NO20100596L - Kinolonanaloger og fremgangsmater - Google Patents
Kinolonanaloger og fremgangsmaterInfo
- Publication number
- NO20100596L NO20100596L NO20100596A NO20100596A NO20100596L NO 20100596 L NO20100596 L NO 20100596L NO 20100596 A NO20100596 A NO 20100596A NO 20100596 A NO20100596 A NO 20100596A NO 20100596 L NO20100596 L NO 20100596L
- Authority
- NO
- Norway
- Prior art keywords
- methods
- quinolone analogs
- present
- compounds
- quinolone
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/16—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Epidemiology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US97804207P | 2007-10-05 | 2007-10-05 | |
US3868108P | 2008-03-21 | 2008-03-21 | |
US4593308P | 2008-04-17 | 2008-04-17 | |
PCT/US2008/078859 WO2009046383A1 (en) | 2007-10-05 | 2008-10-03 | Quinolone analogs and methods related thereto |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20100596L true NO20100596L (no) | 2010-06-10 |
Family
ID=40523786
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20100596A NO20100596L (no) | 2007-10-05 | 2010-04-26 | Kinolonanaloger og fremgangsmater |
Country Status (19)
Country | Link |
---|---|
US (2) | US7928100B2 (ja) |
EP (2) | EP3092901B1 (ja) |
JP (2) | JP5824213B2 (ja) |
KR (2) | KR101601332B1 (ja) |
CN (1) | CN101888780B (ja) |
AU (1) | AU2008308485B2 (ja) |
BR (1) | BRPI0817806A2 (ja) |
CA (1) | CA2701630C (ja) |
DK (1) | DK3092901T3 (ja) |
ES (2) | ES2582662T3 (ja) |
HK (1) | HK1150728A1 (ja) |
IL (2) | IL204844A (ja) |
MX (1) | MX2010003685A (ja) |
NO (1) | NO20100596L (ja) |
NZ (1) | NZ584892A (ja) |
PL (2) | PL2214491T3 (ja) |
PT (2) | PT3092901T (ja) |
RU (1) | RU2549895C2 (ja) |
WO (1) | WO2009046383A1 (ja) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008131134A1 (en) * | 2007-04-17 | 2008-10-30 | Cylene Pharmaceuticals, Inc. | Hydrazide compounds and uses thereof |
BRPI0817806A2 (pt) * | 2007-10-05 | 2014-10-07 | Cylene Pharmaceuticals Inc | Análogos de quinolona e métodos relacionados a estes |
WO2011025889A1 (en) | 2009-08-28 | 2011-03-03 | Takeda Pharmaceutical Company Limited | HEXAHYDROOXAZINOPTERINE COMPOUNDS FOR USE AS mTOR INHIBITORS |
WO2011035332A1 (en) | 2009-09-21 | 2011-03-24 | Chemocentryx, Inc. | Pyrrolidinone carboxamide derivatives as chemerin-r ( chemr23 ) modulators |
TW201242971A (en) | 2011-02-25 | 2012-11-01 | Takeda Pharmaceutical | N-substituted oxazinopteridines and oxazinopteridinones |
EP2685976B1 (en) | 2011-03-17 | 2017-12-27 | Tel HaShomer Medical Research Infrastructure and Services Ltd. | Quinolone analogs for treating autoimmune diseases |
GB201206384D0 (en) * | 2012-04-11 | 2012-05-23 | Redx Pharma Ltd | Antibacterial drug derivatives |
CN104177379B (zh) * | 2013-05-22 | 2016-12-28 | 中国科学院上海药物研究所 | 一种喹诺酮类化合物或其立体化学异构体、包含该化合物的药物组合物及其用途 |
CA2925698C (en) | 2013-11-28 | 2021-11-09 | Tel Hashomer Medical Research Infrastructure And Services Ltd. | Rna polymerase i inhibitors and uses thereof |
AU2015255738C1 (en) * | 2014-05-09 | 2017-09-28 | Pimera, Inc. | Novel compositions, uses and methods for making them |
US9758518B2 (en) | 2015-03-04 | 2017-09-12 | Pimera, Inc. | Compositions, uses and methods for making them |
