NO20091054L - Benzimidazolderivater anvendelige for behandling av vallinoidreceptor TRPV1 relaterte forstyrrelser - Google Patents

Benzimidazolderivater anvendelige for behandling av vallinoidreceptor TRPV1 relaterte forstyrrelser

Info

Publication number
NO20091054L
NO20091054L NO20091054A NO20091054A NO20091054L NO 20091054 L NO20091054 L NO 20091054L NO 20091054 A NO20091054 A NO 20091054A NO 20091054 A NO20091054 A NO 20091054A NO 20091054 L NO20091054 L NO 20091054L
Authority
NO
Norway
Prior art keywords
treatment
benzimidazole derivatives
related disorders
derivatives useful
receptor trpv1
Prior art date
Application number
NO20091054A
Other languages
English (en)
Norwegian (no)
Inventor
William Brown
Shawn Johnstone
Denis Labrecque
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39033277&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20091054(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20091054L publication Critical patent/NO20091054L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20091054A 2006-08-11 2009-03-09 Benzimidazolderivater anvendelige for behandling av vallinoidreceptor TRPV1 relaterte forstyrrelser NO20091054L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83724906P 2006-08-11 2006-08-11
PCT/SE2007/000720 WO2008018827A1 (en) 2006-08-11 2007-08-10 Benzimidazole derivatives useful in treatment of vallinoid receptor trpv1 related disorders

Publications (1)

Publication Number Publication Date
NO20091054L true NO20091054L (no) 2009-03-09

Family

ID=39033277

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20091054A NO20091054L (no) 2006-08-11 2009-03-09 Benzimidazolderivater anvendelige for behandling av vallinoidreceptor TRPV1 relaterte forstyrrelser

Country Status (25)

Country Link
US (2) US7906654B2 (enExample)
EP (1) EP2051967B1 (enExample)
JP (1) JP5140077B2 (enExample)
KR (1) KR101412881B1 (enExample)
CN (2) CN101792436A (enExample)
AR (1) AR062299A1 (enExample)
AU (1) AU2007282186B2 (enExample)
BR (1) BRPI0715746B8 (enExample)
CA (1) CA2660529C (enExample)
CL (1) CL2007002343A1 (enExample)
CO (1) CO6150176A2 (enExample)
ES (1) ES2533971T3 (enExample)
IL (1) IL196672A0 (enExample)
MX (1) MX2009001496A (enExample)
MY (1) MY147649A (enExample)
NO (1) NO20091054L (enExample)
NZ (1) NZ575416A (enExample)
PE (1) PE20081315A1 (enExample)
RU (1) RU2458055C2 (enExample)
SG (1) SG173360A1 (enExample)
TW (1) TWI433839B (enExample)
UA (1) UA96764C2 (enExample)
UY (1) UY30533A1 (enExample)
WO (1) WO2008018827A1 (enExample)
ZA (1) ZA200900961B (enExample)

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EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
CN101983197B (zh) 2008-04-18 2015-04-22 大熊制药株式会社 新型苯并噁嗪苯并咪唑衍生物、含有该衍生物的药物组合物及其用途
KR101293384B1 (ko) 2010-10-13 2013-08-05 주식회사 대웅제약 신규 피리딜 벤조옥사진 유도체, 이를 포함하는 약학 조성물 및 이의 용도
US8716226B2 (en) 2012-07-18 2014-05-06 Saint Louis University 3,5 phenyl-substituted beta amino acid derivatives as integrin antagonists
IN2015DN00099A (enExample) 2012-07-18 2015-05-29 Univ Saint Louis
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CN107001541B (zh) 2014-12-08 2019-11-26 罗门哈斯公司 聚烯烃添加剂、抗垂挂聚烯烃以及其制备方法
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HK1244806A1 (zh) 2015-12-30 2018-08-17 Saint Louis University 作為過氧乙醯硝酸整聯蛋白拮抗劑的間氮雜環氨基苯甲酸衍生物
EP3908574A4 (en) * 2019-01-08 2022-10-26 Neomed Institute CRYSTALLINE FORMS OF (S)-2-(7-CYANO-1H-BENZIMIDAZOLE-1-YL)-N-{1-[4-(1-CYANO-1-METHYLETHYL)PHENYL]ETHYL}ACETAMIDE
TWI873185B (zh) 2019-09-16 2025-02-21 日商武田藥品工業股份有限公司 唑稠合之嗒-3(2h)-酮衍生物
JP7697974B2 (ja) 2020-05-08 2025-06-24 武田薬品工業株式会社 Ｇｐｒ１３９アゴニストの置換ベンゾトリアジノン代謝物
RU2755206C1 (ru) 2020-05-20 2021-09-14 Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) Средство пролонгированного анальгетического действия и лекарственный препарат на его основе
CN117623972A (zh) * 2022-08-17 2024-03-01 上海慧聚药业有限公司 非离子型造影剂中间体的合成

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TWI433839B (zh) 2006-08-11 2014-04-11 Neomed Inst 新穎的苯并咪唑衍生物290

Also Published As

Publication number Publication date
CN101522637A (zh) 2009-09-02
BRPI0715746B8 (pt) 2021-05-25
US20080221188A1 (en) 2008-09-11
PE20081315A1 (es) 2008-11-08
UA96764C2 (ru) 2011-12-12
UY30533A1 (es) 2008-03-31
CO6150176A2 (es) 2010-04-20
EP2051967A1 (en) 2009-04-29
US20110137045A1 (en) 2011-06-09
BRPI0715746A2 (pt) 2013-07-16
US8093402B2 (en) 2012-01-10
ES2533971T3 (es) 2015-04-16
EP2051967B1 (en) 2014-12-31
CA2660529C (en) 2014-10-21
MX2009001496A (es) 2009-02-18
IL196672A0 (en) 2009-11-18
CA2660529A1 (en) 2008-02-14
RU2009103675A (ru) 2010-09-20
SG173360A1 (en) 2011-08-29
JP2010500345A (ja) 2010-01-07
AU2007282186A1 (en) 2008-02-14
CN101792436A (zh) 2010-08-04
BRPI0715746B1 (pt) 2020-09-24
WO2008018827A1 (en) 2008-02-14
AR062299A1 (es) 2008-10-29
TW200817338A (en) 2008-04-16
NZ575416A (en) 2011-10-28
RU2458055C2 (ru) 2012-08-10
AU2007282186B2 (en) 2011-07-07
MY147649A (en) 2012-12-31
KR20090035701A (ko) 2009-04-10
ZA200900961B (en) 2010-07-28
CL2007002343A1 (es) 2008-04-04
US7906654B2 (en) 2011-03-15
TWI433839B (zh) 2014-04-11
EP2051967A4 (en) 2011-06-29
KR101412881B1 (ko) 2014-06-26
JP5140077B2 (ja) 2013-02-06
WO2008018827A8 (en) 2009-02-19

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