NO314302B1 - Matriksmetalloproteinase-inhibitorer, anvendelse derav samt farmasöytisk blanding - Google Patents

Matriksmetalloproteinase-inhibitorer, anvendelse derav samt farmasöytisk blanding Download PDF

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Publication number
NO314302B1
NO314302B1 NO19994125A NO994125A NO314302B1 NO 314302 B1 NO314302 B1 NO 314302B1 NO 19994125 A NO19994125 A NO 19994125A NO 994125 A NO994125 A NO 994125A NO 314302 B1 NO314302 B1 NO 314302B1
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Prior art keywords
methoxy
piperidine
benzenesulfonyl
carboxylic acid
alkyl
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NO19994125A
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English (en)
Norwegian (no)
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NO994125D0 (no
NO994125L (no
Inventor
Aranapakam Mudumbai Venkatesan
George Theodore Grosu
Jamie Marie Davis
Jannie Lea Baker
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American Cyanamid Co
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Publication of NO994125D0 publication Critical patent/NO994125D0/no
Publication of NO994125L publication Critical patent/NO994125L/no
Publication of NO314302B1 publication Critical patent/NO314302B1/no

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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
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NO19994125A 1997-02-27 1999-08-26 Matriksmetalloproteinase-inhibitorer, anvendelse derav samt farmasöytisk blanding NO314302B1 (no)

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WO1998038163A1 (en) 1998-09-03
EE9900371A (et) 2000-04-17
EE04295B1 (et) 2004-06-15
AU726204B2 (en) 2000-11-02
YU41099A (sh) 2002-06-19
CY2477B1 (en) 2005-06-03
NO994125L (no) 1999-10-26
YU40999A (sh) 2002-06-19
HUP0001463A3 (en) 2001-04-28
IL131257A0 (en) 2001-01-28
ATE256107T1 (de) 2003-12-15
CA2282656A1 (en) 1998-09-03
AU6436898A (en) 1998-09-18
DK0970046T3 (da) 2004-04-13
PL335286A1 (en) 2000-04-10
NZ337298A (en) 2002-11-26
UA58543C2 (uk) 2003-08-15
EA199900768A1 (ru) 2000-08-28
ES2217540T3 (es) 2004-11-01
ES2212274T3 (es) 2004-07-16
ATE263554T1 (de) 2004-04-15
CN1252713A (zh) 2000-05-10
JP2001519777A (ja) 2001-10-23

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