TWI730013B (zh) * | 2015-11-20 | 2021-06-11 | 生華生物科技股份有限公司 | 用於治療癌症的四環喹諾酮類似物組合療法 |
US9957282B2 (en) | 2015-12-14 | 2018-05-01 | Senhwa Biosciences, Inc. | Crystalline forms of quinolone analogs and their salts |
TWI765848B (zh) * | 2015-12-14 | 2022-06-01 | 生華生物科技股份有限公司 | 喹諾酮類似物及其鹽的結晶形式 |
ES2959536T3 (es) * | 2015-12-14 | 2024-02-26 | Senhwa Biosciences Inc | Formas cristalinas de análogos de quinolona y sus sales |
WO2018183540A1 (en) | 2017-03-28 | 2018-10-04 | Pimera, Inc. | Novel crystal forms of a pol1 inhibitor |
US11071727B2 (en) | 2018-01-26 | 2021-07-27 | Northwestern University | Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors |
AU2019227294B2 (en) * | 2018-02-15 | 2023-06-15 | Senhwa Biosciences, Inc. | Quinolone analogs and their salts, compositions, and method for their use |
WO2020051342A1 (en) * | 2018-09-06 | 2020-03-12 | Cornell University | Methods for treating metastatic disease using ribosome biogenesis inhibitor cx 5461 |
TW202115091A (zh) * | 2019-08-14 | 2021-04-16 | 生華生物科技股份有限公司 | 喹啉類似物之結晶型及其鹽類、組合物、及彼等之使用方法 |
TW202114694A (zh) * | 2019-08-14 | 2021-04-16 | 生華生物科技股份有限公司 | 四環化合物及其鹽類、組合物、及彼等之使用方法 |
JP2020189888A (ja) * | 2020-08-28 | 2020-11-26 | センワ バイオサイエンシズ インコーポレイテッド | キノロン類似体及びその塩の結晶形 |
CN114573604B (zh) * | 2020-12-01 | 2024-06-18 | 中国科学院上海药物研究所 | 一类基于喹诺酮的化合物、其制备方法、包含其的药物组合物及其用途 |
MX2023011004A (es) | 2021-03-19 | 2024-01-08 | Trained Therapeutix Discovery Inc | Compuestos para regular la inmunidad entrenada y métodos para usarlos. |
CN114409681A (zh) * | 2022-03-18 | 2022-04-29 | 信义核新(北京)生物科技有限公司 | 用于治疗dna损伤修复缺陷肿瘤的喹诺酮类似物及其应用 |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4559157A (en) | 1983-04-21 | 1985-12-17 | Creative Products Resource Associates, Ltd. | Cosmetic applicator useful for skin moisturizing |
LU84979A1 (fr) * | 1983-08-30 | 1985-04-24 | Oreal | Composition cosmetique ou pharmaceutique sous forme aqueuse ou anhydre dont la phase grasse contient un polyether oligomere et polyethers oligomeres nouveaux |
US4820508A (en) | 1987-06-23 | 1989-04-11 | Neutrogena Corporation | Skin protective composition |
US4992478A (en) | 1988-04-04 | 1991-02-12 | Warner-Lambert Company | Antiinflammatory skin moisturizing composition and method of preparing same |
US4938949A (en) | 1988-09-12 | 1990-07-03 | University Of New York | Treatment of damaged bone marrow and dosage units therefor |
US5703055A (en) * | 1989-03-21 | 1997-12-30 | Wisconsin Alumni Research Foundation | Generation of antibodies through lipid mediated DNA delivery |
EG20543A (en) * | 1992-10-30 | 1999-07-31 | Procter & Gamble | Process for preparing of novel antimicrobial -5- (n-heterosubstituted amino) quinolones |
ATE269848T1 (de) | 1999-04-07 | 2004-07-15 | Univ Virginia | Calciumkanalblocker als antikrebsmittel |
AU2002361493A1 (en) | 2001-12-13 | 2003-06-23 | Wockhardt Limited | New generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
US6900224B2 (en) * | 2002-07-31 | 2005-05-31 | The Procter & Gamble Company | Antimicrobial quinolones, their compositions and uses |
PL1675852T3 (pl) * | 2003-09-22 | 2009-07-31 | Janssen Pharmaceutica Nv | 7-amino-alkilidenylo-heterocykliczne chinolony i naftrydony |
