DK1828167T3 - Acrylamidderivater som antibiotiske midler - Google Patents
Acrylamidderivater som antibiotiske midlerInfo
- Publication number
- DK1828167T3 DK1828167T3 DK05858503.5T DK05858503T DK1828167T3 DK 1828167 T3 DK1828167 T3 DK 1828167T3 DK 05858503 T DK05858503 T DK 05858503T DK 1828167 T3 DK1828167 T3 DK 1828167T3
- Authority
- DK
- Denmark
- Prior art keywords
- antibiotic agents
- acrylamide derivatives
- acrylamide
- derivatives
- antibiotic
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
- A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57694504P | 2004-06-04 | 2004-06-04 | |
| PCT/US2005/019805 WO2007053131A2 (en) | 2004-06-04 | 2005-06-06 | Acrylamide derivatives as antibiotic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1828167T3 true DK1828167T3 (da) | 2014-10-20 |
Family
ID=37889654
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK05858503.5T DK1828167T3 (da) | 2004-06-04 | 2005-06-06 | Acrylamidderivater som antibiotiske midler |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8450307B2 (da) |
| EP (2) | EP2848614A3 (da) |
| JP (1) | JP5087406B2 (da) |
| KR (1) | KR101299399B1 (da) |
| CA (1) | CA2568914C (da) |
| CY (1) | CY1115713T1 (da) |
| DK (1) | DK1828167T3 (da) |
| ES (1) | ES2515101T3 (da) |
| PL (1) | PL1828167T3 (da) |
| PT (1) | PT1828167E (da) |
| SI (1) | SI1828167T1 (da) |
| WO (1) | WO2007053131A2 (da) |
Families Citing this family (25)
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| AU773218B2 (en) * | 1999-10-08 | 2004-05-20 | Debiopharm International Sa | Fab I inhibitors |
| DE60230934D1 (de) * | 2001-04-06 | 2009-03-05 | Affinium Pharm Inc | Fab-i-inhibitoren |
| CA2658506C (en) * | 2006-07-20 | 2016-01-26 | Affinium Pharmaceuticals, Inc. | Acrylamide derivatives as fab 1 inhibitors |
| WO2008098374A1 (en) | 2007-02-16 | 2008-08-21 | Affinium Pharmaceuticals, Inc. | Salts, prodrugs and polymorphs of fab i inhibitors |
| CN101965186A (zh) | 2007-11-28 | 2011-02-02 | 塞阔伊亚药品公司 | 抑制细胞色素p450 2d6的化合物和方法 |
| EP2394995B1 (en) | 2009-02-03 | 2014-01-15 | Kumiai Chemical Industry CO., LTD. | Ring-fused 2-pyridone derivatives and herbicides |
| MX2012005759A (es) * | 2009-11-18 | 2012-10-03 | Fab Pharma S A S | Acrilamidas heterociclicas novedosas y su uso como farmacos. |
| EP2560953B1 (en) | 2010-04-21 | 2016-01-06 | Probiodrug AG | Inhibitors of glutaminyl cyclase |
| HUP1000598A2 (en) | 2010-11-05 | 2012-09-28 | Richter Gedeon Nyrt | Indole derivatives |
| AU2011323245B2 (en) | 2010-11-05 | 2016-01-21 | Senomyx, Inc. | Compounds useful as modulators of TRPM8 |
| JP6294822B2 (ja) | 2011-08-10 | 2018-03-14 | ヤンセン・サイエンシズ・アイルランド・ユーシー | 抗菌性ピペリジニル置換３，４−ジヒドロ−１ｈ−［１，８］−ナフチリジノン類 |
| EA038317B1 (ru) | 2011-08-10 | 2021-08-09 | Янссен Сайенсиз Айрлэнд Юси | Антибактериальные 3,4-дигидро-1н-[1,8]нафтиридиноны, замещенные гомопиперидинилом |
| JO3611B1 (ar) * | 2011-08-10 | 2020-08-27 | Janssen Sciences Ireland Uc | سايكلو بنتا (سي (بيرول 4,3 ثاني هيدرو 1 hمستبدله [8,1] نافثيريدينونات مضادة للجراثيم |
| EP2758376A4 (en) * | 2011-09-19 | 2015-04-29 | Vitas Pharma Res Private Ltd | HETEROCYCLIC COMPOUNDS AS INHIBITORS OF FATTY ACID BIOSYNTHESIS FOR BACTERIAL INFECTIONS |
