NO310622B1 - Nye cyklodepsipeptidforbindelser avledet av PF1022 og antelmintisk sammensetning omfattende disse - Google Patents

Nye cyklodepsipeptidforbindelser avledet av PF1022 og antelmintisk sammensetning omfattende disse Download PDF

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Publication number
NO310622B1
NO310622B1 NO19981250A NO981250A NO310622B1 NO 310622 B1 NO310622 B1 NO 310622B1 NO 19981250 A NO19981250 A NO 19981250A NO 981250 A NO981250 A NO 981250A NO 310622 B1 NO310622 B1 NO 310622B1
Authority
NO
Norway
Prior art keywords
group
meleu
phlac
lac
alkylamino
Prior art date
Application number
NO19981250A
Other languages
English (en)
Norwegian (no)
Other versions
NO981250L (no
NO981250D0 (no
Inventor
Norbert Mencke
Peter Jeschke
Makoto Ohyama
Yumiko Okada
Yasushi Murai
Osamu Sakanaka
Katsuharu Iinuma
Maki Matsumoto
Masaaki Takahashi
Achim Harder
Gerhard Bonse
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of NO981250D0 publication Critical patent/NO981250D0/no
Publication of NO981250L publication Critical patent/NO981250L/no
Publication of NO310622B1 publication Critical patent/NO310622B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO19981250A 1995-09-22 1998-03-19 Nye cyklodepsipeptidforbindelser avledet av PF1022 og antelmintisk sammensetning omfattende disse NO310622B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP24405195 1995-09-22
PCT/JP1996/002730 WO1997011064A1 (en) 1995-09-22 1996-09-20 Novel cyclic depsipeptide pf1022 derivatives

Publications (3)

Publication Number Publication Date
NO981250D0 NO981250D0 (no) 1998-03-19
NO981250L NO981250L (no) 1998-05-22
NO310622B1 true NO310622B1 (no) 2001-07-30

Family

ID=17113003

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19981250A NO310622B1 (no) 1995-09-22 1998-03-19 Nye cyklodepsipeptidforbindelser avledet av PF1022 og antelmintisk sammensetning omfattende disse

Country Status (18)

Country Link
US (1) US6329338B1 (OSRAM)
EP (1) EP0903347B1 (OSRAM)
KR (1) KR19990063676A (OSRAM)
CN (1) CN1082051C (OSRAM)
AT (1) ATE299871T1 (OSRAM)
AU (1) AU727532B2 (OSRAM)
BR (1) BR9610527A (OSRAM)
CA (1) CA2232668C (OSRAM)
CZ (1) CZ295705B6 (OSRAM)
DE (1) DE69634961T2 (OSRAM)
DK (1) DK0903347T3 (OSRAM)
ES (1) ES2246496T3 (OSRAM)
HU (1) HU228004B1 (OSRAM)
IL (1) IL123776A (OSRAM)
NO (1) NO310622B1 (OSRAM)
NZ (1) NZ318515A (OSRAM)
PL (1) PL186168B1 (OSRAM)
WO (1) WO1997011064A1 (OSRAM)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998005655A1 (en) * 1996-08-07 1998-02-12 Meiji Seika Kaisha, Ltd. Process for producing cyclodepsipeptide compounds and novel cyclodepsipeptide
AU6229898A (en) * 1997-02-19 1998-09-09 Bayer Aktiengesellschaft Derivatives of cyclodepsipeptide, pf1022 substance
DE19811559A1 (de) * 1998-03-17 1999-09-23 Bayer Ag Cyclooctadepsipeptide
US7109018B1 (en) 1999-09-29 2006-09-19 Meiji Seika Kaisha, Ltd. Transformant producing secondary metabolite modified with functional group and novel biosynthesis genes
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
DE10104362A1 (de) * 2001-02-01 2002-08-08 Bayer Ag Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102008022520A1 (de) 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031284A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102008031283A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
CN107835818B (zh) 2015-05-20 2022-04-29 勃林格殷格翰动物保健美国公司 驱虫缩酚酸肽化合物
KR20220003663A (ko) 2015-12-28 2022-01-10 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 뎁시펩티드 화합물
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN111757880A (zh) 2017-11-07 2020-10-09 拜耳动物保健有限责任公司 用于合成环状缩肽的方法
JP7164608B2 (ja) 2017-11-29 2022-11-01 ゾエティス・サービシーズ・エルエルシー 内部寄生性デプシペプチド
EP3790876B1 (en) 2018-05-10 2025-04-30 Zoetis Services LLC Endoparasitic depsipeptides

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH477172A (de) * 1965-05-18 1969-08-31 Agripat Sa Beifuttermittel
DK431083A (da) * 1982-09-22 1984-03-23 Meiji Seika Co Fremgangsmaade til fremstilling af hydroxylaminderivater
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
CA2132199C (en) * 1992-03-17 2000-01-18 Hitoshi Nishiyama Depsipeptide derivative, production thereof and use thereof
JP2873894B2 (ja) * 1992-10-19 1999-03-24 明治製菓株式会社 環状デプシペプチドおよびその製造法
CN1073560C (zh) * 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
JPH07233068A (ja) * 1993-12-27 1995-09-05 Meiji Seika Kaisha Ltd 高コレステロール血症、高脂血症又は動脈硬化症の治療薬

Also Published As

Publication number Publication date
PL326024A1 (en) 1998-08-17
EP0903347B1 (en) 2005-07-20
HUP0001164A3 (en) 2001-04-28
AU727532B2 (en) 2000-12-14
CA2232668C (en) 2011-10-18
CA2232668A1 (en) 1997-03-27
PL186168B1 (pl) 2003-11-28
EP0903347A4 (OSRAM) 1999-03-24
MX9802268A (es) 1998-08-30
NZ318515A (en) 2000-05-26
JP4001381B1 (OSRAM) 2007-10-31
DE69634961T2 (de) 2006-04-20
AU7001996A (en) 1997-04-09
BR9610527A (pt) 1999-12-21
IL123776A0 (en) 1998-10-30
EP0903347A1 (en) 1999-03-24
KR19990063676A (ko) 1999-07-26
CZ85598A3 (cs) 1998-08-12
DK0903347T3 (da) 2005-11-21
CN1201456A (zh) 1998-12-09
CN1082051C (zh) 2002-04-03
DE69634961D1 (de) 2005-08-25
HU228004B1 (en) 2012-08-28
CZ295705B6 (cs) 2005-10-12
IL123776A (en) 2002-09-12
NO981250L (no) 1998-05-22
US6329338B1 (en) 2001-12-11
NO981250D0 (no) 1998-03-19
WO1997011064A1 (en) 1997-03-27
ES2246496T3 (es) 2006-02-16
HUP0001164A2 (hu) 2000-11-28
ATE299871T1 (de) 2005-08-15

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CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: BAYER INTELLECTUAL PROPERTY GMBH, DE

MK1K Patent expired