WO2006034113A2 (en) * | 2004-09-17 | 2006-03-30 | Cylene Pharmaceuticals, Inc. | Quinolone analogs as cell proliferation inhibitors |
ES2529046T3 (es) * | 2005-08-05 | 2015-02-16 | Senhwa Biosciences, Inc. | Procedimientos de preparación de análogos de quinolona |
WO2007022474A2 (en) * | 2005-08-19 | 2007-02-22 | Cylene Pharmaceuticals, Inc. | HUMAN RIBOSOMAL DNA(rDNA) AND RIBOSOMAL RNA (rRNA) NUCLEIC ACIDS AND USES THEREOF |
AR057555A1 (es) * | 2005-10-27 | 2007-12-05 | Merck Frosst Canada Ltd | Un inhibidor de fosfodiesterasa-4 4-oxo-1-(3-sustituido fenil-1,4-dihidro-1,8-naftiridin-3-carboxamida y un procedimiento de preparacion del mismo |
WO2007056113A2 (en) * | 2005-11-02 | 2007-05-18 | Cylene Pharmaceuticals, Inc. | Methods for targeting quadruplex sequences |
WO2008060693A2 (en) | 2006-05-17 | 2008-05-22 | Cylene Pharmaceuticals, Inc. | Tetracyclic imidazole analogs |
WO2007146813A2 (en) | 2006-06-08 | 2007-12-21 | Cylene Pharmaceuticals, Inc. | Pyridinone analogs as cell proliferation inhibitors |
US20100305136A1 (en) * | 2006-06-08 | 2010-12-02 | Johnny Yasuo Nagasawa | Quinolone analogs derivatized with sulfonic acid, sulfonate or sulfonamide |
GB0701992D0 (en) | 2007-02-02 | 2007-03-14 | 7Tm Pharma As | Grehlin Receptor Modulators |
WO2008131134A1 (en) * | 2007-04-17 | 2008-10-30 | Cylene Pharmaceuticals, Inc. | Hydrazide compounds and uses thereof |
BRPI0817806A2 (pt) | 2007-10-05 | 2014-10-07 | Cylene Pharmaceuticals Inc | Análogos de quinolona e métodos relacionados a estes |
-
2008
- 2008-10-03 BR BRPI0817806-2A2A patent/BRPI0817806A2/pt not_active IP Right Cessation
- 2008-10-03 MX MX2010003685A patent/MX2010003685A/es not_active Application Discontinuation
- 2008-10-03 CN CN200880119635.6A patent/CN101888780B/zh active Active
- 2008-10-03 CA CA2701630A patent/CA2701630C/en active Active
- 2008-10-03 PL PL08835342.0T patent/PL2214491T3/pl unknown
- 2008-10-03 KR KR1020107009924A patent/KR101601332B1/ko active IP Right Grant
- 2008-10-03 KR KR1020167002742A patent/KR101682867B1/ko active IP Right Grant
- 2008-10-03 ES ES08835342.0T patent/ES2582662T3/es active Active
- 2008-10-03 WO PCT/US2008/078859 patent/WO2009046383A1/en active Application Filing
- 2008-10-03 EP EP16171555.2A patent/EP3092901B1/en active Active
- 2008-10-03 JP JP2010528194A patent/JP5824213B2/ja active Active
- 2008-10-03 PT PT161715552T patent/PT3092901T/pt unknown
- 2008-10-03 EP EP08835342.0A patent/EP2214491B1/en active Active
- 2008-10-03 DK DK16171555.2T patent/DK3092901T3/da active
- 2008-10-03 AU AU2008308485A patent/AU2008308485B2/en active Active
- 2008-10-03 NZ NZ584892A patent/NZ584892A/en unknown
- 2008-10-03 PL PL16171555T patent/PL3092901T3/pl unknown
- 2008-10-03 ES ES16171555T patent/ES2791305T3/es active Active
- 2008-10-03 US US12/245,619 patent/US7928100B2/en active Active
- 2008-10-03 PT PT88353420T patent/PT2214491T/pt unknown
- 2008-10-03 RU RU2010117225/04A patent/RU2549895C2/ru not_active Application Discontinuation
-
2010
- 2010-04-06 IL IL204844A patent/IL204844A/en active IP Right Grant
- 2010-04-26 NO NO20100596A patent/NO20100596L/no not_active Application Discontinuation
-
2011
- 2011-03-09 US US13/043,956 patent/US8853234B2/en active Active
- 2011-05-17 HK HK11104885.7A patent/HK1150728A1/xx unknown
