NO974563L - Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene - Google Patents
Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelseneInfo
- Publication number
- NO974563L NO974563L NO974563A NO974563A NO974563L NO 974563 L NO974563 L NO 974563L NO 974563 A NO974563 A NO 974563A NO 974563 A NO974563 A NO 974563A NO 974563 L NO974563 L NO 974563L
- Authority
- NO
- Norway
- Prior art keywords
- residue
- alkynyl
- cycloalkyl
- alkenyl
- phenyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Nye taxoider med den generelle formel (I): R-CO-O». ? der Z-0 (I) R l5etyr en substituert alkylrest eller en alkenyl-, alkynyl-, cyklo- alkyl-, eventuelt substituert cykloalkenyl-, fenyl- eller hetero- cyklisk, eventuelt arcinatlsk gruppe med 5 eller 6 kjedeledd. Z betyr et hydrogenatcra eller en rest med den generelle fonnel: der Ri betyr en eventuelt substituert benzylgruppe, tlonyl- eller furoyl- gruppe eller en rest Rg-O-CO-, der Rg betyr en alkyl-, alkenyl-, alkynyl-, cykloalkyl-, cykloalkenyl-, blcykloalkyl-, eventuelt substituert fenyl- eller heterocyklylrest, R3 betyr en alkyl-, alkenyl-, alkynyl-, cykloalkyl-, fenyl-, naftyl- eller heterocyklisk, aramtlsU gnippe. De nye forbindelser med den generelle fonr^l (I) der Z betyr en rest med den generelle fonnel (II) har Interes- sante, antltumorale egenskaper.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9503868A FR2732342B1 (fr) | 1995-04-03 | 1995-04-03 | Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent |
| PCT/FR1996/000487 WO1996031493A1 (fr) | 1995-04-03 | 1996-04-01 | Nouveaux taxoïdes, leur preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO974563D0 NO974563D0 (no) | 1997-10-02 |
| NO974563L true NO974563L (no) | 1997-11-24 |
Family
ID=9477663
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO974563A NO974563L (no) | 1995-04-03 | 1997-10-02 | Nye taxoider, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US5959125A (no) |
| EP (1) | EP0821680B1 (no) |
| JP (1) | JPH11504004A (no) |
| KR (1) | KR19980703520A (no) |
| CN (1) | CN1073106C (no) |
| AP (1) | AP784A (no) |
| AR (1) | AR002730A1 (no) |
| AT (1) | ATE195940T1 (no) |
| AU (1) | AU703918B2 (no) |
| BG (1) | BG62964B1 (no) |
| BR (1) | BR9604799A (no) |
| CA (1) | CA2214322C (no) |
| CZ (1) | CZ287430B6 (no) |
| DE (1) | DE69610085T2 (no) |
| DK (1) | DK0821680T3 (no) |
| EA (1) | EA000726B1 (no) |
| ES (1) | ES2151155T3 (no) |
| FR (1) | FR2732342B1 (no) |
| GE (1) | GEP19991872B (no) |
| GR (1) | GR3034203T3 (no) |
| HU (1) | HUP9802042A3 (no) |
| IL (1) | IL117760A (no) |
| MX (1) | MX9707427A (no) |
| NO (1) | NO974563L (no) |
| NZ (1) | NZ305898A (no) |
| PL (1) | PL322581A1 (no) |
| PT (1) | PT821680E (no) |
| RO (1) | RO115879B1 (no) |
| SK (1) | SK282047B6 (no) |
| TW (1) | TW347389B (no) |
| WO (1) | WO1996031493A1 (no) |
| ZA (1) | ZA962633B (no) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6495579B1 (en) | 1996-12-02 | 2002-12-17 | Angiotech Pharmaceuticals, Inc. | Method for treating multiple sclerosis |
| FR2764118B1 (fr) * | 1997-05-30 | 2000-08-04 | Thomson Csf | Transistor bipolaire stabilise avec elements isolants electriques |
| US6156789A (en) * | 1998-03-17 | 2000-12-05 | Rhone-Poulenc Rorer S.A. | Method for treating abnormal cell proliferation in the brain |
| EP1176957A1 (en) * | 1999-05-03 | 2002-02-06 | Aventis Pharma S.A. | Method for treating abnormal cell proliferation in the brain |
| US6649632B2 (en) * | 2000-02-02 | 2003-11-18 | Fsu Research Foundation, Inc. | C10 ester substituted taxanes |
| NZ514407A (en) * | 2000-02-02 | 2004-12-24 | Univ Florida State Res Found | C10 carbamoyloxy substituted taxanes as antitumor agents |
| TR200102855T1 (tr) * | 2000-02-02 | 2002-06-21 | Florida State University Research Foundation, Inc | Antitümör ajanları olarak C10 karbonat ikameli taksanlar. |
