NZ545864A - Benzimidazole derivates: preparation and pharmaceutical applications - Google Patents

Benzimidazole derivates: preparation and pharmaceutical applications

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Publication number
NZ545864A
NZ545864A NZ545864A NZ54586404A NZ545864A NZ 545864 A NZ545864 A NZ 545864A NZ 545864 A NZ545864 A NZ 545864A NZ 54586404 A NZ54586404 A NZ 54586404A NZ 545864 A NZ545864 A NZ 545864A
Authority
NZ
New Zealand
Prior art keywords
hydroxy
benzimidazol
acrylamide
propyl
ethyl
Prior art date
Application number
NZ545864A
Other languages
English (en)
Inventor
Dizhong Chen
Hong Yan Song
Eric T Sun
Niefang Yu
Yong Zou
Original Assignee
S Bio Pte Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by S Bio Pte Ltd filed Critical S Bio Pte Ltd
Publication of NZ545864A publication Critical patent/NZ545864A/en

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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US7781595B2 (en) 2010-08-24
US9402829B2 (en) 2016-08-02
US10736881B2 (en) 2020-08-11
KR20070030162A (ko) 2007-03-15
US8551988B2 (en) 2013-10-08
US20170360757A1 (en) 2017-12-21
CA2539766A1 (en) 2005-03-31
JP5042626B2 (ja) 2012-10-03
PT1673349E (pt) 2010-09-28
US20140005194A1 (en) 2014-01-02
US9717713B2 (en) 2017-08-01
TWI349664B (en) 2011-10-01
MY142589A (en) 2010-12-15
US20070043043A1 (en) 2007-02-22
US20150157608A1 (en) 2015-06-11
US10201527B2 (en) 2019-02-12
BRPI0414581B1 (pt) 2020-01-21
ATE472534T1 (de) 2010-07-15
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AU2004274382A1 (en) 2005-03-31
JP2007505942A (ja) 2007-03-15
WO2005028447A1 (en) 2005-03-31
BRPI0414581A (pt) 2006-11-07
KR101127201B1 (ko) 2012-04-12
US9024029B2 (en) 2015-05-05
TW200530195A (en) 2005-09-16
CA2539766C (en) 2013-07-02
US20160279102A1 (en) 2016-09-29
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US20100256138A1 (en) 2010-10-07
AR046411A1 (es) 2005-12-07
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