 (es)
NZ (1) NZ509291A (es)
OA (1) OA11706A (es)
PA (1) PA8477801A1 (es)
PE (1) PE20000869A1 (es)
PL (1) PL195736B1 (es)
PT (1) PT1098898E (es)
SK (1) SK285311B6 (es)
SV (1) SV1999000096A (es)
TN (1) TNSN99145A1 (es)
TR (1) TR200100111T2 (es)
TW (1) TWI245770B (es)
WO (1) WO2000004033A1 (es)
YU (1) YU3401A (es)
ZA (1) ZA200100417B (es)

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US7300924B2 (en) 2003-04-25 2007-11-27 Gilead Sciences, Inc. Anti-infective phosphonate analogs
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Also Published As

Publication number Publication date
YU3401A (sh) 2005-06-10
EA200100053A1 (ru) 2001-08-27
TWI245770B (en) 2005-12-21
AU5037999A (en) 2000-02-07
KR20010071952A (ko) 2001-07-31
US20030100537A1 (en) 2003-05-29
CN1324363A (zh) 2001-11-28
PT1098898E (pt) 2003-04-30
NO329676B1 (no) 2010-11-29
NZ509291A (en) 2003-05-30
BRPI9912156B1 (pt) 2016-07-26
EA003191B1 (ru) 2003-02-27
JO2114B1 (en) 2000-05-21
KR100694721B1 (ko) 2007-03-15
JP3437553B2 (ja) 2003-08-18
EP1240903A2 (en) 2002-09-18
PA8477801A1 (es) 2000-05-24
GT199900111A (es) 2001-01-05
ATE229964T1 (de) 2003-01-15
DE69904600T2 (de) 2003-11-13
ES2189450T3 (es) 2003-07-01
US6514953B1 (en) 2003-02-04
DZ2845A1 (fr) 2003-12-01
ID28070A (id) 2001-05-03
BR9912156A (pt) 2001-04-10
US20030096795A1 (en) 2003-05-22
DK1098898T3 (da) 2003-04-07
WO2000004033A1 (en) 2000-01-27
PL195736B1 (pl) 2007-10-31
HK1034261A1 (en) 2001-10-19
HU229700B1 (en) 2014-05-28
AR019388A1 (es) 2002-02-13
EP1240903A3 (en) 2003-02-12
TR200100111T2 (tr) 2002-02-21
IL140824A0 (en) 2002-02-10
EE200100038A (et) 2002-06-17
CN1188422C (zh) 2005-02-09
DE69904600D1 (de) 2003-01-30
HRP20010046A2 (en) 2002-02-28
CZ2001219A3 (cs) 2001-07-11
AP2001002039A0 (en) 2001-03-31
NO20010282D0 (no) 2001-01-17
JP2003521447A (ja) 2003-07-15
SV1999000096A (es) 2000-07-06
BG105253A (en) 2001-12-29
MY122323A (en) 2006-04-29
GB9815567D0 (en) 1998-09-16
IS5808A (is) 2001-01-12
TNSN99145A1 (fr) 2005-11-10
IL140824A (en) 2004-09-27
BRPI9912156B8 (pt) 2021-05-25
HUP0103432A2 (hu) 2002-04-29
HUP0103432A3 (en) 2003-01-28
SK285311B6 (sk) 2006-10-05
PE20000869A1 (es) 2000-09-08
MA26660A1 (fr) 2004-12-20
AU766056B2 (en) 2003-10-09
CA2337857A1 (en) 2000-01-27
CO5090836A1 (es) 2001-10-30
ZA200100417B (en) 2002-02-27
EP1098898B1 (en) 2002-12-18
EP1098898A1 (en) 2001-05-16
GC0000105A (en) 2005-06-29
PL345620A1 (en) 2002-01-02
CA2337857C (en) 2011-01-25
NO20010282L (no) 2001-03-07
SK762001A3 (en) 2001-10-08
GEP20033030B (en) 2003-07-25
CZ300447B6 (cs) 2009-05-20

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