-
2014
- 2014-05-14 JP JP2014100136A patent/JP2014159474A/ja not_active Withdrawn
-
2017
- 2017-01-02 IL IL249906A patent/IL249906B/en active IP Right Grant
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20100596L (no) | Kinolonanaloger og fremgangsmater | |
CY1120935T1 (el) | Νεες συνθεσεις, χρησεις και μεθοδοι για την παρασκευη αυτων | |
CY1122330T1 (el) | Συνθεσεις δισκιων μηλεϊνικης νερατινιμπης | |
CL2014000746A1 (es) | Compuestos derivados de 3-pirimidin-4-il-oxazolidin-2-ona y sus sales, como inhibidores de las proteinas idh mutantes; composicion farmaceutica que los comprende, utiles para el tratamiento de trastornos de la proliferacion celular tal como el cancer. | |
CL2012003415A1 (es) | Compuestos derivados de 2-oxo-piperidina y 1,1-dioxido-tiazina, inhibidores de mdm2; composicion farmaceutica que los comprende; y su uso para el tratamiento del cancer . | |
CO2018000668A2 (es) | Nuevos compuestos bicíclicos como inhibidores duales de atx/ca | |
CO2017011151A2 (es) | Nuevos compuestos bicíclicos como inhibidores de la atx | |
CY1118859T1 (el) | 6-αλκινυλο-πυριδινες ως μιμητες smac | |
CL2012002189A1 (es) | Compuestos derivados de pirrolidina-2-carboxamidas sustituidas; inhibidores de la interaccion mdm2-p53; composicion farmaceutica; y su uso para el tratamiento del cancer, en particular de tumores solidos. | |
CL2014002873A1 (es) | Compuestos derivados de pirimidin-amina o triazin-amina, inhibidores de adn-pk; composicion farmaceutica; y su uso para el tratamiento del cancer. | |
EA200971051A1 (ru) | Ингибиторы p70 s6 киназы | |
BR112012008385A2 (pt) | inibidores de p13 cinase e uso dos mesmos. | |
CO2017011152A2 (es) | Nuevos compuestos bicíclicos como inhibidores duales de atx / ca. | |
MX2015011898A (es) | Compuestos de pirazolo y usos de los mismos. | |
MX2016015565A (es) | Ciertos inhibidores de la proteina quinasa. | |
TR201900274T4 (tr) | Geliştirilmiş adenovirüs formülasyonları. | |
MX351165B (es) | Antagonistas de trpv1. | |
NO20090596L (no) | Antivirale fosfinatforbindelser | |
CL2015001279A1 (es) | Compuestos derivados de piridina, inhibidores del transportador de uratos urat 1; composicion farmaceutica que los comprende; uso para el tratamiento o prevencion de enfermedades tales como gota, hiperuricemia, hipertensión, enfermedades renales, entre otras. | |
CL2008000202A1 (es) | Compuestos derivados de n-aril-acetamida, antagonista trpv1;composicion farmaceutica que los comprende, utiles en el tratamiento del dolor. | |
CL2011002965A1 (es) | Compuestos derivados de piperidinas sustituidas; procedimiento de preparacion; composicion farmaceutica; y uso de dichos compuestos para el tratamiento y/o profilaxis de trastornos cardiovasculares, tromboembolicos y/o tumores. | |
GT201500143A (es) | Composiciones que comprenden vortioxetina y donepezilo campo tecnico | |
TN2018000057A1 (en) | Compounds useful for inhibiting ror-gamma-t. | |
DK3002009T3 (da) | Behandling af imatinib-resistent kronisk myeloid leukæmi, som har mutationen 1457t>c i bcrabl-genet, under anvendelse af forbindelsen bosutinib | |
WO2016141042A3 (en) | Novel compositions, uses and methods for making them |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |