NO971773D0 - 5-lipoksygenase-inhibitorer - Google Patents

5-lipoksygenase-inhibitorer

Info

Publication number
NO971773D0
NO971773D0 NO971773A NO971773A NO971773D0 NO 971773 D0 NO971773 D0 NO 971773D0 NO 971773 A NO971773 A NO 971773A NO 971773 A NO971773 A NO 971773A NO 971773 D0 NO971773 D0 NO 971773D0
Authority
NO
Norway
Prior art keywords
alkyl
halo
cyano
alkylene
hydroxy
Prior art date
Application number
NO971773A
Other languages
English (en)
Other versions
NO971773L (no
NO314629B1 (no
Inventor
Rodney W Stevens
Takashi Mano
Kazunari Nakao
Yoshiyuki Okumura
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO971773D0 publication Critical patent/NO971773D0/no
Publication of NO971773L publication Critical patent/NO971773L/no
Publication of NO314629B1 publication Critical patent/NO314629B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO19971773A 1994-10-18 1997-04-17 5-lipoksygenase-inhibitorer NO314629B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP9401747 1994-10-18
PCT/IB1995/000408 WO1996011911A1 (en) 1994-10-18 1995-05-29 5-lipoxygenase inhibitors

Publications (3)

Publication Number Publication Date
NO971773D0 true NO971773D0 (no) 1997-04-17
NO971773L NO971773L (no) 1997-06-17
NO314629B1 NO314629B1 (no) 2003-04-22

Family

ID=14098722

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19971773A NO314629B1 (no) 1994-10-18 1997-04-17 5-lipoksygenase-inhibitorer

Country Status (31)

Country Link
EP (1) EP0787127B1 (no)
JP (1) JP3032579B2 (no)
CN (1) CN1093536C (no)
AT (1) ATE198474T1 (no)
AU (1) AU681520B2 (no)
BG (1) BG61768B1 (no)
CA (1) CA2202057C (no)
CO (1) CO4480026A1 (no)
CZ (1) CZ287350B6 (no)
DE (1) DE69519804T2 (no)
DK (1) DK0787127T3 (no)
ES (1) ES2153033T3 (no)
FI (1) FI971632A (no)
GR (1) GR3035471T3 (no)
HU (1) HU221543B (no)
IL (1) IL115581A (no)
LV (1) LV11468B (no)
MY (1) MY114680A (no)
NO (1) NO314629B1 (no)
NZ (1) NZ285163A (no)
PE (1) PE49196A1 (no)
PL (1) PL180104B1 (no)
RU (1) RU2136666C1 (no)
SI (1) SI9500392A (no)
SK (1) SK281577B6 (no)
TR (1) TR199501274A2 (no)
TW (1) TW411339B (no)
UA (1) UA45312C2 (no)
WO (1) WO1996011911A1 (no)
YU (1) YU65995A (no)
ZA (1) ZA958748B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6239285B1 (en) 1998-02-06 2001-05-29 Pfizer Inc Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems
US6194585B1 (en) * 1998-12-22 2001-02-27 Pfizer Inc. Process for preparing 5-lipoxygenase inhibitors
US6346624B1 (en) * 1999-08-31 2002-02-12 Pfizer Inc Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems
US6344563B1 (en) 1999-08-31 2002-02-05 Timothy Norris Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems
SG87145A1 (en) * 1999-08-31 2002-03-19 Pfizer Prod Inc Process for making 5-lipoxygenase inhibitors having varied heterocyclic ring systems
ES2398093T3 (es) * 2000-03-24 2013-03-13 Euro-Celtique S.A. Pirazoles, triazoles y tetrazoles sustituidos con arilo como bloqueantes de los canales de sodio
CA2444735C (en) * 2001-04-20 2012-10-23 Novozymes A/S Lipoxygenase
GB0302094D0 (en) 2003-01-29 2003-02-26 Pharmagene Lab Ltd EP4 receptor antagonists
GB0324269D0 (en) 2003-10-16 2003-11-19 Pharmagene Lab Ltd EP4 receptor antagonists
UA92833C2 (en) 2006-11-27 2010-12-10 Пфайзер Продактс Инк. Pyrazole analogues
EA201000703A1 (ru) * 2007-11-26 2010-12-30 Пфайзер Инк. Производные пиразола в качестве ингибиторов 5-lo
CN104144920A (zh) * 2012-02-28 2014-11-12 皮拉马尔企业有限公司 作为gpr促效剂的苯基烷酸衍生物
HRP20220331T1 (hr) 2018-03-08 2022-05-13 Incyte Corporation Spojevi aminopirazin diola kao inhibitori pi3k-y
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0462830B1 (en) * 1990-06-21 1995-10-18 Zeneca Limited Cyclic ether derivatives
IE913866A1 (en) * 1990-11-28 1992-06-03 Ici Plc Aryl derivatives
EP0505122A1 (en) * 1991-03-21 1992-09-23 Zeneca Limited Alpha, alpha-dialkylbenzyl derivatives
EP0540165A1 (en) * 1991-10-03 1993-05-05 Zeneca Limited Alkanoic acid derivatives
AU685122B2 (en) * 1993-06-14 1998-01-15 Pfizer Inc. Imidazole lipoxygenase inhibitors

Also Published As

Publication number Publication date
TW411339B (en) 2000-11-11
CZ117797A3 (cs) 1998-06-17
RU2136666C1 (ru) 1999-09-10
DK0787127T3 (da) 2001-02-05
SK281577B6 (sk) 2001-05-10
EP0787127A1 (en) 1997-08-06
HUT77363A (hu) 1998-03-30
GR3035471T3 (en) 2001-05-31
FI971632A0 (fi) 1997-04-17
EP0787127B1 (en) 2001-01-03
YU65995A (sh) 1999-06-15
FI971632A (fi) 1997-04-17
BG61768B1 (bg) 1998-05-29
UA45312C2 (uk) 2002-04-15
TR199501274A2 (tr) 1996-06-21
CZ287350B6 (en) 2000-10-11
CA2202057A1 (en) 1996-04-25
NO971773L (no) 1997-06-17
NZ285163A (en) 1998-08-26
AU2417495A (en) 1996-05-06
SK128795A3 (en) 1996-07-03
SI9500392A (en) 1996-08-31
AU681520B2 (en) 1997-08-28
NO314629B1 (no) 2003-04-22
CN1093536C (zh) 2002-10-30
ZA958748B (en) 1997-04-17
LV11468A (lv) 1996-08-20
JP3032579B2 (ja) 2000-04-17
MY114680A (en) 2002-12-31
IL115581A (en) 1999-10-28
HU221543B (hu) 2002-11-28
PE49196A1 (es) 1996-11-21
BG100070A (bg) 1996-05-31
DE69519804T2 (de) 2001-04-19
PL319727A1 (en) 1997-08-18
LV11468B (en) 1996-12-20
ES2153033T3 (es) 2001-02-16
DE69519804D1 (de) 2001-02-08
PL180104B1 (pl) 2000-12-29
CA2202057C (en) 2001-10-09
ATE198474T1 (de) 2001-01-15
CO4480026A1 (es) 1997-07-09
IL115581A0 (en) 1996-01-19
JPH11507322A (ja) 1999-06-29
CN1169722A (zh) 1998-01-07
WO1996011911A1 (en) 1996-04-25

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