| JP2004339475A (ja) * | 2003-02-03 | 2004-12-02 | Merck Patent Gmbh | フッ化物、オキシフッ化物、フルオロ硫化物および／またはオキシフルオロ硫化物に基づく真珠光沢顔料 |
| CA2526278A1 (en) * | 2003-05-20 | 2004-12-02 | Aronex Pharmaceuticals, Inc. | Combination chemotherapy comprising a liposomal platinum complex |
| SV2006002010A (es) * | 2004-02-13 | 2006-08-23 | Univ Florida State Res Found | Taxanos sustituidos con esteres de ciclopentilo en c10 |
| EP1848423A4 (en) * | 2005-02-14 | 2008-12-31 | Univ Florida State Res Found | C10 CYCLOPROPYL ESTER SUBSTITUTED TAXAN COMPOSITIONS |
| EP2276755A4 (en) * | 2008-03-31 | 2011-05-04 | Univ Florida State Res Found | C (10) -ETHYESTER- AND C (10) -CYCLOPROPYLESTER-SUBSTITUTED TAXANES |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE136460T1 (de) * | 1992-07-01 | 1996-04-15 | Bristol Myers Squibb Co | Fluor-taxole mit antitumor-wirkung |
| US5254580A (en) * | 1993-01-19 | 1993-10-19 | Bristol-Myers Squibb Company | 7,8-cyclopropataxanes |
| FR2698871B1 (fr) * | 1992-12-09 | 1995-02-24 | Rhone Poulenc Rorer Sa | Nouveau taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent. |
| IL107950A (en) * | 1992-12-15 | 2001-04-30 | Upjohn Co | b 7, b 8 - Matano - Taxols, their preparation and pharmaceutical preparations against malignant tumors containing them |
-
1995
- 1995-04-03 FR FR9503868A patent/FR2732342B1/fr not_active Expired - Fee Related
-
1996
- 1996-04-01 KR KR1019970706924A patent/KR19980703520A/ko not_active Application Discontinuation
- 1996-04-01 CZ CZ19973109A patent/CZ287430B6/cs not_active IP Right Cessation
- 1996-04-01 JP JP8530026A patent/JPH11504004A/ja not_active Ceased
- 1996-04-01 TW TW085103805A patent/TW347389B/zh active
- 1996-04-01 DE DE69610085T patent/DE69610085T2/de not_active Expired - Fee Related
- 1996-04-01 SK SK1333-97A patent/SK282047B6/sk unknown
- 1996-04-01 DK DK96911009T patent/DK0821680T3/da active
- 1996-04-01 NZ NZ305898A patent/NZ305898A/xx unknown
- 1996-04-01 AP APAP/P/1997/001094A patent/AP784A/en active
- 1996-04-01 CA CA002214322A patent/CA2214322C/fr not_active Expired - Fee Related
- 1996-04-01 IL IL11776096A patent/IL117760A/en not_active IP Right Cessation
- 1996-04-01 MX MX9707427A patent/MX9707427A/es not_active IP Right Cessation
- 1996-04-01 EA EA199700288A patent/EA000726B1/ru not_active IP Right Cessation
- 1996-04-01 GE GEAP19963965A patent/GEP19991872B/en unknown
- 1996-04-01 US US08/930,561 patent/US5959125A/en not_active Expired - Fee Related
- 1996-04-01 WO PCT/FR1996/000487 patent/WO1996031493A1/fr not_active Application Discontinuation
- 1996-04-01 AT AT96911009T patent/ATE195940T1/de not_active IP Right Cessation
- 1996-04-01 RO RO97-01817A patent/RO115879B1/ro unknown
- 1996-04-01 ES ES96911009T patent/ES2151155T3/es not_active Expired - Lifetime
- 1996-04-01 PL PL96322581A patent/PL322581A1/xx unknown
- 1996-04-01 CN CN96192946A patent/CN1073106C/zh not_active Expired - Fee Related
- 1996-04-01 AU AU54028/96A patent/AU703918B2/en not_active Ceased
- 1996-04-01 PT PT96911009T patent/PT821680E/pt unknown
- 1996-04-01 HU HU9802042A patent/HUP9802042A3/hu unknown
- 1996-04-01 EP EP96911009A patent/EP0821680B1/fr not_active Expired - Lifetime
- 1996-04-01 BR BR9604799A patent/BR9604799A/pt not_active Application Discontinuation
- 1996-04-02 ZA ZA962633A patent/ZA962633B/xx unknown
- 1996-04-03 AR ARP960102049A patent/AR002730A1/es not_active Application Discontinuation
-
1997
- 1997-10-02 NO NO974563A patent/NO974563L/no not_active Application Discontinuation
- 1997-10-03 BG BG101940A patent/BG62964B1/bg unknown
-
2000
- 2000-08-31 GR GR20000400100T patent/GR3034203T3/el not_active IP Right Cessation
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |