OA10325A - Crystalline N-acetyl neuraminic acid derivatives and processes for their preparation - Google Patents

Crystalline N-acetyl neuraminic acid derivatives and processes for their preparation Download PDF

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Publication number
OA10325A
OA10325A OA60842A OA60842A OA10325A OA 10325 A OA10325 A OA 10325A OA 60842 A OA60842 A OA 60842A OA 60842 A OA60842 A OA 60842A OA 10325 A OA10325 A OA 10325A
Authority
OA
OAPI
Prior art keywords
crystalline form
hydrate
tetradeoxy
acetamido
glycero
Prior art date
Application number
OA60842A
Other languages
English (en)
French (fr)
Inventor
Christopher Williamson
William James White
Vipulkumar Patel
Original Assignee
Biota Scient Management
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Management filed Critical Biota Scient Management
Publication of OA10325A publication Critical patent/OA10325A/fr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
OA60842A 1993-12-17 1996-06-14 Crystalline N-acetyl neuraminic acid derivatives and processes for their preparation OA10325A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB939325841A GB9325841D0 (en) 1993-12-17 1993-12-17 Chemical compounds

Publications (1)

Publication Number Publication Date
OA10325A true OA10325A (en) 1997-10-07

Family

ID=10746778

Family Applications (2)

Application Number Title Priority Date Filing Date
OA60842A OA10325A (en) 1993-12-17 1996-06-14 Crystalline N-acetyl neuraminic acid derivatives and processes for their preparation
OA1200000004A OA11275A (en) 1993-12-17 2000-01-06 Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation.

Family Applications After (1)

Application Number Title Priority Date Filing Date
OA1200000004A OA11275A (en) 1993-12-17 2000-01-06 Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation.

Country Status (44)