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| AU2013301452B2 (en) | 2012-08-10 | 2017-06-01 | Janssen Sciences Ireland Uc | New antibacterial compounds |
| JP6250667B2 (ja) * | 2012-08-10 | 2017-12-20 | ヤンセン・サイエンシズ・アイルランド・ユーシー | 新しい抗菌化合物 |
| WO2014072930A2 (en) * | 2012-11-09 | 2014-05-15 | Aurigene Discovery Technologies Limited | Fused pyridine derivatives as antibacterial agents |
| BR112018006471B1 (pt) | 2015-10-01 | 2024-02-27 | Senomyx, Inc | Composto, composição, método de modular o membro de melastina do canal potencial do receptor transitório 8 (trpm8), método de modular a sensação de resfrescância de uma composição e método de induzir uma sensação de refrescância em um ser humano ou animal |
| MX2018010254A (es) | 2016-02-26 | 2018-12-19 | Debiopharm Int Sa | Medicamento para el tratamiento de infecciones de pie diabetico. |
| BR112021009106A2 (pt) * | 2018-11-12 | 2021-08-10 | Debiopharm International S.A. | compostos antibióticos, métodos de fabricação dos mesmos, composições farmacêuticas que os contêm e seus usos |
| US10947253B2 (en) | 2019-08-05 | 2021-03-16 | Ankh Life Sciences Limited | Fused polycyclic dimers |
| WO2021243273A1 (en) * | 2020-05-29 | 2021-12-02 | Taxis Pharmaceuticals, Inc. | Bacterial efflux pump inhibitors |
| CN111991385A (zh) * | 2020-08-17 | 2020-11-27 | 暨南大学 | 棕榈油酸在抑制水产病原菌中的应用 |
| WO2022187329A1 (en) * | 2021-03-03 | 2022-09-09 | The Board Of Trustees Of The University Of Illinois | Fabi inhibitors for gram-negative pathogens |
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-
2005
- 2005-06-06 WO PCT/US2005/019805 patent/WO2007053131A2/en active Application Filing
- 2005-06-06 EP EP14179596.3A patent/EP2848614A3/en not_active Withdrawn
- 2005-06-06 SI SI200531900T patent/SI1828167T1/sl unknown
- 2005-06-06 PT PT58585035T patent/PT1828167E/pt unknown
- 2005-06-06 PL PL05858503T patent/PL1828167T3/pl unknown
- 2005-06-06 ES ES05858503.5T patent/ES2515101T3/es active Active
- 2005-06-06 JP JP2007543017A patent/JP5087406B2/ja not_active Expired - Fee Related
- 2005-06-06 EP EP05858503.5A patent/EP1828167B1/en active Active
- 2005-06-06 DK DK05858503.5T patent/DK1828167T3/da active
- 2005-06-06 US US11/628,569 patent/US8450307B2/en active Active
- 2005-06-06 CA CA2568914A patent/CA2568914C/en not_active Expired - Fee Related
- 2005-06-06 KR KR1020077000169A patent/KR101299399B1/ko active IP Right Grant
-
2013
- 2013-04-25 US US13/870,193 patent/US20140107106A1/en not_active Abandoned
-
2014
- 2014-10-31 CY CY20141100905T patent/CY1115713T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007053131A3 (en) | 2007-08-02 |
| EP2848614A3 (en) | 2015-07-29 |
| PT1828167E (pt) | 2014-10-08 |
| US20140107106A1 (en) | 2014-04-17 |
| KR20080016517A (ko) | 2008-02-21 |
| CA2568914A1 (en) | 2005-12-04 |
| EP1828167B1 (en) | 2014-08-06 |
| US8450307B2 (en) | 2013-05-28 |
| PL1828167T3 (pl) | 2015-02-27 |
| US20100093705A1 (en) | 2010-04-15 |
| CA2568914C (en) | 2013-09-24 |
| KR101299399B1 (ko) | 2013-08-22 |
| SI1828167T1 (sl) | 2014-12-31 |
| ES2515101T3 (es) | 2014-10-29 |
| EP1828167A2 (en) | 2007-09-05 |
| JP5087406B2 (ja) | 2012-12-05 |
| CY1115713T1 (el) | 2017-01-25 |
| EP2848614A2 (en) | 2015-03-18 |
| WO2007053131A2 (en) | 2007-05-10 |
| JP2008505194A (ja) | 2008-02-21 |
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