NO315424B1 - Substituerte tiofenalkenylkarboksylsyreguanidider, fremgangsmåter for deresfremstilling, deres anvendelse for fremstilling av medikamenteller diagnostikum samt medikament inneholdende forbindelsene - Google Patents

Substituerte tiofenalkenylkarboksylsyreguanidider, fremgangsmåter for deresfremstilling, deres anvendelse for fremstilling av medikamenteller diagnostikum samt medikament inneholdende forbindelsene Download PDF

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Publication number
NO315424B1
NO315424B1 NO19970697A NO970697A NO315424B1 NO 315424 B1 NO315424 B1 NO 315424B1 NO 19970697 A NO19970697 A NO 19970697A NO 970697 A NO970697 A NO 970697A NO 315424 B1 NO315424 B1 NO 315424B1
Authority
NO
Norway
Prior art keywords
compound
preparation
treatment
drug
thiophenyl
Prior art date
Application number
NO19970697A
Other languages
English (en)
Norwegian (no)
Other versions
NO970697L (no
NO970697D0 (no
Inventor
Jan-Robert Schwark
Joachim Brendel
Heinz-Werner Kleemann
Hans-Jochen Lang
Andreas Weichert
Udo Albus
Wolfgang Scholz
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of NO970697D0 publication Critical patent/NO970697D0/no
Publication of NO970697L publication Critical patent/NO970697L/no
Publication of NO315424B1 publication Critical patent/NO315424B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28—Halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/34—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO19970697A 1996-02-15 1997-02-14 Substituerte tiofenalkenylkarboksylsyreguanidider, fremgangsmåter for deresfremstilling, deres anvendelse for fremstilling av medikamenteller diagnostikum samt medikament inneholdende forbindelsene NO315424B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19605610A DE19605610A1 (de) 1996-02-15 1996-02-15 Substituierte Thiophenylalkenylcarbonsäureguanidide, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament

Publications (3)

Publication Number Publication Date
NO970697D0 NO970697D0 (no) 1997-02-14
NO970697L NO970697L (no) 1997-08-18
NO315424B1 true NO315424B1 (no) 2003-09-01

Family

ID=7785491

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19970697A NO315424B1 (no) 1996-02-15 1997-02-14 Substituerte tiofenalkenylkarboksylsyreguanidider, fremgangsmåter for deresfremstilling, deres anvendelse for fremstilling av medikamenteller diagnostikum samt medikament inneholdende forbindelsene

Country Status (29)

Country Link
US (1) US5756535A (enExample)
EP (1) EP0790245B1 (enExample)
JP (1) JP4402747B2 (enExample)
KR (1) KR970061887A (enExample)
AR (1) AR005812A1 (enExample)
AT (1) ATE202096T1 (enExample)
AU (1) AU706554B2 (enExample)
BR (1) BR9700990A (enExample)
CA (1) CA2197628C (enExample)
CZ (1) CZ45597A3 (enExample)
DE (2) DE19605610A1 (enExample)
DK (1) DK0790245T3 (enExample)
ES (1) ES2158383T3 (enExample)
GR (1) GR3036122T3 (enExample)
HR (1) HRP970081B1 (enExample)
HU (1) HUP9700437A3 (enExample)
ID (1) ID15889A (enExample)
IL (1) IL120214A (enExample)
MX (1) MX9701163A (enExample)
NO (1) NO315424B1 (enExample)
NZ (1) NZ314230A (enExample)
PL (1) PL318412A1 (enExample)
PT (1) PT790245E (enExample)
RU (1) RU2193033C2 (enExample)
SI (1) SI0790245T1 (enExample)
SK (1) SK282440B6 (enExample)
TR (1) TR199700109A2 (enExample)
TW (1) TW445261B (enExample)
ZA (1) ZA971260B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19634229A1 (de) * 1996-08-23 1998-02-26 Basf Ag Photostabile UV-A-Filter enthaltende kosmetische Zubereitungen
US6011059A (en) * 1997-12-24 2000-01-04 Bristol-Myers Squibb Company Acyl guanidine sodium/proton exchange inhibitors and method
US6160134A (en) * 1997-12-24 2000-12-12 Bristol-Myers Squibb Co. Process for preparing chiral cyclopropane carboxylic acids and acyl guanidines
AU4360200A (en) 1999-04-23 2000-11-10 Bristol-Myers Squibb Company Bicyclic acyl guanidine sodium/proton exchange inhibitors and method
PL217872B1 (pl) 2001-10-19 2014-08-29 Toyama Chemical Co Ltd Pochodna eteru alkilowego lub jej sól, stanowiąca 1-{3-[2-(1-benzotiofen-5-ylo)etoksy]propylo}-3-azetydynol lub jego sól

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2734904A (en) * 1956-02-14 Xcxnhxc-nh
US4544670A (en) * 1982-08-24 1985-10-01 William H. Rorer, Inc. Method of treating coccidiosis with acyl guanidines
GB9012252D0 (en) * 1990-06-01 1990-07-18 Lilly Industries Ltd Pharmaceutical compounds
TW415937B (en) * 1994-01-25 2000-12-21 Hoechst Ag Phenyl-substituted alkylcarboxylic acid guanidides bearing perfluoroalkyl groups, process for their preparation, their use as a medicament or diagnostic, and medicament containing them
DE4402057A1 (de) * 1994-01-25 1995-08-03 Hoechst Ag Perfluoralkylgruppen tragende phenyl-substituierte Alkylcarbonsäure-guanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
DE4412334A1 (de) * 1994-04-11 1995-10-19 Hoechst Ag Substituierte N-Heteroaroylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
DE4421536A1 (de) * 1994-06-20 1995-12-21 Hoechst Ag Perfluoralkylgruppen tragende phenylsubstituierte Alkenylcarbonsäure-guanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament

Also Published As

Publication number Publication date
TR199700109A2 (tr) 1997-09-21
HUP9700437A3 (en) 2000-03-28
JP4402747B2 (ja) 2010-01-20
SI0790245T1 (en) 2001-08-31
PL318412A1 (en) 1997-08-18
PT790245E (pt) 2001-10-30
SK282440B6 (sk) 2002-02-05
AR005812A1 (es) 1999-07-14
EP0790245B1 (de) 2001-06-13
US5756535A (en) 1998-05-26
JPH09249660A (ja) 1997-09-22
SK21397A3 (en) 1997-09-10
DK0790245T3 (da) 2001-09-03
GR3036122T3 (en) 2001-09-28
ATE202096T1 (de) 2001-06-15
BR9700990A (pt) 1998-09-01
AU1265997A (en) 1997-08-21
EP0790245A1 (de) 1997-08-20
HRP970081B1 (en) 2003-04-30
RU2193033C2 (ru) 2002-11-20
IL120214A (en) 2000-08-31
HU9700437D0 (en) 1997-04-28
NO970697L (no) 1997-08-18
CZ45597A3 (en) 1997-09-17
NZ314230A (en) 1997-12-19
CA2197628A1 (en) 1997-08-16
HUP9700437A2 (hu) 1998-08-28
KR970061887A (ko) 1997-09-12
ID15889A (id) 1997-08-14
MX9701163A (es) 1997-08-30
ZA971260B (en) 1997-08-15
CA2197628C (en) 2006-05-16
IL120214A0 (en) 1997-06-10
HRP970081A2 (en) 1998-04-30
DE19605610A1 (de) 1997-08-21
TW445261B (en) 2001-07-11
DE59703746D1 (de) 2001-07-19
ES2158383T3 (es) 2001-09-01
NO970697D0 (no) 1997-02-14
AU706554B2 (en) 1999-06-17

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