Country Link
US (2) US6294572B1 (ko)
EP (1) EP0734382B1 (ko)
JP (1) JP3317972B2 (ko)
KR (1) KR100403256B1 (ko)
CN (2) CN1502621A (ko)
AP (2) AP9600810A0 (ko)
AT (1) ATE199255T1 (ko)
BG (1) BG63338B1 (ko)
BR (2) BR9408340A (ko)
CA (1) CA2177990C (ko)
CO (1) CO4340619A1 (ko)
CZ (1) CZ289234B6 (ko)
DE (1) DE69426726T2 (ko)
DK (1) DK0734382T3 (ko)
EE (1) EE03353B1 (ko)
EG (1) EG20597A (ko)
ES (1) ES2155517T3 (ko)
FI (1) FI120453B (ko)
GB (1) GB9325841D0 (ko)
GR (1) GR3035681T3 (ko)
HK (1) HK1014187A1 (ko)
HR (1) HRP941001B1 (ko)
HU (1) HU221971B1 (ko)
IL (1) IL112011A (ko)
IS (1) IS4240A (ko)
MA (1) MA23396A1 (ko)
MY (1) MY116221A (ko)
NO (1) NO314759B1 (ko)
NZ (1) NZ277789A (ko)
OA (2) OA10325A (ko)
PE (1) PE31095A1 (ko)
PL (1) PL186384B1 (ko)
PT (1) PT734382E (ko)
RO (1) RO114792B1 (ko)
RU (1) RU2134690C1 (ko)
SA (1) SA94150417B1 (ko)
SG (1) SG46669A1 (ko)
SI (1) SI0734382T1 (ko)
SK (1) SK282972B6 (ko)
SV (1) SV1994000076A (ko)
TW (1) TW452577B (ko)
UA (1) UA46723C2 (ko)
WO (1) WO1995016680A1 (ko)
ZA (1) ZA9410003B (ko)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9325841D0 (en) * 1993-12-17 1994-02-23 Glaxo Group Ltd Chemical compounds
US5866601A (en) * 1995-02-27 1999-02-02 Gilead Sciences, Inc. Carbocyclic compounds
HU228450B1 (en) 1995-02-27 2013-03-28 Gilead Sciences Inc Novel selective inhibitors of viral or bacterial neuraminidases
US5763483A (en) * 1995-12-29 1998-06-09 Gilead Sciences, Inc. Carbocyclic compounds
EP0823428B1 (en) * 1996-07-22 2002-01-02 Sankyo Company Limited Neuraminic acid derivatives, their preparation and their medical use
US6340702B1 (en) 1996-07-22 2002-01-22 Sankyo Company, Limited Neuraminic acid derivatives, their preparation and their medical use
US6451766B1 (en) 1996-07-22 2002-09-17 Sankyo Company, Limited Neuraminic acid derivatives, their preparation and their medical use
US5859284A (en) * 1996-08-23 1999-01-12 Gilead Sciences, Inc. Preparation of carbocyclic compounds
US6518438B2 (en) 1996-08-23 2003-02-11 Gilead Sciences, Inc. Preparation of cyclohexene carboxylate derivatives
US5994377A (en) * 1996-10-21 1999-11-30 Gilead Sciences, Inc. Piperidine compounds
US5886213A (en) * 1997-08-22 1999-03-23 Gilead Sciences, Inc. Preparation of carbocyclic compounds
TW477783B (en) * 1997-12-12 2002-03-01 Gilead Sciences Inc Novel compounds useful as neuraminidase inhibitors and pharmaceutical compositions containing same
TWI291462B (en) 2000-04-25 2007-12-21 Daiichi Sankyo Co Ltd Hydrate crystal of neuraminic acid compound
US20080063722A1 (en) * 2006-09-08 2008-03-13 Advanced Inhalation Research, Inc. Composition of a Spray-Dried Powder for Pulmonary Delivery of a Long Acting Neuraminidase Inhibitor (LANI)
EP2792676A4 (en) * 2011-12-16 2015-10-07 Daiichi Sankyo Co Ltd PROCESS FOR PREPARING NEURAMINE ACID DERIVATIVES
CN109232677B (zh) * 2018-10-18 2021-12-28 中国科学院合肥物质科学研究院 一种使n-乙酰神经氨酸水合物转化为n-乙酰神经氨酸的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP249A (en) * 1990-04-24 1993-03-17 Biota Scient Management Pty Ltd Anti-viral compounds.
AU659501B2 (en) * 1991-10-23 1995-05-18 Biota Scientific Management Pty Ltd Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of alpha-D-neuraminic acid
US5639786A (en) 1992-12-04 1997-06-17 Biota Scientific Management, Pty., Ltd. Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of α-D-neuraninic acid
GB9325841D0 (en) * 1993-12-17 1994-02-23 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
PL315055A1 (en) 1996-09-30
CN1142820A (zh) 1997-02-12
RU2134690C1 (ru) 1999-08-20
WO1995016680A1 (en) 1995-06-22
AP541A (en) 1996-10-01
NO314759B1 (no) 2003-05-19
SK282972B6 (sk) 2003-01-09
BG63338B1 (bg) 2001-10-31
GB9325841D0 (en) 1994-02-23
CZ169396A3 (en) 1996-11-13
UA46723C2 (uk) 2002-06-17
CN1132829C (zh) 2003-12-31
BG100709A (bg) 1997-01-31
EP0734382B1 (en) 2001-02-21
NZ277789A (en) 1999-04-29
JP3317972B2 (ja) 2002-08-26
CZ289234B6 (cs) 2001-12-12
HU9601642D0 (en) 1996-08-28
DE69426726T2 (de) 2001-06-21
KR100403256B1 (ko) 2004-04-30
SA94150417B1 (ar) 2005-12-18
EE03353B1 (et) 2001-02-15
ES2155517T3 (es) 2001-05-16
NO962545D0 (no) 1996-06-14
FI962464A (fi) 1996-06-13
US6294572B1 (en) 2001-09-25
NO962545L (no) 1996-06-14
DE69426726D1 (de) 2001-03-29
SI0734382T1 (en) 2001-08-31
FI120453B (fi) 2009-10-30
CA2177990C (en) 2000-04-25
IL112011A0 (en) 1995-03-15
AU689185B2 (en) 1998-03-26
HU221971B1 (hu) 2003-03-28
EG20597A (en) 1999-09-30
IS4240A (is) 1995-06-18
SG46669A1 (en) 1998-02-20
CA2177990A1 (en) 1995-06-22
US20020037865A1 (en) 2002-03-28
TW452577B (en) 2001-09-01
CO4340619A1 (es) 1996-07-30
EP0734382A1 (en) 1996-10-02
BR9408340A (pt) 1997-08-19
AP9600810A0 (en) 1996-07-31
MA23396A1 (fr) 1995-07-01
DK0734382T3 (da) 2001-03-19
HRP941001B1 (en) 2001-06-30
HK1014187A1 (en) 1999-09-24
IL112011A (en) 1998-08-16
PT734382E (pt) 2001-06-29
OA11275A (en) 2002-11-20
ZA9410003B (en) 1995-07-25
PL186384B1 (pl) 2004-01-30
CN1502621A (zh) 2004-06-09
FI962464A0 (fi) 1996-06-13
GR3035681T3 (en) 2001-06-29
RO114792B1 (ro) 1999-07-30
HUT74938A (en) 1997-03-28
HRP941001A2 (en) 1997-06-30
BR1100548KB1 (pt) 2011-11-01
AU1314495A (en) 1995-07-03
ATE199255T1 (de) 2001-03-15
MY116221A (en) 2003-12-31
JPH09506601A (ja) 1997-06-30
SV1994000076A (es) 1995-10-26
AP9400705A0 (en) 1995-01-31
PE31095A1 (es) 1995-10-18
SK78596A3 (en) 1997-03-05

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